paragraph_index
int64
sec
string
p_has_citation
int64
cites
string
citeids
list
pmid
int64
cited_id
string
sentences
string
all_sent_cites
list
sent_len
int64
sentence_batch_index
int64
sent_has_citation
float64
qc_fail
bool
cited_sentence
string
cites_in_sentence
list
cln_sentence
string
is_cap
bool
is_alpha
bool
ends_wp
bool
cit_qc
bool
lgtm
bool
__index_level_0__
int64
2
DISCUSSION
0
null
null
17,182,632
pmid-15205459|pmid-8390996
Hepatotoxicity was chemistry-, sequence- and design-dependent, as it was only observed with LNA containing ASOs, and the onset occurred at slightly different dose levels for different compounds.
null
194
200
0
false
null
null
Hepatotoxicity was chemistry-, sequence- and design-dependent, as it was only observed with LNA containing ASOs, and the onset occurred at slightly different dose levels for different compounds.
true
true
true
true
true
37
2
DISCUSSION
0
null
null
17,182,632
pmid-15205459|pmid-8390996
The fact that the MOE ASOs in some cases (compare 2a with 2b, and 6 with 7b and 8b) produced similar reductions in target RNA without producing observable toxicity suggest that the toxicity is not secondary to reduction in target gene expression.
null
246
201
0
false
null
null
The fact that the MOE ASOs in some cases (compare 2a with 2b, and 6 with 7b and 8b) produced similar reductions in target RNA without producing observable toxicity suggest that the toxicity is not secondary to reduction in target gene expression.
true
true
true
true
true
37
2
DISCUSSION
0
null
null
17,182,632
pmid-15205459|pmid-8390996
This is further supported by the observation of severe hepatotoxicity with control 5b, which has >3 mismatches to all known mouse sequences.
null
140
202
0
false
null
null
This is further supported by the observation of severe hepatotoxicity with control 5b, which has >3 mismatches to all known mouse sequences.
true
true
true
true
true
37
2
DISCUSSION
0
null
null
17,182,632
pmid-15205459|pmid-8390996
Hepatotoxicity also seemed to be the most severe for the more potent LNA ASO designs regardless of target (see 4b, mismatch 5b, 7b and 10b).
null
140
203
0
false
null
null
Hepatotoxicity also seemed to be the most severe for the more potent LNA ASO designs regardless of target (see 4b, mismatch 5b, 7b and 10b).
true
true
true
true
true
37
2
DISCUSSION
0
null
null
17,182,632
pmid-15205459|pmid-8390996
Thus, therapeutic index was not improved, and was likely decreased relative to the MOE ASOs.
null
92
204
0
false
null
null
Thus, therapeutic index was not improved, and was likely decreased relative to the MOE ASOs.
true
true
true
true
true
37
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
The hepatotoxicity was evident from the observation of multiple parameters, including histopathological evaluation of liver tissue upon necropsy as well as large increases in plasma levels of aminotransferases (ALT and AST).
[ "42", "43", "44" ]
224
205
0
false
The hepatotoxicity was evident from the observation of multiple parameters, including histopathological evaluation of liver tissue upon necropsy as well as large increases in plasma levels of aminotransferases (ALT and AST).
[]
The hepatotoxicity was evident from the observation of multiple parameters, including histopathological evaluation of liver tissue upon necropsy as well as large increases in plasma levels of aminotransferases (ALT and AST).
true
true
true
true
true
38
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
Furthermore, the toxicity was commonly accompanied by large increases in liver and/or spleen weights, likely as a consequence arising from a response to hepatic injury induced by the LNA ASOs.
[ "42", "43", "44" ]
192
206
0
false
Furthermore, the toxicity was commonly accompanied by large increases in liver and/or spleen weights, likely as a consequence arising from a response to hepatic injury induced by the LNA ASOs.
[]
Furthermore, the toxicity was commonly accompanied by large increases in liver and/or spleen weights, likely as a consequence arising from a response to hepatic injury induced by the LNA ASOs.
true
true
true
true
true
38
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
In several cases, the toxicity was severe enough to cause extensive weight loss in the animals.
[ "42", "43", "44" ]
95
207
0
false
In several cases, the toxicity was severe enough to cause extensive weight loss in the animals.
[]
In several cases, the toxicity was severe enough to cause extensive weight loss in the animals.
true
true
true
true
true
38
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
Histology data clearly demonstrated both LNA oligonucleotide-indiced liver necrosis and activation of apoptosis pathways, as evidenced by H&E staining, as well as cleaved caspase 3, increased Bax expression and increased expression of the M30 neo-epitope.
[ "42", "43", "44" ]
255
208
0
false
Histology data clearly demonstrated both LNA oligonucleotide-indiced liver necrosis and activation of apoptosis pathways, as evidenced by H&E staining, as well as cleaved caspase 3, increased Bax expression and increased expression of the M30 neo-epitope.
[]
Histology data clearly demonstrated both LNA oligonucleotide-indiced liver necrosis and activation of apoptosis pathways, as evidenced by H&E staining, as well as cleaved caspase 3, increased Bax expression and increased expression of the M30 neo-epitope.
true
true
true
true
true
38
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
The upregulation of the pro-apoptotic protein Bax suggests involvement of the p53-mediated apoptosis pathway, as Bax is a key response gene to p53 activation (42,43).
[ "42", "43", "44" ]
166
209
0
false
The upregulation of the pro-apoptotic protein Bax suggests involvement of the p53-mediated apoptosis pathway, as Bax is a key response gene to p53 activation.
[ "42,43" ]
The upregulation of the pro-apoptotic protein Bax suggests involvement of the p53-mediated apoptosis pathway, as Bax is a key response gene to p53 activation.
true
true
true
true
true
38
3
DISCUSSION
1
44
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
Furthermore, GADD45β, a key downstream target gene of p53 during DNA damage and repair process (44), was highly up-regulated in the injured hepatocytes.
[ "42", "43", "44" ]
152
210
1
false
Furthermore, GADD45β, a key downstream target gene of p53 during DNA damage and repair process, was highly up-regulated in the injured hepatocytes.
[ "44" ]
Furthermore, GADD45β, a key downstream target gene of p53 during DNA damage and repair process, was highly up-regulated in the injured hepatocytes.
true
true
true
true
true
38
3
DISCUSSION
1
42
[ "b42", "b43", "b44" ]
17,182,632
pmid-14963330|pmid-12667443|pmid-10749144
GADD45β appears to help protect cells against programmed cell death through blocking the c-jun N-terminal kinase cascade, and is probably induced in response to cellular damage.
[ "42", "43", "44" ]
177
211
0
false
GADD45β appears to help protect cells against programmed cell death through blocking the c-jun N-terminal kinase cascade, and is probably induced in response to cellular damage.
[]
GADD45β appears to help protect cells against programmed cell death through blocking the c-jun N-terminal kinase cascade, and is probably induced in response to cellular damage.
true
true
true
true
true
38
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
It is unclear why LNA oligonucleotides cause this level of hepatotoxicity though the corresponding MOE oligonucleotides do not.
[ "45", "8" ]
127
212
0
false
It is unclear why LNA oligonucleotides cause this level of hepatotoxicity though the corresponding MOE oligonucleotides do not.
[]
It is unclear why LNA oligonucleotides cause this level of hepatotoxicity though the corresponding MOE oligonucleotides do not.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
One possibility is that antisense effects on genes partially complementary to the hepatotoxic ASOs are playing a role in the toxicity, as LNA ASOs have been shown to decrease the selectivity for a perfectly complementary target relative to the corresponding MOE ASOs (45).
[ "45", "8" ]
272
213
1
false
One possibility is that antisense effects on genes partially complementary to the hepatotoxic ASOs are playing a role in the toxicity, as LNA ASOs have been shown to decrease the selectivity for a perfectly complementary target relative to the corresponding MOE ASOs.
[ "45" ]
One possibility is that antisense effects on genes partially complementary to the hepatotoxic ASOs are playing a role in the toxicity, as LNA ASOs have been shown to decrease the selectivity for a perfectly complementary target relative to the corresponding MOE ASOs.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
However, this seems unlikely because multiple unrelated LNA sequences cause similar toxicities.
[ "45", "8" ]
95
214
0
false
However, this seems unlikely because multiple unrelated LNA sequences cause similar toxicities.
[]
However, this seems unlikely because multiple unrelated LNA sequences cause similar toxicities.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
All oligonucleotides were prepared and purified in the same laboratory using the identical methods.
[ "45", "8" ]
99
215
0
false
All oligonucleotides were prepared and purified in the same laboratory using the identical methods.
[]
All oligonucleotides were prepared and purified in the same laboratory using the identical methods.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
The impurity profiles of LNA and MOE ASOs were nearly identical, and contained only the expected impurities resulting from PS oligonucleotide synthesis (PO, N-1, etc.
[ "45", "8" ]
166
216
0
false
The impurity profiles of LNA and MOE ASOs were nearly identical, and contained only the expected impurities resulting from PS oligonucleotide synthesis (PO, N-1, etc.
[]
The impurity profiles of LNA and MOE ASOs were nearly identical, and contained only the expected impurities resulting from PS oligonucleotide synthesis (PO, N-1, etc.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
This makes it extremely unlikely that the toxicity is due to impurities resulting from LNA, but not MOE oligonucleotide synthesis.
[ "45", "8" ]
130
217
0
false
This makes it extremely unlikely that the toxicity is due to impurities resulting from LNA, but not MOE oligonucleotide synthesis.
[]
This makes it extremely unlikely that the toxicity is due to impurities resulting from LNA, but not MOE oligonucleotide synthesis.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
Additionally, since the metabolically unstable PO containing ASO 11b (which should be metabolized in vivo to LNA nucleosides and nucleotides) was non-toxic, it is not likely that the toxicity is due to the LNA monomers.
[ "45", "8" ]
219
218
0
false
Additionally, since the metabolically unstable PO containing ASO 11b (which should be metabolized in vivo to LNA nucleosides and nucleotides) was non-toxic, it is not likely that the toxicity is due to the LNA monomers.
[]
Additionally, since the metabolically unstable PO containing ASO 11b (which should be metabolized in vivo to LNA nucleosides and nucleotides) was non-toxic, it is not likely that the toxicity is due to the LNA monomers.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
This suggests that the intact LNA containing PS oligonucleotides are responsible for the observed toxicity.
[ "45", "8" ]
107
219
0
false
This suggests that the intact LNA containing PS oligonucleotides are responsible for the observed toxicity.
[]
This suggests that the intact LNA containing PS oligonucleotides are responsible for the observed toxicity.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
There are distinct structural differences between MOE and LNA which may allow LNA containing oligonucleotides to selectively effect hepatotoxicity.
[ "45", "8" ]
147
220
0
false
There are distinct structural differences between MOE and LNA which may allow LNA containing oligonucleotides to selectively effect hepatotoxicity.
[]
There are distinct structural differences between MOE and LNA which may allow LNA containing oligonucleotides to selectively effect hepatotoxicity.
true
true
true
true
true
39
4
DISCUSSION
1
8
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
Perhaps importantly, the rigid acyclic 2′-methoxyethyl side chain of MOE protects the corresponding 3′-phosphorothioate linkage from interactions via increased steric bulk and hydration (8), relative to the compact and more hydrophobic cyclic structure of LNA.
[ "45", "8" ]
260
221
1
false
Perhaps importantly, the rigid acyclic 2′-methoxyethyl side chain of MOE protects the corresponding 3′-phosphorothioate linkage from interactions via increased steric bulk and hydration, relative to the compact and more hydrophobic cyclic structure of LNA.
[ "8" ]
Perhaps importantly, the rigid acyclic 2′-methoxyethyl side chain of MOE protects the corresponding 3′-phosphorothioate linkage from interactions via increased steric bulk and hydration, relative to the compact and more hydrophobic cyclic structure of LNA.
true
true
true
true
true
39
4
DISCUSSION
1
45
[ "b45", "b8" ]
17,182,632
NA|pmid-10360355|pmid-9880552|NA|pmid-11181921|pmid-14570775|pmid-10932156|pmid-11160622|pmid-11160622|pmid-15716585|pmid-17030687|pmid-17030687|pmid-12438559|pmid-15625915|pmid-10360355
This could cause selective binding affinity differences between MOE and LNA oligonucleotides for as yet unknown macromolecular binding partners, and/or result in differential compartmentalization of the two classes of oligonucleotides within liver tissue.
[ "45", "8" ]
255
222
0
false
This could cause selective binding affinity differences between MOE and LNA oligonucleotides for as yet unknown macromolecular binding partners, and/or result in differential compartmentalization of the two classes of oligonucleotides within liver tissue.
[]
This could cause selective binding affinity differences between MOE and LNA oligonucleotides for as yet unknown macromolecular binding partners, and/or result in differential compartmentalization of the two classes of oligonucleotides within liver tissue.
true
true
true
true
true
39
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
The mild hepatotoxicity induced 4 days after a single administration of LNA ASO 4b occurred concurrently with apoptosis and activation of Bax and caspase 3 in hepatocytes as evidenced by histopathological evaluation.
[ "41", "46", "47", "48" ]
216
223
0
false
The mild hepatotoxicity induced 4 days after a single administration of LNA ASO 4b occurred concurrently with apoptosis and activation of Bax and caspase 3 in hepatocytes as evidenced by histopathological evaluation.
[]
The mild hepatotoxicity induced 4 days after a single administration of LNA ASO 4b occurred concurrently with apoptosis and activation of Bax and caspase 3 in hepatocytes as evidenced by histopathological evaluation.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
Furthermore, an increase in p-eIF2α was observed to coincide with the onset of toxicity.
[ "41", "46", "47", "48" ]
88
224
0
false
Furthermore, an increase in p-eIF2α was observed to coincide with the onset of toxicity.
[]
Furthermore, an increase in p-eIF2α was observed to coincide with the onset of toxicity.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
Phosphorylated eIF2α inhibits translation initiation, and has been shown to mediate apoptosis, possibly by preventing the synthesis of short lived anti-apoptotic factors (41,46).
[ "41", "46", "47", "48" ]
178
225
0
false
Phosphorylated eIF2α inhibits translation initiation, and has been shown to mediate apoptosis, possibly by preventing the synthesis of short lived anti-apoptotic factors.
[ "41,46" ]
Phosphorylated eIF2α inhibits translation initiation, and has been shown to mediate apoptosis, possibly by preventing the synthesis of short lived anti-apoptotic factors.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
There are four known kinases which phosphorylate eIF2α: PKR, which is activated by binding of double stranded RNA (dsRNA); GCN2, which is activated by amino acid deprivation; HRI, which is activated by low heme levels; and PERK, which responds to stress in the endoplasmic reticulum.
[ "41", "46", "47", "48" ]
283
226
0
false
There are four known kinases which phosphorylate eIF2α: PKR, which is activated by binding of double stranded RNA (dsRNA); GCN2, which is activated by amino acid deprivation; HRI, which is activated by low heme levels; and PERK, which responds to stress in the endoplasmic reticulum.
[]
There are four known kinases which phosphorylate eIF2α: PKR, which is activated by binding of double stranded RNA (dsRNA); GCN2, which is activated by amino acid deprivation; HRI, which is activated by low heme levels; and PERK, which responds to stress in the endoplasmic reticulum.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
It is unclear from our data how treatment with hepatotoxic LNA oligonucleotides results in increased phosphorylation of eIF2α; however, it is tempting to speculate that PKR could be involved.
[ "41", "46", "47", "48" ]
191
227
0
false
It is unclear from our data how treatment with hepatotoxic LNA oligonucleotides results in increased phosphorylation of eIF2α; however, it is tempting to speculate that PKR could be involved.
[]
It is unclear from our data how treatment with hepatotoxic LNA oligonucleotides results in increased phosphorylation of eIF2α; however, it is tempting to speculate that PKR could be involved.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
PKR is activated by binding of dsRNA to distinct dsRNA binding domains which serve as allosteric inhibitors of the kinase domain (47,48).
[ "41", "46", "47", "48" ]
137
228
0
false
PKR is activated by binding of dsRNA to distinct dsRNA binding domains which serve as allosteric inhibitors of the kinase domain.
[ "47,48" ]
PKR is activated by binding of dsRNA to distinct dsRNA binding domains which serve as allosteric inhibitors of the kinase domain.
true
true
true
true
true
40
5
DISCUSSION
1
41
[ "b41", "b46", "b47", "b48" ]
17,182,632
NA|NA|NA|NA|NA|pmid-16717090|pmid-11555640|pmid-11032824|pmid-8995434
It remains to be determined if LNA oligonucleotides interact with PKR, and more extensive mechanistic work is required to confirm both p-eIF2α mediation of an acute apoptotic response in hepatocytes, and elucidate the precise biochemical mechanism responsible for the observed hepatotoxicity.
[ "41", "46", "47", "48" ]
292
229
0
false
It remains to be determined if LNA oligonucleotides interact with PKR, and more extensive mechanistic work is required to confirm both p-eIF2α mediation of an acute apoptotic response in hepatocytes, and elucidate the precise biochemical mechanism responsible for the observed hepatotoxicity.
[]
It remains to be determined if LNA oligonucleotides interact with PKR, and more extensive mechanistic work is required to confirm both p-eIF2α mediation of an acute apoptotic response in hepatocytes, and elucidate the precise biochemical mechanism responsible for the observed hepatotoxicity.
true
true
true
true
true
40
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
In conclusion, we have shown that optimization of size and gap configuration employing LNA containing ASOs can improve potency in mouse liver.
[ "27", "49" ]
142
230
0
false
In conclusion, we have shown that optimization of size and gap configuration employing LNA containing ASOs can improve potency in mouse liver.
[]
In conclusion, we have shown that optimization of size and gap configuration employing LNA containing ASOs can improve potency in mouse liver.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
However, this potency increase is strongly correlated with the onset of a severe hepatotoxicity not seen with the corresponding MOE ASOs, and therapeutic index is not improved.
[ "27", "49" ]
176
231
0
false
However, this potency increase is strongly correlated with the onset of a severe hepatotoxicity not seen with the corresponding MOE ASOs, and therapeutic index is not improved.
[]
However, this potency increase is strongly correlated with the onset of a severe hepatotoxicity not seen with the corresponding MOE ASOs, and therapeutic index is not improved.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
These results suggest that while LNA ASOs have the potential to improve potency of antisense therapeutics, they impose a significant risk of hepatotoxicity.
[ "27", "49" ]
156
232
0
false
These results suggest that while LNA ASOs have the potential to improve potency of antisense therapeutics, they impose a significant risk of hepatotoxicity.
[]
These results suggest that while LNA ASOs have the potential to improve potency of antisense therapeutics, they impose a significant risk of hepatotoxicity.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
The toxicities observed herein also pose challenges for interpreting target validation and pharmacology experiments using LNA ASOs in rodent models.
[ "27", "49" ]
148
233
0
false
The toxicities observed herein also pose challenges for interpreting target validation and pharmacology experiments using LNA ASOs in rodent models.
[]
The toxicities observed herein also pose challenges for interpreting target validation and pharmacology experiments using LNA ASOs in rodent models.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
It is possible more extensive screening efforts may identify less toxic LNA sequences, or that other ASO designs utilizing LNA may not elicit hepatotoxicity.
[ "27", "49" ]
157
234
0
false
It is possible more extensive screening efforts may identify less toxic LNA sequences, or that other ASO designs utilizing LNA may not elicit hepatotoxicity.
[]
It is possible more extensive screening efforts may identify less toxic LNA sequences, or that other ASO designs utilizing LNA may not elicit hepatotoxicity.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
Additionally, bicyclic nucleosides similar to LNA such as amino-LNA, thio-LNA (27) and ENA (which contains one extra methylene unit in the bicyclic bridge) (49) have been reported to show antisense effects similar to LNA and MOE ASOs.
[ "27", "49" ]
234
235
1
false
Additionally, bicyclic nucleosides similar to LNA such as amino-LNA, thio-LNA and ENA (which contains one extra methylene unit in the bicyclic bridge) have been reported to show antisense effects similar to LNA and MOE ASOs.
[ "27", "49" ]
Additionally, bicyclic nucleosides similar to LNA such as amino-LNA, thio-LNA and ENA (which contains one extra methylene unit in the bicyclic bridge) have been reported to show antisense effects similar to LNA and MOE ASOs.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
Although optimized designs of one or more of these modifications may ultimately improve potency while maintaining the safety profile of MOE ASOs, no detailed characterization of their toxicological properties has yet been reported.
[ "27", "49" ]
231
236
0
false
Although optimized designs of one or more of these modifications may ultimately improve potency while maintaining the safety profile of MOE ASOs, no detailed characterization of their toxicological properties has yet been reported.
[]
Although optimized designs of one or more of these modifications may ultimately improve potency while maintaining the safety profile of MOE ASOs, no detailed characterization of their toxicological properties has yet been reported.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
It is clear that additional structure–activity and structure–toxicity relationship studies will be required to more fully assess the therapeutic potential of LNA and other bicyclic nucleoside modified oligonucleotides.
[ "27", "49" ]
218
237
0
false
It is clear that additional structure–activity and structure–toxicity relationship studies will be required to more fully assess the therapeutic potential of LNA and other bicyclic nucleoside modified oligonucleotides.
[]
It is clear that additional structure–activity and structure–toxicity relationship studies will be required to more fully assess the therapeutic potential of LNA and other bicyclic nucleoside modified oligonucleotides.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
Ultimately, the value of LNA oligonucleotide drugs will be determined in human clinical trials, where they are currently being developed for the treatment of cancer.
[ "27", "49" ]
165
238
0
false
Ultimately, the value of LNA oligonucleotide drugs will be determined in human clinical trials, where they are currently being developed for the treatment of cancer.
[]
Ultimately, the value of LNA oligonucleotide drugs will be determined in human clinical trials, where they are currently being developed for the treatment of cancer.
true
true
true
true
true
41
6
DISCUSSION
1
27
[ "b27", "b49" ]
17,182,632
NA|pmid-16978088
Our results are based only on studies in rodents; however, caution should be exercised in the clinical development of LNA modified oligonucleotides, especially for chronic, non-life threatening indications.
[ "27", "49" ]
206
239
0
false
Our results are based only on studies in rodents; however, caution should be exercised in the clinical development of LNA modified oligonucleotides, especially for chronic, non-life threatening indications.
[]
Our results are based only on studies in rodents; however, caution should be exercised in the clinical development of LNA modified oligonucleotides, especially for chronic, non-life threatening indications.
true
true
true
true
true
41
0
INTRODUCTION
1
1–4
[ "B1 B2 B3 B4", "B1", "B5" ]
17,567,608
pmid-15568977|pmid-10357855|pmid-11516927|pmid-10754547|pmid-15568977|pmid-12142524
Homologous recombination (HR) is a template-dependent, high-fidelity DNA damage repair and tolerance pathway that negotiates complex DNA damage, such as double-stranded DNA breaks (DSBs), gaps, and interstrand crosslinks, as well as stalled or collapsed replication forks (1–4).
[ "1–4", "1", "5" ]
278
240
1
false
Homologous recombination (HR) is a template-dependent, high-fidelity DNA damage repair and tolerance pathway that negotiates complex DNA damage, such as double-stranded DNA breaks (DSBs), gaps, and interstrand crosslinks, as well as stalled or collapsed replication forks.
[ "1–4" ]
Homologous recombination (HR) is a template-dependent, high-fidelity DNA damage repair and tolerance pathway that negotiates complex DNA damage, such as double-stranded DNA breaks (DSBs), gaps, and interstrand crosslinks, as well as stalled or collapsed replication forks.
true
true
true
true
true
42
0
INTRODUCTION
1
1–4
[ "B1 B2 B3 B4", "B1", "B5" ]
17,567,608
pmid-15568977|pmid-10357855|pmid-11516927|pmid-10754547|pmid-15568977|pmid-12142524
Defects in HR lead to sensitivity to genotoxic agents and genomic instability (1,5).
[ "1–4", "1", "5" ]
84
241
0
false
Defects in HR lead to sensitivity to genotoxic agents and genomic instability.
[ "1,5" ]
Defects in HR lead to sensitivity to genotoxic agents and genomic instability.
true
true
true
true
true
42
1
INTRODUCTION
1
10
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
The process of HR can be conceptually divided into three stages.
[ "10", "2" ]
64
242
0
false
The process of HR can be conceptually divided into three stages.
[]
The process of HR can be conceptually divided into three stages.
true
true
true
true
true
43
1
INTRODUCTION
1
10
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
In presynapsis, the lesion is processed to a single-stranded DNA (ssDNA) intermediate.
[ "10", "2" ]
86
243
0
false
In presynapsis, the lesion is processed to a single-stranded DNA (ssDNA) intermediate.
[]
In presynapsis, the lesion is processed to a single-stranded DNA (ssDNA) intermediate.
true
true
true
true
true
43
1
INTRODUCTION
1
10
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
In vivo, ssDNA is likely bound by the ssDNA-binding protein RPA, requiring mediator proteins, such as Rad52 and the Rad55-Rad57 heterodimer, to allow formation of the presynaptic filament of Rad51-ATP-ssDNA (6–9).
[ "10", "2" ]
213
244
0
false
In vivo, ssDNA is likely bound by the ssDNA-binding protein RPA, requiring mediator proteins, such as Rad52 and the Rad55-Rad57 heterodimer, to allow formation of the presynaptic filament of Rad51-ATP-ssDNA (6–9).
[]
In vivo, ssDNA is likely bound by the ssDNA-binding protein RPA, requiring mediator proteins, such as Rad52 and the Rad55-Rad57 heterodimer, to allow formation of the presynaptic filament of Rad51-ATP-ssDNA (6–9).
true
true
true
true
true
43
1
INTRODUCTION
1
10
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
During synapsis, the presynaptic filament mediates homology search and DNA strand invasion to form a joint molecule or D–loop (10).
[ "10", "2" ]
131
245
1
false
During synapsis, the presynaptic filament mediates homology search and DNA strand invasion to form a joint molecule or D–loop.
[ "10" ]
During synapsis, the presynaptic filament mediates homology search and DNA strand invasion to form a joint molecule or D–loop.
true
true
true
true
true
43
1
INTRODUCTION
1
10
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
In postsynapsis, Rad51 is assumed to dissociate from the product heteroduplex DNA to allow DNA synthesis from the invading 3′ end.
[ "10", "2" ]
130
246
0
false
In postsynapsis, Rad51 is assumed to dissociate from the product heteroduplex DNA to allow DNA synthesis from the invading 3′ end.
[]
In postsynapsis, Rad51 is assumed to dissociate from the product heteroduplex DNA to allow DNA synthesis from the invading 3′ end.
true
true
true
true
true
43
1
INTRODUCTION
1
2
[ "B10", "B2" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
After DNA synthesis, different sub-pathways (Synthesis-Dependent Strand Annealing, DSB Repair) generate contiguous chromosomes (2).
[ "10", "2" ]
131
247
1
false
After DNA synthesis, different sub-pathways (Synthesis-Dependent Strand Annealing, DSB Repair) generate contiguous chromosomes.
[ "2" ]
After DNA synthesis, different sub-pathways (Synthesis-Dependent Strand Annealing, DSB Repair) generate contiguous chromosomes.
true
true
true
true
true
43
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Rad51 and Rad54 are two key proteins in HR (1).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
47
248
1
false
Rad51 and Rad54 are two key proteins in HR.
[ "1" ]
Rad51 and Rad54 are two key proteins in HR.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Like RecA, Rad51 forms a helical filament on DNA in the presence of ATP and catalyzes homology search and DNA strand invasion (10–13).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
134
249
0
false
Like RecA, Rad51 forms a helical filament on DNA in the presence of ATP and catalyzes homology search and DNA strand invasion.
[ "10–13" ]
Like RecA, Rad51 forms a helical filament on DNA in the presence of ATP and catalyzes homology search and DNA strand invasion.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
This reaction produces heteroduplex DNA, a central recombination intermediate.
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
78
250
0
false
This reaction produces heteroduplex DNA, a central recombination intermediate.
[]
This reaction produces heteroduplex DNA, a central recombination intermediate.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
DNA-binding and DNA-strand exchange activity by budding yeast Rad51 in vitro requires ATP-binding but not ATP hydrolysis as revealed by the analysis of mutants in the invariant lysine residue within the Walker A box (K191 in budding yeast), as well as by using slow or non-hydrolyzable ATP analogs (10,14–19).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
309
251
0
false
DNA-binding and DNA-strand exchange activity by budding yeast Rad51 in vitro requires ATP-binding but not ATP hydrolysis as revealed by the analysis of mutants in the invariant lysine residue within the Walker A box, as well as by using slow or non-hydrolyzable ATP analogs.
[ "K191 in budding yeast", "10,14–19" ]
DNA-binding and DNA-strand exchange activity by budding yeast Rad51 in vitro requires ATP-binding but not ATP hydrolysis as revealed by the analysis of mutants in the invariant lysine residue within the Walker A box, as well as by using slow or non-hydrolyzable ATP analogs.
true
true
true
true
true
44
2
INTRODUCTION
1
20
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
However, in vivo ATP hydrolysis appears to be required for protein function (20).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
81
252
1
false
However, in vivo ATP hydrolysis appears to be required for protein function.
[ "20" ]
However, in vivo ATP hydrolysis appears to be required for protein function.
true
true
true
true
true
44
2
INTRODUCTION
1
14
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Saccharomyces cerevisiae Rad51-K191R encodes a protein that can presumably bind ATP, although this was never directly demonstrated, but not hydrolyze ATP (14).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
159
253
1
false
Saccharomyces cerevisiae Rad51-K191R encodes a protein that can presumably bind ATP, although this was never directly demonstrated, but not hydrolyze ATP.
[ "14" ]
Saccharomyces cerevisiae Rad51-K191R encodes a protein that can presumably bind ATP, although this was never directly demonstrated, but not hydrolyze ATP.
true
true
true
true
true
44
2
INTRODUCTION
1
20
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
The mutant protein when expressed at native levels in haploid cells conferred severe sensitivity to IR and a DSB-repair defect (20).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
132
254
1
false
The mutant protein when expressed at native levels in haploid cells conferred severe sensitivity to IR and a DSB-repair defect.
[ "20" ]
The mutant protein when expressed at native levels in haploid cells conferred severe sensitivity to IR and a DSB-repair defect.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Similarly, the equivalent RecA mutant (RecA-K72R) cannot complement the UV sensitivity of a RecA-deficient strain (21,22).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
122
255
0
false
Similarly, the equivalent RecA mutant (RecA-K72R) cannot complement the UV sensitivity of a RecA-deficient strain.
[ "21,22" ]
Similarly, the equivalent RecA mutant (RecA-K72R) cannot complement the UV sensitivity of a RecA-deficient strain.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Other ATPase defective RecA mutants show less severe defects in vivo (23,24).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
77
256
0
false
Other ATPase defective RecA mutants show less severe defects in vivo.
[ "23,24" ]
Other ATPase defective RecA mutants show less severe defects in vivo.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
When expressed at high levels, budding yeast Rad51-K191R complements the MMS- and IR-sensitivity of a Rad51-deficient strain to near completion (14,20).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
152
257
0
false
When expressed at high levels, budding yeast Rad51-K191R complements the MMS- and IR-sensitivity of a Rad51-deficient strain to near completion.
[ "14,20" ]
When expressed at high levels, budding yeast Rad51-K191R complements the MMS- and IR-sensitivity of a Rad51-deficient strain to near completion.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
The importance of ATP hydrolysis for the in vivo function of RecA-like proteins is underlined by the dominant-negative effect exerted by the equivalent human Rad51-K133R mutant protein when expressed in mouse, chicken or human cells (25–28).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
241
258
0
false
The importance of ATP hydrolysis for the in vivo function of RecA-like proteins is underlined by the dominant-negative effect exerted by the equivalent human Rad51-K133R mutant protein when expressed in mouse, chicken or human cells (25–28).
[]
The importance of ATP hydrolysis for the in vivo function of RecA-like proteins is underlined by the dominant-negative effect exerted by the equivalent human Rad51-K133R mutant protein when expressed in mouse, chicken or human cells (25–28).
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
The in vitro and in vivo results regarding the requirement of ATP hydrolysis for Rad51 (RecA) function present an apparent contradiction.
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
137
259
0
false
The in vitro and in vivo results regarding the requirement of ATP hydrolysis for Rad51 (RecA) function present an apparent contradiction.
[]
The in vitro and in vivo results regarding the requirement of ATP hydrolysis for Rad51 (RecA) function present an apparent contradiction.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
However, in vitro DNA strand invasion assays typically sidestep the requirement for product release by Rad51 (or RecA), which is achieved by SDS/proteinase K treatment.
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
168
260
0
false
However, in vitro DNA strand invasion assays typically sidestep the requirement for product release by Rad51 (or RecA), which is achieved by SDS/proteinase K treatment.
[]
However, in vitro DNA strand invasion assays typically sidestep the requirement for product release by Rad51 (or RecA), which is achieved by SDS/proteinase K treatment.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Indeed, biochemical and electron microscopic analysis of the human Rad51 protein showed that Rad51-DNA complexes are stabilized under conditions that inhibit ATP hydrolysis (15,16), suggesting a need of ATP hydrolysis for Rad51 turnover from dsDNA.
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
248
261
0
false
Indeed, biochemical and electron microscopic analysis of the human Rad51 protein showed that Rad51-DNA complexes are stabilized under conditions that inhibit ATP hydrolysis, suggesting a need of ATP hydrolysis for Rad51 turnover from dsDNA.
[ "15,16" ]
Indeed, biochemical and electron microscopic analysis of the human Rad51 protein showed that Rad51-DNA complexes are stabilized under conditions that inhibit ATP hydrolysis, suggesting a need of ATP hydrolysis for Rad51 turnover from dsDNA.
true
true
true
true
true
44
2
INTRODUCTION
1
19
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
Also experiments with RecA protein have demonstrated the need for ATP hydrolysis to release the heteroduplex product (19).
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
122
262
1
false
Also experiments with RecA protein have demonstrated the need for ATP hydrolysis to release the heteroduplex product.
[ "19" ]
Also experiments with RecA protein have demonstrated the need for ATP hydrolysis to release the heteroduplex product.
true
true
true
true
true
44
2
INTRODUCTION
1
1
[ "B1", "B20", "B14", "B20", "B21", "B22", "B23", "B24", "B14", "B20", "B15", "B16", "B19" ]
17,567,608
pmid-15568977|pmid-12192033|pmid-8910403|pmid-12192033|pmid-8133517|pmid-8371266|pmid-9973562|pmid-9973561|pmid-8910403|pmid-12192033|pmid-16388992|NA|pmid-2147722|pmid-17030607|pmid-12359723|pmid-16979659|pmid-16388992|NA
These experiments suggest that ATP hydrolysis by Rad51 is needed to enhance filament dynamics.
[ "1", "20", "14", "20", "21", "22", "23", "24", "14", "20", "15", "16", "19" ]
94
263
0
false
These experiments suggest that ATP hydrolysis by Rad51 is needed to enhance filament dynamics.
[]
These experiments suggest that ATP hydrolysis by Rad51 is needed to enhance filament dynamics.
true
true
true
true
true
44
3
INTRODUCTION
1
31
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Rad54 protein is a member of the Swi2/Snf2 family of dsDNA-dependent ATPases (29,30) and processively translocates along the dsDNA lattice at up to 300 bp/sec (31).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
164
264
1
false
Rad54 protein is a member of the Swi2/Snf2 family of dsDNA-dependent ATPases and processively translocates along the dsDNA lattice at up to 300 bp/sec.
[ "29,30", "31" ]
Rad54 protein is a member of the Swi2/Snf2 family of dsDNA-dependent ATPases and processively translocates along the dsDNA lattice at up to 300 bp/sec.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Deletion of the RAD54 gene in budding yeast confers as strong a mitotic recombination defect or IR sensitivity as a deficiency in the RAD51 gene (1,32).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
152
265
0
false
Deletion of the RAD54 gene in budding yeast confers as strong a mitotic recombination defect or IR sensitivity as a deficiency in the RAD51 gene.
[ "1,32" ]
Deletion of the RAD54 gene in budding yeast confers as strong a mitotic recombination defect or IR sensitivity as a deficiency in the RAD51 gene.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
In vivo function of Rad54 protein is largely compromised in the rad54-K341R mutant, which encodes a mutant Rad54 protein that is defective in ATP hydrolysis (33–36).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
165
266
0
false
In vivo function of Rad54 protein is largely compromised in the rad54-K341R mutant, which encodes a mutant Rad54 protein that is defective in ATP hydrolysis (33–36).
[]
In vivo function of Rad54 protein is largely compromised in the rad54-K341R mutant, which encodes a mutant Rad54 protein that is defective in ATP hydrolysis (33–36).
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Rad51 and Rad54 act in a single molecular pathway and physically interact (37–39).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
82
267
0
false
Rad51 and Rad54 act in a single molecular pathway and physically interact (37–39).
[]
Rad51 and Rad54 act in a single molecular pathway and physically interact.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Rad54 was found to stabilize Rad51-ssDNA filaments in the presynaptic phase of recombination in an ATPase-independent fashion (40–42).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
134
268
0
false
Rad54 was found to stabilize Rad51-ssDNA filaments in the presynaptic phase of recombination in an ATPase-independent fashion (40–42).
[]
Rad54 was found to stabilize Rad51-ssDNA filaments in the presynaptic phase of recombination in an ATPase-independent fashion.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Rad54 also stimulates DNA strand exchange at the synaptic stage (35,43–46).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
75
269
0
false
Rad54 also stimulates DNA strand exchange at the synaptic stage (35,43–46).
[]
Rad54 also stimulates DNA strand exchange at the synaptic stage (35,43–46).
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
The mechanism of this stimulation is not fully understood but requires the motor function of Rad54 and depends on its ATPase activity.
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
134
270
0
false
The mechanism of this stimulation is not fully understood but requires the motor function of Rad54 and depends on its ATPase activity.
[]
The mechanism of this stimulation is not fully understood but requires the motor function of Rad54 and depends on its ATPase activity.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Possible mechanisms include the sliding of the target dsDNA during homology search, opening the target dsDNA by translocating on duplex DNA, or removing Rad51 from dsDNA that inhibit Rad51-mediated DNA strand exchange (29,30).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
226
271
0
false
Possible mechanisms include the sliding of the target dsDNA during homology search, opening the target dsDNA by translocating on duplex DNA, or removing Rad51 from dsDNA that inhibit Rad51-mediated DNA strand exchange.
[ "29,30" ]
Possible mechanisms include the sliding of the target dsDNA during homology search, opening the target dsDNA by translocating on duplex DNA, or removing Rad51 from dsDNA that inhibit Rad51-mediated DNA strand exchange.
true
true
true
true
true
45
3
INTRODUCTION
1
29
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Moreover, Rad54 was demonstrated to be able to remodel nucleosomes in vitro, although no effect of Rad54 on nucleosome positioning during DSB repair has been identified in budding yeast (42,47–49).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
197
272
0
false
Moreover, Rad54 was demonstrated to be able to remodel nucleosomes in vitro, although no effect of Rad54 on nucleosome positioning during DSB repair has been identified in budding yeast (42,47–49).
[]
Moreover, Rad54 was demonstrated to be able to remodel nucleosomes in vitro, although no effect of Rad54 on nucleosome positioning during DSB repair has been identified in budding yeast.
true
true
true
true
true
45
3
INTRODUCTION
1
52
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
During postsynapsis, Rad54 was shown to enhance branch migration during DNA strand exchange (50,51), but it is unclear whether Rad54 acts as a junction-specific motor protein like RuvB in bacteria (52).
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
202
273
1
false
During postsynapsis, Rad54 was shown to enhance branch migration during DNA strand exchange, but it is unclear whether Rad54 acts as a junction-specific motor protein like RuvB in bacteria.
[ "50,51", "52" ]
During postsynapsis, Rad54 was shown to enhance branch migration during DNA strand exchange, but it is unclear whether Rad54 acts as a junction-specific motor protein like RuvB in bacteria.
true
true
true
true
true
45
3
INTRODUCTION
1
53
[ "B29", "B30", "B31", "B1", "B32", "B29", "B30", "B50", "B51", "B52", "B53" ]
17,567,608
pmid-12826279|pmid-16935872|pmid-16818238|pmid-15568977|pmid-12560498|pmid-12826279|pmid-16935872|pmid-11459988|pmid-16862129|pmid-8631697|pmid-12087154|pmid-12192033|pmid-17030607|pmid-12192033|pmid-17030607|pmid-12748644|pmid-12748645|pmid-12192033|pmid-16980587
Overexpression of Rad54 leads to a decrease in conversion tract length (53) not increase as predicted, if Rad54 were to drive branch migration.
[ "29", "30", "31", "1", "32", "29", "30", "50", "51", "52", "53" ]
143
274
1
false
Overexpression of Rad54 leads to a decrease in conversion tract length not increase as predicted, if Rad54 were to drive branch migration.
[ "53" ]
Overexpression of Rad54 leads to a decrease in conversion tract length not increase as predicted, if Rad54 were to drive branch migration.
true
true
true
true
true
45
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
Genetic analysis suggests that Rad54 acts at a step after Rad51 protein, consistent with cytological data showing that RAD54 is not required for Rad51 focus formation (54–58).
[ "59", "60", "61", "41", "62" ]
175
275
0
false
Genetic analysis suggests that Rad54 acts at a step after Rad51 protein, consistent with cytological data showing that RAD54 is not required for Rad51 focus formation (54–58).
[]
Genetic analysis suggests that Rad54 acts at a step after Rad51 protein, consistent with cytological data showing that RAD54 is not required for Rad51 focus formation.
true
true
true
true
true
46
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
Together with data from chromatin immunoprecipitation experiments (59,60), these results suggest that the critical function of Rad54 is either during synapsis or postsynapsis but the results are not able to distinguish between both possibilities.
[ "59", "60", "61", "41", "62" ]
246
276
0
false
Together with data from chromatin immunoprecipitation experiments, these results suggest that the critical function of Rad54 is either during synapsis or postsynapsis but the results are not able to distinguish between both possibilities.
[ "59,60" ]
Together with data from chromatin immunoprecipitation experiments, these results suggest that the critical function of Rad54 is either during synapsis or postsynapsis but the results are not able to distinguish between both possibilities.
true
true
true
true
true
46
4
INTRODUCTION
1
61
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
Since Rad54 is a dsDNA motor protein that interacts with Rad51, we have focused on the interaction between Rad54 and the Rad51-dsDNA filament (61).
[ "59", "60", "61", "41", "62" ]
147
277
1
false
Since Rad54 is a dsDNA motor protein that interacts with Rad51, we have focused on the interaction between Rad54 and the Rad51-dsDNA filament.
[ "61" ]
Since Rad54 is a dsDNA motor protein that interacts with Rad51, we have focused on the interaction between Rad54 and the Rad51-dsDNA filament.
true
true
true
true
true
46
4
INTRODUCTION
1
41
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
We discovered that Rad54 remodels the Rad51-dsDNA filament, resulting in the dissociation of Rad51 from dsDNA (41).
[ "59", "60", "61", "41", "62" ]
115
278
1
false
We discovered that Rad54 remodels the Rad51-dsDNA filament, resulting in the dissociation of Rad51 from dsDNA.
[ "41" ]
We discovered that Rad54 remodels the Rad51-dsDNA filament, resulting in the dissociation of Rad51 from dsDNA.
true
true
true
true
true
46
4
INTRODUCTION
1
62
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
Using electron microscopic analysis, Rad54 was found to preferentially localize to one terminus of the Rad51-dsDNA filament, consistent with Rad54 translocating along dsDNA and then docking at the end of the Rad51 filament or directly binding the filament end from solution (62).
[ "59", "60", "61", "41", "62" ]
279
279
1
false
Using electron microscopic analysis, Rad54 was found to preferentially localize to one terminus of the Rad51-dsDNA filament, consistent with Rad54 translocating along dsDNA and then docking at the end of the Rad51 filament or directly binding the filament end from solution.
[ "62" ]
Using electron microscopic analysis, Rad54 was found to preferentially localize to one terminus of the Rad51-dsDNA filament, consistent with Rad54 translocating along dsDNA and then docking at the end of the Rad51 filament or directly binding the filament end from solution.
true
true
true
true
true
46
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
These data support a model, in which Rad54 acts as a turnover factor for the Rad51-heteroduplex DNA product complex, resulting in product release by Rad51 to allow access of the DNA synthesis machinery to the invading 3′ end.
[ "59", "60", "61", "41", "62" ]
225
280
0
false
These data support a model, in which Rad54 acts as a turnover factor for the Rad51-heteroduplex DNA product complex, resulting in product release by Rad51 to allow access of the DNA synthesis machinery to the invading 3′ end.
[]
These data support a model, in which Rad54 acts as a turnover factor for the Rad51-heteroduplex DNA product complex, resulting in product release by Rad51 to allow access of the DNA synthesis machinery to the invading 3′ end.
true
true
true
true
true
46
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
This model also rationalizes significant differences between RecA and Rad51.
[ "59", "60", "61", "41", "62" ]
76
281
0
false
This model also rationalizes significant differences between RecA and Rad51.
[]
This model also rationalizes significant differences between RecA and Rad51.
true
true
true
true
true
46
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
RecA exhibits ∼200-fold higher ATPase activity on dsDNA and releases from DNA after ATP hydrolysis, whereas Rad51 appears to be much less dynamic in filament assembly/disassembly (10,15,16,19).
[ "59", "60", "61", "41", "62" ]
193
282
0
false
RecA exhibits ∼200-fold higher ATPase activity on dsDNA and releases from DNA after ATP hydrolysis, whereas Rad51 appears to be much less dynamic in filament assembly/disassembly (10,15,16,19).
[]
RecA exhibits ∼200-fold higher ATPase activity on dsDNA and releases from DNA after ATP hydrolysis, whereas Rad51 appears to be much less dynamic in filament assembly/disassembly.
true
true
true
true
true
46
4
INTRODUCTION
1
59
[ "B59", "B60", "B61", "B41", "B62" ]
17,567,608
pmid-12887907|pmid-12887906|pmid-12359723|pmid-12453424|pmid-16785421|pmid-12359723|pmid-16818238|pmid-16916635|pmid-16785421
The function of Rad54 as a Rad51 turnover factor is consistent with the absence of a Rad54 homolog in bacteria, because RecA is capable of turnover using its intrinsic ATPase activity.
[ "59", "60", "61", "41", "62" ]
184
283
0
false
The function of Rad54 as a Rad51 turnover factor is consistent with the absence of a Rad54 homolog in bacteria, because RecA is capable of turnover using its intrinsic ATPase activity.
[]
The function of Rad54 as a Rad51 turnover factor is consistent with the absence of a Rad54 homolog in bacteria, because RecA is capable of turnover using its intrinsic ATPase activity.
true
true
true
true
true
46
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
Here, we analyzed the roles of both the Rad51 and Rad54 ATPase activities in turnover of the Rad51-dsDNA filament.
[ "28" ]
114
284
0
false
Here, we analyzed the roles of both the Rad51 and Rad54 ATPase activities in turnover of the Rad51-dsDNA filament.
[]
Here, we analyzed the roles of both the Rad51 and Rad54 ATPase activities in turnover of the Rad51-dsDNA filament.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
The results revealed a number of surprising features of the S. cerevisiae ATPase-deficient Rad51-K191R and Rad51-K191A proteins.
[ "28" ]
128
285
0
false
The results revealed a number of surprising features of the S. cerevisiae ATPase-deficient Rad51-K191R and Rad51-K191A proteins.
[]
The results revealed a number of surprising features of the S. cerevisiae ATPase-deficient Rad51-K191R and Rad51-K191A proteins.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
First, unexpectedly Rad51-K191A protein bound ATP, albeit with reduced affinity, similar to human Rad51-K133A (28).
[ "28" ]
115
286
1
false
First, unexpectedly Rad51-K191A protein bound ATP, albeit with reduced affinity, similar to human Rad51-K133A.
[ "28" ]
First, unexpectedly Rad51-K191A protein bound ATP, albeit with reduced affinity, similar to human Rad51-K133A.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
Second, the Rad51-K191R mutant protein displayed a DNA binding defect.
[ "28" ]
70
287
0
false
Second, the Rad51-K191R mutant protein displayed a DNA binding defect.
[]
Second, the Rad51-K191R mutant protein displayed a DNA binding defect.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
Third, once formed the Rad51-K191R-dsDNA complexes were exceptionally stable.
[ "28" ]
77
288
0
false
Third, once formed the Rad51-K191R-dsDNA complexes were exceptionally stable.
[]
Third, once formed the Rad51-K191R-dsDNA complexes were exceptionally stable.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
We demonstrate that the Rad54 ATPase activity was specifically enhanced in its interaction with the Rad51-dsDNA filament.
[ "28" ]
121
289
0
false
We demonstrate that the Rad54 ATPase activity was specifically enhanced in its interaction with the Rad51-dsDNA filament.
[]
We demonstrate that the Rad54 ATPase activity was specifically enhanced in its interaction with the Rad51-dsDNA filament.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
Efficient Rad51 turnover from dsDNA required both the Rad51 and Rad54 ATPase activities.
[ "28" ]
88
290
0
false
Efficient Rad51 turnover from dsDNA required both the Rad51 and Rad54 ATPase activities.
[]
Efficient Rad51 turnover from dsDNA required both the Rad51 and Rad54 ATPase activities.
true
true
true
true
true
47
5
INTRODUCTION
1
28
[ "B28" ]
17,567,608
pmid-17302439|pmid-16818238|pmid-16818238|pmid-16818238|pmid-16818238
These results show that Rad51 is not a passive remodeling target of Rad54 and uncovered an intricate cooperation between the Rad51 and Rad54 ATPase activities in Rad51 turnover.
[ "28" ]
177
291
0
false
These results show that Rad51 is not a passive remodeling target of Rad54 and uncovered an intricate cooperation between the Rad51 and Rad54 ATPase activities in Rad51 turnover.
[]
These results show that Rad51 is not a passive remodeling target of Rad54 and uncovered an intricate cooperation between the Rad51 and Rad54 ATPase activities in Rad51 turnover.
true
true
true
true
true
47
0
DISCUSSION
0
null
null
17,567,608
pmid-15568977|pmid-10357855|pmid-11516927|pmid-10754547|pmid-15568977|pmid-12142524
Rad51 and Rad54 are key DNA-dependent ATPases functioning in HR in eukaryotes.
null
78
292
0
false
null
null
Rad51 and Rad54 are key DNA-dependent ATPases functioning in HR in eukaryotes.
true
true
true
true
true
48
0
DISCUSSION
0
null
null
17,567,608
pmid-15568977|pmid-10357855|pmid-11516927|pmid-10754547|pmid-15568977|pmid-12142524
Our analysis uncovered unexpected biochemical properties of the ATPase-deficient Rad51-K191R and Rad51-K191A mutant proteins.
null
125
293
0
false
null
null
Our analysis uncovered unexpected biochemical properties of the ATPase-deficient Rad51-K191R and Rad51-K191A mutant proteins.
true
true
true
true
true
48
0
DISCUSSION
0
null
null
17,567,608
pmid-15568977|pmid-10357855|pmid-11516927|pmid-10754547|pmid-15568977|pmid-12142524
Kinetic analysis and experiments with different nucleotide cofactors revealed an intricate relationship between the Rad51 and Rad54 ATPase activities, demonstrating that both ATPase activities are required for efficient turnover of the Rad51-dsDNA filament.
null
257
294
0
false
null
null
Kinetic analysis and experiments with different nucleotide cofactors revealed an intricate relationship between the Rad51 and Rad54 ATPase activities, demonstrating that both ATPase activities are required for efficient turnover of the Rad51-dsDNA filament.
true
true
true
true
true
48
1
DISCUSSION
1
72
[ "B72", "B14", "B44", "B44", "B20", "B28" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
The Walker A motif is a phosphate-binding loop that is found in many purine nucleotide-binding proteins including RecA and Rad51 (72).
[ "72", "14", "44", "44", "20", "28" ]
134
295
1
false
The Walker A motif is a phosphate-binding loop that is found in many purine nucleotide-binding proteins including RecA and Rad51.
[ "72" ]
The Walker A motif is a phosphate-binding loop that is found in many purine nucleotide-binding proteins including RecA and Rad51.
true
true
true
true
true
49
1
DISCUSSION
1
72
[ "B72", "B14", "B44", "B44", "B20", "B28" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
Mutations in the central lysine residue are often used to dissociate ATP binding and ATP hydrolysis, relying on an often untested assumption that the lysine to arginine substituted protein (e.g.
[ "72", "14", "44", "44", "20", "28" ]
194
296
0
false
Mutations in the central lysine residue are often used to dissociate ATP binding and ATP hydrolysis, relying on an often untested assumption that the lysine to arginine substituted protein (e.g.
[]
Mutations in the central lysine residue are often used to dissociate ATP binding and ATP hydrolysis, relying on an often untested assumption that the lysine to arginine substituted protein (e.g.
true
true
true
true
true
49
1
DISCUSSION
1
72
[ "B72", "B14", "B44", "B44", "B20", "B28" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
Rad51-K191R) binds but does not hydrolyze ATP, whereas the lysine to alanine substituted protein (e.g.
[ "72", "14", "44", "44", "20", "28" ]
102
297
0
false
Rad51-K191R) binds but does not hydrolyze ATP, whereas the lysine to alanine substituted protein (e.g.
[]
Rad51-K191R) binds but does not hydrolyze ATP, whereas the lysine to alanine substituted protein (e.g.
true
true
true
true
true
49
1
DISCUSSION
1
72
[ "B72", "B14", "B44", "B44", "B20", "B28" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
Rad51-K191A) cannot bind ATP.
[ "72", "14", "44", "44", "20", "28" ]
29
298
0
false
Rad51-K191A) cannot bind ATP.
[]
Rad51-K191A) cannot bind ATP.
true
true
true
true
true
49
1
DISCUSSION
1
72
[ "B72", "B14", "B44", "B44", "B20", "B28" ]
17,567,608
pmid-8066464|pmid-10357855|pmid-6329717|pmid-8910403|pmid-11030336|pmid-11030336|pmid-12192033|pmid-17302439
Surprisingly, we find that both Rad51-K191R and Rad51-K191A mutant proteins bind ATP, albeit with reduced affinity compared with the wild-type protein (Table 1).
[ "72", "14", "44", "44", "20", "28" ]
161
299
0
false
Surprisingly, we find that both Rad51-K191R and Rad51-K191A mutant proteins bind ATP, albeit with reduced affinity compared with the wild-type protein (Table 1).
[]
Surprisingly, we find that both Rad51-K191R and Rad51-K191A mutant proteins bind ATP, albeit with reduced affinity compared with the wild-type protein (Table 1).
true
true
true
true
true
49