Datasets:

uuid
stringlengths
4
8
template_uuid
stringclasses
40 values
question
stringlengths
13
193
answer
stringlengths
29
2.2k
benchmark_query
stringlengths
133
622
execution_results
stringlengths
2
1.14M
query_type
stringclasses
2 values
sql_category
stringclasses
26 values
bio_category
stringclasses
14 values
Q1.187
Q1
Is CCKAR a druggable gene?
There are currently 4 approved drugs which target CCKAR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CCKAR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5575', 'drugName': 'Proglumide', 'drugIsApproved': True, 'newLinkedTargets_string': 'CCKBR (ENSG00000110148), CCKAR (ENSG00000163394)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2693', 'drugName': 'Sincalide', 'drugIsApproved': True, 'newLinkedTargets_string': 'CCKAR (ENSG0...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.42
Q1
Is AFP a druggable gene?
There are currently no approved drugs targeting AFP, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%AFP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_262', 'drugName': 'Yttrium Y 90 Tacatuzumab Tetraxetan', 'drugIsApproved': False, 'newLinkedTargets_string': 'AFP (ENSG00000081051)', 'maxClinicalTrialPhase': -1}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.697
Q1
Is IL33 a druggable gene?
There are currently no approved drugs targeting IL33, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL33 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2908', 'drugName': 'Itepekimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL33 (ENSG00000137033)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2323', 'drugName': 'Etokimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL33 (ENSG00000137033)', 'maxClinical...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.110
Q1
Is BDKRB2 a druggable gene?
There are currently 2 approved drugs which target BDKRB2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BDKRB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3024', 'drugName': 'Icatibant', 'drugIsApproved': True, 'newLinkedTargets_string': 'BDKRB2 (ENSG00000168398)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_226', 'drugName': 'Icatibant Acetate', 'drugIsApproved': True, 'newLinkedTargets_string': 'BDKRB2 (ENSG00000168398)', 'ma...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.39
Q1
Is ADRB2 a druggable gene?
There are currently 90 approved drugs which target ADRB2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADRB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3721', 'drugName': 'Levosalbutamol', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1445', 'drugName': 'Terbutaline Sulfate', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADRB2 (ENSG00000169252)...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.571
Q1
Is HBA1 a druggable gene?
There is 1 drug, Voxelotor, that targets HBA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HBA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2318', 'drugName': 'Voxelotor', 'drugIsApproved': True, 'newLinkedTargets_string': 'HBA1 (ENSG00000206172), HBA2 (ENSG00000188536), HBB (ENSG00000244734)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5816', 'drugName': 'Efaproxiral', 'drugIsApproved': False, 'newLinkedTargets...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1024
Q1
Is P2RX3 a druggable gene?
There are currently no approved drugs targeting P2RX3, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%P2RX3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_913', 'drugName': 'Gefapixant', 'drugIsApproved': False, 'newLinkedTargets_string': 'P2RX3 (ENSG00000109991)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_601', 'drugName': 'Camlipixant', 'drugIsApproved': False, 'newLinkedTargets_string': 'P2RX3 (ENSG00000109991)', 'maxClini...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1299
Q1
Is RPS4Y1 a druggable gene?
There is 1 drug, Ataluren, that targets RPS4Y1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS4Y1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1478
Q1
Is TRAV29DV5 a druggable gene?
There are currently no approved drugs targeting TRAV29DV5, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TRAV29DV5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1483', 'drugName': 'Medi-500', 'drugIsApproved': False, 'newLinkedTargets_string': 'TRAV29DV5 (ENSG00000211810), TRAC (ENSG00000277734), TRBV7-9 (ENSG00000278030), TRGV3 (ENSG00000211699)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_5971', 'drugName': 'Tol-101', 'drugIsAppro...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.486
Q1
Is FZD2 a druggable gene?
There are currently no approved drugs targeting FZD2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FZD2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5828', 'drugName': 'Vantictumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'FZD2 (ENSG00000180340), FZD7 (ENSG00000155760), FZD1 (ENSG00000157240), FZD5 (ENSG00000163251), FZD8 (ENSG00000177283)', 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_5825', 'drugName': 'Vant...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.470
Q1
Is FKBP1A a druggable gene?
There are currently 5 approved drugs which target FKBP1A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FKBP1A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5128', 'drugName': 'Tacrolimus', 'drugIsApproved': True, 'newLinkedTargets_string': 'FKBP1A (ENSG00000088832)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1925', 'drugName': 'Everolimus', 'drugIsApproved': True, 'newLinkedTargets_string': 'FKBP1A (ENSG00000088832)', 'maxClin...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.895
Q1
Is MMP13 a druggable gene?
There are currently 4 approved drugs which target MMP13, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MMP13 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_289', 'drugName': 'Doxycycline Anhydrous', 'drugIsApproved': True, 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP8 (ENSG00000118113), MMP7 (ENSG00000137673), MMP1 (ENSG00000196611)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_287', 'drugName': 'Doxycycline Anhydrou...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.952
Q1
Is NDUFAF3 a druggable gene?
There are currently 2 approved drugs which target NDUFAF3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFAF3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.25
Q1
Is ADH6 a druggable gene?
There is 1 drug, Nitrefazole, that targets ADH6, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADH6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1036
Q1
Is PARP2 a druggable gene?
There are currently 7 approved drugs which target PARP2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PARP2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_100', 'drugName': 'Talazoparib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PARP2 (ENSG00000129484), PARP1 (ENSG00000143799)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2224', 'drugName': 'Talazoparib Tosylate', 'drugIsApproved': True, 'newLinkedTargets_string': 'P...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1222
Q1
Is RNPEPL1 a druggable gene?
There are currently no approved drugs targeting RNPEPL1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RNPEPL1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_582', 'drugName': 'Tosedostat', 'drugIsApproved': False, 'newLinkedTargets_string': 'ANPEP (ENSG00000166825), NPEPPS (ENSG00000141279), RNPEP (ENSG00000176393), METAP1 (ENSG00000164024), LNPEP (ENSG00000113441), DNPEP (ENSG00000123992), ENPEP (ENSG00000138792), XPNPEP1 (ENSG00000108039), L...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.69
Q1
Is APCS a druggable gene?
There are currently no approved drugs targeting APCS, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%APCS %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5164', 'drugName': 'Dezamizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'APCS (ENSG00000132703)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_1308', 'drugName': 'Miridesap', 'drugIsApproved': False, 'newLinkedTargets_string': 'APCS (ENSG00000132703)', 'maxClinic...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.889
Q1
Is MKNK2 a druggable gene?
There are currently no approved drugs targeting MKNK2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MKNK2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1066', 'drugName': 'Tomivosertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'MKNK2 (ENSG00000099875), MKNK1 (ENSG00000079277)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1297
Q1
Is RPS3A a druggable gene?
There is 1 drug, Ataluren, that targets RPS3A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS3A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.368
Q1
Is DNMT3A a druggable gene?
There are currently 2 approved drugs which target DNMT3A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DNMT3A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4132', 'drugName': 'Azacitidine', 'drugIsApproved': True, 'newLinkedTargets_string': 'DNMT1 (ENSG00000130816), DNMT3A (ENSG00000119772)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4131', 'drugName': 'Azacitidine', 'drugIsApproved': True, 'newLinkedTargets_string': 'DNMT1 (E...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.508
Q1
Is GABRQ a druggable gene?
There are currently 66 approved drugs which target GABRQ, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GABRQ %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1494', 'drugName': 'Thiopental', 'drugIsApproved': True, 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG00000011677)...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.855
Q1
Is MAP3K8 a druggable gene?
There are currently no approved drugs targeting MAP3K8, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAP3K8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6134', 'drugName': 'Tilpisertib', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAP3K8 (ENSG00000107968)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1348
Q1
Is SELPLG a druggable gene?
There are currently no approved drugs targeting SELPLG, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SELPLG %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3018', 'drugName': 'Neihulizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'SELPLG (ENSG00000110876)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.385
Q1
Is E2F8 a druggable gene?
There are currently no approved drugs targeting E2F8, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%E2F8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4614', 'drugName': 'Edifoligide Sodium', 'drugIsApproved': False, 'newLinkedTargets_string': 'E2F1 (ENSG00000101412), E2F2 (ENSG00000007968), E2F3 (ENSG00000112242), E2F4 (ENSG00000205250), E2F5 (ENSG00000133740), E2F6 (ENSG00000169016), E2F7 (ENSG00000165891), E2F8 (ENSG00000129173)', 'ma...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.739
Q1
Is KCNA6 a druggable gene?
There are currently 5 approved drugs which target KCNA6, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNA6 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.722
Q1
Is ITGB1 a druggable gene?
There is 1 drug, Natalizumab, that targets ITGB1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ITGB1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5016', 'drugName': 'Natalizumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ITGA4 (ENSG00000115232), ITGB7 (ENSG00000139626), ITGB1 (ENSG00000150093)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5015', 'drugName': 'Natalizumab', 'drugIsApproved': True, 'newLinkedTa...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.456
Q1
Is FDPS a druggable gene?
There are currently 9 approved drugs which target FDPS, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FDPS %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4717', 'drugName': 'Risedronate Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'FDPS (ENSG00000160752)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5882', 'drugName': 'Alendronic Acid', 'drugIsApproved': True, 'newLinkedTargets_string': 'FDPS (ENSG00000160752)',...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.266
Q1
Is CHRNA3 a druggable gene?
There are currently 6 approved drugs which target CHRNA3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRNA3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5467', 'drugName': 'Trimethaphan Camsylate', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRNB4 (ENSG00000117971), CHRNA3 (ENSG00000080644)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4467', 'drugName': 'Trimethaphan', 'drugIsApproved': True, 'newLinkedTargets_strin...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.76
Q1
Is APP a druggable gene?
There is 1 drug, Aducanumab, that targets APP, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%APP %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4177', 'drugName': 'Aducanumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'APP (ENSG00000142192)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3123', 'drugName': 'Tramiprosate', 'drugIsApproved': False, 'newLinkedTargets_string': 'APP (ENSG00000142192)', 'maxClinica...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.446
Q1
Is FAAH a druggable gene?
There is 1 drug, Acetaminophen, that targets FAAH, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FAAH %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_147', 'drugName': 'Acetaminophen', 'drugIsApproved': True, 'newLinkedTargets_string': 'PTGS2 (ENSG00000073756), PTGS1 (ENSG00000095303), TRPV1 (ENSG00000196689), FAAH (ENSG00000117480)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_146', 'drugName': 'Acetaminophen', 'drugIsApp...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.397
Q1
Is EGR1 a druggable gene?
There are currently no approved drugs targeting EGR1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EGR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_862', 'drugName': 'Brivoligide', 'drugIsApproved': False, 'newLinkedTargets_string': 'EGR1 (ENSG00000120738)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.178
Q1
Is CASP3 a druggable gene?
There are currently no approved drugs targeting CASP3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CASP3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_45', 'drugName': 'Emricasan', 'drugIsApproved': False, 'newLinkedTargets_string': 'CASP4 (ENSG00000196954), CASP9 (ENSG00000132906), CASP3 (ENSG00000164305), CASP5 (ENSG00000137757), CASP6 (ENSG00000138794), CASP7 (ENSG00000165806), CASP8 (ENSG00000064012), CASP1 (ENSG00000137752), CASP2 (...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1343
Q1
Is SCTR a druggable gene?
There are currently 3 approved drugs which target SCTR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SCTR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4400', 'drugName': 'Secretin', 'drugIsApproved': True, 'newLinkedTargets_string': 'SCTR (ENSG00000080293)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4712', 'drugName': 'Secretin Synthetic Human', 'drugIsApproved': True, 'newLinkedTargets_string': 'SCTR (ENSG00000080293)', ...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1113
Q1
Is PPARA a druggable gene?
There are currently 7 approved drugs which target PPARA, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PPARA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_347', 'drugName': 'Fenofibric Acid', 'drugIsApproved': True, 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4561', 'drugName': 'Ciprofibrate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PPARA (ENSG00000186951)', 'max...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1059
Q1
Is PDE7A a druggable gene?
There are currently 4 approved drugs which target PDE7A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE7A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_766', 'drugName': 'Flavoxate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE8B (ENSG00000113231), PDE8A (ENSG00000073417), PDE7A (ENSG00000205268), PDE7B (ENSG00000171408), PDE4A (ENSG00000065989), PDE4D (ENSG00000113448), PDE4B (ENSG00000184588), PDE4C (ENSG00000105650)', 'maxCl...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.599
Q1
Is HPD a druggable gene?
There is 1 drug, Nitisinone, that targets HPD, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HPD %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4714', 'drugName': 'Nitisinone', 'drugIsApproved': True, 'newLinkedTargets_string': 'HPD (ENSG00000158104)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.62
Q1
Is ANGPT2 a druggable gene?
There is 1 drug, Faricimab, that targets ANGPT2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ANGPT2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_864', 'drugName': 'Faricimab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ANGPT2 (ENSG00000091879), VEGFA (ENSG00000112715)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_865', 'drugName': 'Faricimab', 'drugIsApproved': True, 'newLinkedTargets_string': 'ANGPT2 (ENSG00...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.877
Q1
Is MEN1 a druggable gene?
There are currently no approved drugs targeting MEN1, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MEN1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1716', 'drugName': 'Revumenib', 'drugIsApproved': False, 'newLinkedTargets_string': 'MEN1 (ENSG00000133895), KMT2A (ENSG00000118058)', 'maxClinicalTrialPhase': 1}, {'UUID': 'DrugGeneTargets_v2_3382', 'drugName': 'Sndx-5613', 'drugIsApproved': False, 'newLinkedTargets_string': 'MEN1 (ENSG00...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1146
Q1
Is PRMT5 a druggable gene?
There are currently no approved drugs targeting PRMT5, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PRMT5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1649', 'drugName': 'Pemrametostat', 'drugIsApproved': False, 'newLinkedTargets_string': 'PRMT5 (ENSG00000100462)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1442
Q1
Is TNF a druggable gene?
There are currently 5 approved drugs which target TNF, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNF %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6275', 'drugName': 'Infliximab', 'drugIsApproved': True, 'newLinkedTargets_string': 'TNF (ENSG00000232810)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_393', 'drugName': 'Golimumab', 'drugIsApproved': True, 'newLinkedTargets_string': 'TNF (ENSG00000232810)', 'maxClinicalTria...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.280
Q1
Is CLEC4C a druggable gene?
There are currently no approved drugs targeting CLEC4C, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CLEC4C %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4112', 'drugName': 'Litifilimab', 'drugIsApproved': False, 'newLinkedTargets_string': 'CLEC4C (ENSG00000198178)', 'maxClinicalTrialPhase': 3}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.37
Q1
Is ADRA2C a druggable gene?
There are currently 58 approved drugs which target ADRA2C, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADRA2C %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4923', 'drugName': 'Brimonidine Tartrate', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADRA2A (ENSG00000150594), ADRA2C (ENSG00000184160), ADRA2B (ENSG00000274286)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5012', 'drugName': 'Tizanidine Hydrochloride', 'drugIsAppr...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.666
Q1
Is IL10RA a druggable gene?
There are currently no approved drugs targeting IL10RA, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL10RA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4152', 'drugName': 'Pegilodecakin', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL10RB (ENSG00000243646), IL10RA (ENSG00000110324)', 'maxClinicalTrialPhase': 3}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1385
Q1
Is SNCA a druggable gene?
There are currently no approved drugs targeting SNCA, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SNCA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1283', 'drugName': 'Prasinezumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'SNCA (ENSG00000145335)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5903', 'drugName': 'Cinpanemab', 'drugIsApproved': False, 'newLinkedTargets_string': 'SNCA (ENSG00000145335)', 'maxClin...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1344
Q1
Is SDC1 a druggable gene?
There are currently no approved drugs targeting SDC1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SDC1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_294', 'drugName': 'Indatuximab Ravtansine', 'drugIsApproved': False, 'newLinkedTargets_string': 'SDC1 (ENSG00000115884)', 'maxClinicalTrialPhase': 1}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.983
Q1
Is NISCH a druggable gene?
There is 1 drug, Moxonidine, that targets NISCH, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NISCH %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2347', 'drugName': 'Moxonidine', 'drugIsApproved': True, 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3253', 'drugName': 'Rilmenidine', 'drugIsApproved': False, 'newLinkedTargets_string': 'NISCH (ENSG00000010322)', 'maxClin...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.743
Q1
Is KCNC1 a druggable gene?
There are currently 5 approved drugs which target KCNC1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNC1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.193
Q1
Is CCR1 a druggable gene?
There are currently no approved drugs targeting CCR1, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CCR1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_194', 'drugName': 'Bms-817399', 'drugIsApproved': False, 'newLinkedTargets_string': 'CCR1 (ENSG00000163823)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_200', 'drugName': 'Ccx354', 'drugIsApproved': False, 'newLinkedTargets_string': 'CCR1 (ENSG00000163823)', 'maxClinicalTria...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.924
Q1
Is MYH7B a druggable gene?
There is 1 drug, Mavacamten, that targets MYH7B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MYH7B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1036', 'drugName': 'Mavacamten', 'drugIsApproved': True, 'newLinkedTargets_string': 'MYH7 (ENSG00000092054), MYH6 (ENSG00000197616), MYH7B (ENSG00000078814), MYL3 (ENSG00000160808), MYL2 (ENSG00000111245), MYL7 (ENSG00000106631), MYL4 (ENSG00000198336)', 'maxClinicalTrialPhase': 4}, {'UUID...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.458
Q1
Is FFAR2 a druggable gene?
There are currently no approved drugs targeting FFAR2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FFAR2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5482', 'drugName': 'Glpg-0974', 'drugIsApproved': False, 'newLinkedTargets_string': 'FFAR2 (ENSG00000126262)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.680
Q1
Is IL18R1 a druggable gene?
There are currently no approved drugs targeting IL18R1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL18R1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2219', 'drugName': 'Iboctadekin', 'drugIsApproved': False, 'newLinkedTargets_string': 'IL18RAP (ENSG00000115607), IL18R1 (ENSG00000115604)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.765
Q1
Is KCNJ3 a druggable gene?
There is 1 drug, Vernakalant, that targets KCNJ3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNJ3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_716', 'drugName': 'Vernakalant', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1386
Q1
Is SOAT1 a druggable gene?
There is 1 drug, Benfluorex, that targets SOAT1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SOAT1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5285', 'drugName': 'Benfluorex', 'drugIsApproved': True, 'newLinkedTargets_string': 'SOAT1 (ENSG00000057252)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6272', 'drugName': 'Pactimibe', 'drugIsApproved': False, 'newLinkedTargets_string': 'SOAT2 (ENSG00000167780), SOAT1 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.733
Q1
Is KCNA1 a druggable gene?
There are currently 5 approved drugs which target KCNA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.414
Q1
Is EPHA7 a druggable gene?
There is 1 drug, Vandetanib, that targets EPHA7, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EPHA7 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'drugIsApproved': True, 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (E...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.830
Q1
Is LTA a druggable gene?
There are currently no approved drugs targeting LTA, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%LTA %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_937', 'drugName': 'Pateclizumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'LTA (ENSG00000226979)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_5474', 'drugName': 'Baminercept', 'drugIsApproved': False, 'newLinkedTargets_string': 'LTA (ENSG00000226979), LTB (ENSG00...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.620
Q1
Is HTR2A a druggable gene?
There are currently 65 approved drugs which target HTR2A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HTR2A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4892', 'drugName': 'Carphenazine', 'drugIsApproved': True, 'newLinkedTargets_string': 'HTR2A (ENSG00000102468), HTR2C (ENSG00000147246), DRD2 (ENSG00000149295)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5097', 'drugName': 'Pimavanserin Tartrate', 'drugIsApproved': True, 'n...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.116
Q1
Is BLK a druggable gene?
There is 1 drug, Dasatinib, that targets BLK, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%BLK %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4602', 'drugName': 'Dasatinib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDGFRB (ENSG00000113721), FYN (ENSG00000010810), SRC (ENSG00000197122), LCK (ENSG00000182866), YES1 (ENSG00000176105), BLK (ENSG00000136573), HCK (ENSG00000101336), LYN (ENSG00000254087), FRK (ENSG000001118...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.419
Q1
Is EPHB4 a druggable gene?
There is 1 drug, Vandetanib, that targets EPHB4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EPHB4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1936', 'drugName': 'Vandetanib', 'drugIsApproved': True, 'newLinkedTargets_string': 'TEK (ENSG00000120156), ERBB2 (ENSG00000141736), EGFR (ENSG00000146648), ERBB4 (ENSG00000178568), ERBB3 (ENSG00000065361), EPHA2 (ENSG00000142627), EPHB2 (ENSG00000133216), EPHA5 (ENSG00000145242), EPHA4 (E...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1464
Q1
Is TNNI3 a druggable gene?
There are currently no approved drugs targeting TNNI3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNNI3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2198', 'drugName': 'Levosimendan', 'drugIsApproved': False, 'newLinkedTargets_string': 'PDE3A (ENSG00000172572), PDE3B (ENSG00000152270), TNNC1 (ENSG00000114854), TNNI3 (ENSG00000129991), TNNT2 (ENSG00000118194)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2199', 'drugName':...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.975
Q1
Is NDUFV1 a druggable gene?
There are currently 2 approved drugs which target NDUFV1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%NDUFV1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1888', 'drugName': 'Metformin Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'GPD2 (ENSG00000115159), MT-ND6 (ENSG00000198695), NDUFA10 (ENSG00000130414), NDUFS8 (ENSG00000110717), MT-ND4L (ENSG00000212907), NDUFA6 (ENSG00000184983), MT-ND1 (ENSG00000198888), NDUFB6 (EN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.608
Q1
Is HSD3B2 a druggable gene?
There is 1 drug, Trilostane, that targets HSD3B2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%HSD3B2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2278', 'drugName': 'Trilostane', 'drugIsApproved': True, 'newLinkedTargets_string': 'HSD3B2 (ENSG00000203859)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1537
Q1
Is XPO1 a druggable gene?
There is 1 drug, Selinexor, that targets XPO1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%XPO1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_58', 'drugName': 'Selinexor', 'drugIsApproved': True, 'newLinkedTargets_string': 'XPO1 (ENSG00000082898)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.91
Q1
Is ATP4B a druggable gene?
There are currently 14 approved drugs which target ATP4B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ATP4B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5144', 'drugName': 'Rabeprazole Sodium', 'drugIsApproved': True, 'newLinkedTargets_string': 'ATP4A (ENSG00000105675), ATP4B (ENSG00000186009)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4835', 'drugName': 'Pantoprazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'A...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.853
Q1
Is MAP3K13 a druggable gene?
There are currently no approved drugs targeting MAP3K13, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAP3K13 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1172
Q1
Is PSMC3 a druggable gene?
There are currently 4 approved drugs which target PSMC3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PSMC3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1469
Q1
Is TOP2A a druggable gene?
There are currently 15 approved drugs which target TOP2A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TOP2A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2612', 'drugName': 'Teniposide', 'drugIsApproved': True, 'newLinkedTargets_string': 'TOP2A (ENSG00000131747), TOP2B (ENSG00000077097)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_4763', 'drugName': 'Etoposide', 'drugIsApproved': True, 'newLinkedTargets_string': 'TOP2A (ENSG0...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.758
Q1
Is KCNH4 a druggable gene?
There are currently 5 approved drugs which target KCNH4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNH4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5118', 'drugName': 'Guanidine Hydrochloride', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNQ1 (ENSG00000053918), KCND3 (ENSG00000171385), KCNH2 (ENSG00000055118), KCNA2 (ENSG00000177301), KCNA1 (ENSG00000111262), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNA7 (ENSG000001...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.501
Q1
Is GABRB3 a druggable gene?
There are currently 67 approved drugs which target GABRB3, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GABRB3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2287', 'drugName': 'Clomethiazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256), GABRQ (ENSG00000268089), GABRA3 (ENSG000000116...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.12
Q1
Is ACHE a druggable gene?
There are currently 31 approved drugs which target ACHE, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ACHE %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1632', 'drugName': 'Galantamine Hydrobromide', 'drugIsApproved': True, 'newLinkedTargets_string': 'ACHE (ENSG00000087085)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_516', 'drugName': 'Pyridostigmine', 'drugIsApproved': True, 'newLinkedTargets_string': 'ACHE (ENSG0000008708...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.398
Q1
Is ELANE a druggable gene?
There is 1 drug, .Alpha.1-Proteinase Inhibitor Human, that targets ELANE, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ELANE %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2772', 'drugName': '.Alpha.1-Proteinase Inhibitor Human', 'drugIsApproved': True, 'newLinkedTargets_string': 'ELANE (ENSG00000197561)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3534', 'drugName': 'Sivelestat', 'drugIsApproved': False, 'newLinkedTargets_string': 'ELANE (ENS...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.286
Q1
Is COL11A2 a druggable gene?
There are currently 2 approved drugs which target COL11A2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%COL11A2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5818', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1072
Q1
Is PGA5 a druggable gene?
There is 1 drug, Sucralfate, that targets PGA5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PGA5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4142', 'drugName': 'Sucralfate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PGA5 (ENSG00000256713)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5872', 'drugName': 'Sucralfate', 'drugIsApproved': True, 'newLinkedTargets_string': 'PGA5 (ENSG00000256713)', 'maxClinical...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.695
Q1
Is IL2RG a druggable gene?
There are currently 4 approved drugs which target IL2RG, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL2RG %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2628', 'drugName': 'Basiliximab', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5681', 'drugName': 'Daclizumab', 'drugIsApproved': True, 'newLinkedTar...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1261
Q1
Is RPL37A a druggable gene?
There is 1 drug, Ataluren, that targets RPL37A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPL37A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3776', 'drugName': 'Ataluren', 'drugIsApproved': True, 'newLinkedTargets_string': 'RPSA (ENSG00000168028), RPS27 (ENSG00000177954), RPS6 (ENSG00000137154), RPS2 (ENSG00000140988), RPS3 (ENSG00000149273), RPS3A (ENSG00000145425), RPS4X (ENSG00000198034), RPS4Y1 (ENSG00000129824), RPS5 (ENSG...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1439
Q1
Is TLR9 a druggable gene?
There are currently 2 approved drugs which target TLR9, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TLR9 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3879', 'drugName': 'Hydroxychloroquine Sulfate', 'drugIsApproved': True, 'newLinkedTargets_string': 'TLR9 (ENSG00000239732), TLR7 (ENSG00000196664)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3878', 'drugName': 'Hydroxychloroquine Sulfate', 'drugIsApproved': True, 'newLinke...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.694
Q1
Is IL2RB a druggable gene?
There are currently 4 approved drugs which target IL2RB, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%IL2RB %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5633', 'drugName': 'Denileukin Diftitox', 'drugIsApproved': True, 'newLinkedTargets_string': 'IL2RA (ENSG00000134460), IL2RG (ENSG00000147168), IL2RB (ENSG00000100385), EEF2 (ENSG00000167658)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_2628', 'drugName': 'Basiliximab', 'dru...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.856
Q1
Is MAP3K9 a druggable gene?
There are currently no approved drugs targeting MAP3K9, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MAP3K9 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6091', 'drugName': 'Cep-1347', 'drugIsApproved': False, 'newLinkedTargets_string': 'MAP3K13 (ENSG00000073803), MAP3K12 (ENSG00000139625), MAP3K10 (ENSG00000130758), MAP3K9 (ENSG00000006432), MAP3K11 (ENSG00000173327)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_6088', 'drugN...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.161
Q1
Is CACNG2 a druggable gene?
There are currently 9 approved drugs which target CACNG2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CACNG2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_142', 'drugName': 'Gabapentin', 'drugIsApproved': True, 'newLinkedTargets_string': 'CACNA1H (ENSG00000196557), CACNA2D1 (ENSG00000153956), CACNA1C (ENSG00000151067), CACNA2D3 (ENSG00000157445), CACNA1S (ENSG00000081248), CACNA2D2 (ENSG00000007402), CACNA1D (ENSG00000157388), CACNA1A (ENSG0...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.900
Q1
Is MMP8 a druggable gene?
There are currently 4 approved drugs which target MMP8, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MMP8 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2398', 'drugName': 'Doxycycline Hyclate', 'drugIsApproved': True, 'newLinkedTargets_string': 'MMP13 (ENSG00000137745), MMP1 (ENSG00000196611), MMP7 (ENSG00000137673), MMP8 (ENSG00000118113)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3046', 'drugName': 'Doxycycline', 'drugI...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1219
Q1
Is RHD a druggable gene?
There are currently no approved drugs targeting RHD, but there are 4 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RHD %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3177', 'drugName': 'Roledumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RHD (ENSG00000187010)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_6033', 'drugName': 'Rozrolimupab', 'drugIsApproved': False, 'newLinkedTargets_string': 'RHD (ENSG00000187010)', 'maxClinica...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.259
Q1
Is CHRM1 a druggable gene?
There are currently 55 approved drugs which target CHRM1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CHRM1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2995', 'drugName': 'Glycopyrronium', 'drugIsApproved': True, 'newLinkedTargets_string': 'CHRM3 (ENSG00000133019), CHRM1 (ENSG00000168539)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_6050', 'drugName': 'Trihexyphenidyl Hydrochloride', 'drugIsApproved': True, 'newLinkedTarget...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.337
Q1
Is CXCL12 a druggable gene?
There are currently no approved drugs targeting CXCL12, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CXCL12 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3593', 'drugName': 'Olaptesed Pegol', 'drugIsApproved': False, 'newLinkedTargets_string': 'CXCL12 (ENSG00000107562)', 'maxClinicalTrialPhase': 2}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1443
Q1
Is TNFRSF10A a druggable gene?
There are currently no approved drugs targeting TNFRSF10A, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%TNFRSF10A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5538', 'drugName': 'Mapatumumab', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNFRSF10A (ENSG00000104689)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_638', 'drugName': 'Dulanermin', 'drugIsApproved': False, 'newLinkedTargets_string': 'TNFRSF10A (ENSG00000104689), T...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1045
Q1
Is PDE2A a druggable gene?
There are currently 2 approved drugs which target PDE2A, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PDE2A %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6107', 'drugName': 'Dipyridamole', 'drugIsApproved': True, 'newLinkedTargets_string': 'PDE5A (ENSG00000138735), PDE4A (ENSG00000065989), PDE3A (ENSG00000172572), PDE6H (ENSG00000139053), PDE6G (ENSG00000185527), PDE2A (ENSG00000186642), PDE7A (ENSG00000205268), PDE1A (ENSG00000115252), PDE...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.518
Q1
Is GHRHR a druggable gene?
There are currently 3 approved drugs which target GHRHR, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GHRHR %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2825', 'drugName': 'Tesamorelin', 'drugIsApproved': True, 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5465', 'drugName': 'Sermorelin Acetate', 'drugIsApproved': True, 'newLinkedTargets_string': 'GHRHR (ENSG00000106128)', '...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1021
Q1
Is OPRM1 a druggable gene?
There are currently 82 approved drugs which target OPRM1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%OPRM1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_1750', 'drugName': 'Methadone', 'drugIsApproved': True, 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3858', 'drugName': 'Diacetylmorphine', 'drugIsApproved': True, 'newLinkedTargets_string': 'OPRM1 (ENSG00000112038)', 'maxC...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.773
Q1
Is KCNMA1 a druggable gene?
There are currently no approved drugs targeting KCNMA1, but there are 3 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNMA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_2864', 'drugName': 'Flindokalner', 'drugIsApproved': False, 'newLinkedTargets_string': 'KCNMA1 (ENSG00000156113), KCNQ2 (ENSG00000075043), KCNQ3 (ENSG00000184156), KCNQ4 (ENSG00000117013), KCNQ5 (ENSG00000185760)', 'maxClinicalTrialPhase': 3}, {'UUID': 'DrugGeneTargets_v2_2869', 'drugName'...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1349
Q1
Is SEM1 a druggable gene?
There are currently 4 approved drugs which target SEM1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%SEM1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_559', 'drugName': 'Bortezomib', 'drugIsApproved': True, 'newLinkedTargets_string': 'PSMD1 (ENSG00000173692), PSMB2 (ENSG00000126067), PSMB1 (ENSG00000008018), PSMB5 (ENSG00000100804), PSMB8 (ENSG00000204264), PSMB9 (ENSG00000240065), PSMB6 (ENSG00000142507), PSMD14 (ENSG00000115233), PSMA1...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.766
Q1
Is KCNJ5 a druggable gene?
There is 1 drug, Vernakalant, that targets KCNJ5, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%KCNJ5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_716', 'drugName': 'Vernakalant', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCND3 (ENSG00000171385), KCNA5 (ENSG00000130037), KCNJ3 (ENSG00000162989), KCNJ5 (ENSG00000120457), KCNH2 (ENSG00000055118), SCN5A (ENSG00000183873)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1127
Q1
Is PRKAB2 a druggable gene?
There are currently no approved drugs targeting PRKAB2, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%PRKAB2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5888', 'drugName': 'Acadesine', 'drugIsApproved': False, 'newLinkedTargets_string': 'PRKAA2 (ENSG00000162409), PRKAB2 (ENSG00000131791), PRKAG1 (ENSG00000181929), PRKAG2 (ENSG00000106617), PRKAB1 (ENSG00000111725), PRKAA1 (ENSG00000132356), PRKAG3 (ENSG00000115592)', 'maxClinicalTrialPhase...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.524
Q1
Is GLRA1 a druggable gene?
There are currently 6 approved drugs which target GLRA1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%GLRA1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5597', 'drugName': 'Isoflurane', 'drugIsApproved': True, 'newLinkedTargets_string': 'KCNK10 (ENSG00000100433), KCNK9 (ENSG00000169427), GABRA1 (ENSG00000022355), GABRB2 (ENSG00000145864), GABRG2 (ENSG00000113327), GABRB3 (ENSG00000166206), GABRA4 (ENSG00000109158), GABRG3 (ENSG00000182256)...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.23
Q1
Is ADH4 a druggable gene?
There is 1 drug, Nitrefazole, that targets ADH4, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%ADH4 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_6344', 'drugName': 'Nitrefazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'ADH1A (ENSG00000187758), ADH4 (ENSG00000198099), ADH1B (ENSG00000196616), ADH1C (ENSG00000248144), ADH7 (ENSG00000196344), ADH5 (ENSG00000197894), ADH6 (ENSG00000172955)', 'maxClinicalTrialPhase': 4}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.358
Q1
Is DGAT1 a druggable gene?
There are currently no approved drugs targeting DGAT1, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%DGAT1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3433', 'drugName': 'Pradigastat', 'drugIsApproved': False, 'newLinkedTargets_string': 'DGAT1 (ENSG00000185000)', 'maxClinicalTrialPhase': 3}]
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.1304
Q1
Is RPS6KA3 a druggable gene?
There are currently no approved drugs targeting RPS6KA3, but there is 1 drug in a clinical trial indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%RPS6KA3 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3347', 'drugName': 'Tas0612', 'drugIsApproved': False, 'newLinkedTargets_string': 'RPS6KB2 (ENSG00000175634), RPS6KB1 (ENSG00000108443), AKT2 (ENSG00000105221), AKT3 (ENSG00000117020), AKT1 (ENSG00000142208), RPS6KA3 (ENSG00000177189), RPS6KA2 (ENSG00000071242), RPS6KA6 (ENSG00000072133), ...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.342
Q1
Is CYP11A1 a druggable gene?
There are currently 3 approved drugs which target CYP11A1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CYP11A1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_3930', 'drugName': 'Levoketoconazole', 'drugIsApproved': True, 'newLinkedTargets_string': 'CYP11B1 (ENSG00000160882), CYP11B2 (ENSG00000179142), CYP17A1 (ENSG00000148795), CYP11A1 (ENSG00000140459)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_3932', 'drugName': 'Levoketocona...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.433
Q1
Is EZH2 a druggable gene?
There are currently 2 approved drugs which target EZH2, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%EZH2 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4960', 'drugName': 'Tazemetostat Hydrobromide', 'drugIsApproved': True, 'newLinkedTargets_string': 'EZH2 (ENSG00000106462)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_1211', 'drugName': 'Tazemetostat', 'drugIsApproved': True, 'newLinkedTargets_string': 'EZH2 (ENSG0000010646...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.475
Q1
Is FN1 a druggable gene?
There is 1 drug, Ocriplasmin, that targets FN1, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%FN1 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5819', 'drugName': 'Ocriplasmin', 'drugIsApproved': True, 'newLinkedTargets_string': 'FN1 (ENSG00000115414), COL1A2 (ENSG00000164692), COL1A1 (ENSG00000108821), COL2A1 (ENSG00000139219), COL3A1 (ENSG00000168542), COL4A1 (ENSG00000187498), COL5A1 (ENSG00000130635), COL6A1 (ENSG00000142156),...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.219
Q1
Is CD5 a druggable gene?
There are currently no approved drugs targeting CD5, but there are 2 drugs in clinical trials indicating that it may be a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%CD5 %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_4551', 'drugName': 'Telimomab Aritox', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD5 (ENSG00000110448)', 'maxClinicalTrialPhase': 2}, {'UUID': 'DrugGeneTargets_v2_4169', 'drugName': 'Zolimomab Aritox', 'drugIsApproved': False, 'newLinkedTargets_string': 'CD5 (ENSG00000110448)', ...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target
Q1.916
Q1
Is MTNR1B a druggable gene?
There are currently 4 approved drugs which target MTNR1B, indicating that it is a druggable gene.
SELECT DISTINCT UUID, drugName, drugIsApproved, newLinkedTargets_string, maxClinicalTrialPhase FROM `{project_id}.{dataset_name}.DrugGeneTargets_ComprehensiveAnnotations_updated` WHERE newLinkedTargets_string LIKE "%MTNR1B %" ORDER BY maxClinicalTrialPhase DESC LIMIT 100
[{'UUID': 'DrugGeneTargets_v2_5938', 'drugName': 'Ramelteon', 'drugIsApproved': True, 'newLinkedTargets_string': 'MTNR1A (ENSG00000168412), MTNR1B (ENSG00000134640)', 'maxClinicalTrialPhase': 4}, {'UUID': 'DrugGeneTargets_v2_5737', 'drugName': 'Melatonin', 'drugIsApproved': True, 'newLinkedTargets_string': 'MTNR1A (ENS...
general
Similarity Search, Order By, Distinct
Approval Status, Genetic Target