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time-dependent inhibition of bacterial beta-lactamases by clavulanic acid and sulbactam has extended the use of penicillins which are highly susceptible to beta-lactamase inactivation .
NA
{ "id": "C0038665", "name": "sulbactam", "pos": [ 78, 87 ] }
{ "id": "C0030842", "name": "penicillins", "pos": [ 112, 123 ] }
digoxin interacts with other drugs at any stage of absorption ( e.g . cholestyramine ) , distribution ( e.g . quinidine ) , metabolism ( e.g . phenytoin ) or elimination ( e.g . diltiazem ) .
NA
{ "id": "C0025519", "name": "metabolism", "pos": [ 124, 134 ] }
{ "id": "C0221102", "name": "elimination", "pos": [ 158, 169 ] }
these observations indicate that both renal and metabolic elimination processes for theophylline are less active in the normal elderly .
NA
{ "id": "C0025519", "name": "metabolic", "pos": [ 48, 57 ] }
{ "id": "C0221102", "name": "elimination", "pos": [ 58, 69 ] }
the authors describe the ct findings in 10 cases of pulmonary aspergillosis which include allergic bronchopulmonary aspergillosis , aspergilloma and invasive pulmonary aspergillosis .
NA
{ "id": "C2350529", "name": "pulmonary aspergillosis", "pos": [ 52, 75 ] }
{ "id": "C0276653", "name": "invasive", "pos": [ 149, 157 ] }
assay of von willebrand 's disease ( vwd ) plasmas with the elisa for vwf : ag demonstrated reduced levels of this antigen in type i vwd , normal levels in type iia , and a severe reduction of vwf : ag in type iii vwd .
NA
{ "id": "C0042974", "name": "von willebrand 's disease", "pos": [ 9, 34 ] }
{ "id": "C1264041", "name": "type", "pos": [ 205, 209 ] }
fracture involving both the enamel and the dentine was the most commonly recorded class of trauma ( 42.7 % of cases ) .
NA
{ "id": "C0016658", "name": "fracture", "pos": [ 0, 8 ] }
{ "id": "C0043251", "name": "trauma", "pos": [ 91, 97 ] }
trauma to the maxillary dental arch occurred most frequently at home , while trauma to more than one tooth ( multiple trauma ) occurred most commonly at school .
NA
{ "id": "C0043251", "name": "trauma", "pos": [ 0, 6 ] }
{ "id": "C0026771", "name": "multiple", "pos": [ 109, 117 ] }
following voltage activation of the passive cl- permeability of the mitochondria-rich ( m.r . ) cells sulfate flux-ratio increased to a value predicted from the ussing flux-ratio equation for a monovalent anion .
NA
{ "id": "C0038720", "name": "sulfate", "pos": [ 102, 109 ] }
{ "id": "C0003075", "name": "anion", "pos": [ 205, 210 ] }
the effect of intraperitoneally administered gold thioglucose on growth , food consumption and accumulation of gold in various organs of the chicken ( gallus domesticus ) .
NA
{ "id": "C0018033", "name": "gold thioglucose", "pos": [ 45, 61 ] }
{ "id": "C0018026", "name": "gold", "pos": [ 111, 115 ] }
gold detected in blood , heart , liver , gallbladder , spleen , proventriculus , gizzard , duodenum , kidney , pectoral muscle , small intestine , lung and brain of the dead chickens accumulated most highly in heart and followed by spleen , but in the surviving chicken a little gold was only found in liver , spleen and kidney of some gtg-treated chickens .
NA
{ "id": "C0018026", "name": "gold", "pos": [ 0, 4 ] }
{ "id": "C0018033", "name": "gtg", "pos": [ 336, 339 ] }
hence , the inhibition of this rate may be an important function underlying the complement-mediated processing of immune complexes , and a decreased ability of the complement system to mediate this process in the presence of c4b1 , in contrast to c4a3 , could explain , at least in part , the association between the c4a-null phenotype and autoimmune diseases such as systemic lupus erythematosus .
NA
{ "id": "C0004364", "name": "autoimmune diseases", "pos": [ 340, 359 ] }
{ "id": "C0024141", "name": "systemic lupus erythematosus", "pos": [ 368, 396 ] }
maximal chemotaxis was achieved with a concentration of 5 ng/ml for limb bud cells and as low as 15 pg/ml for muscle-derived fibroblasts .
NA
{ "id": "C0007634", "name": "cells", "pos": [ 77, 82 ] }
{ "id": "C0016030", "name": "fibroblasts", "pos": [ 125, 136 ] }
the binding of the lectins suggested that eep is composed of proteins having galactose or n-acetylgalactosamine groups as well as fucose residues .
NA
{ "id": "C0023206", "name": "lectins", "pos": [ 19, 26 ] }
{ "id": "C0033684", "name": "proteins", "pos": [ 61, 69 ] }
chronological distribution of this intermediate filament-associated protein ( ifap ) and vimentin during fetal development of the cornea in rabbit was analysed immunohistochemically .
NA
{ "id": "C0021769", "name": "intermediate", "pos": [ 35, 47 ] }
{ "id": "C0042666", "name": "vimentin", "pos": [ 89, 97 ] }
during an early stage of corneal development ( day 13 of gestation ) , both this ifap and vimentin were present in the stromal cells in the presumptive corneal region .
NA
{ "id": "C0021769", "name": "ifap", "pos": [ 81, 85 ] }
{ "id": "C0042666", "name": "vimentin", "pos": [ 90, 98 ] }
at day 17 and 21 , the corneal endothelial layer was developed and contained both the ifap and vimentin .
NA
{ "id": "C0021769", "name": "ifap", "pos": [ 86, 90 ] }
{ "id": "C0042666", "name": "vimentin", "pos": [ 95, 103 ] }
however , in the corneal stromal cells , the concentration of ifap ( based on the densities of the immunostaining reaction ) progressively decreased during the later stages of fetal development ( day 24 to day 28 ) , while relative concentrations of vimentin were not reduced significantly .
NA
{ "id": "C0021769", "name": "ifap", "pos": [ 62, 66 ] }
{ "id": "C0042666", "name": "vimentin", "pos": [ 250, 258 ] }
in the corneal stromal cells in the adult rabbit , the ifap was not detectable while vimentin was still present .
NA
{ "id": "C0021769", "name": "ifap", "pos": [ 55, 59 ] }
{ "id": "C0042666", "name": "vimentin", "pos": [ 85, 93 ] }
segregation of the x-linked mink markers alpha-galactosidase ( gla ) , phosphoglycerate kinase-1 ( pgk1 ) , hypoxanthine phosphoribosyltransferase ( hprt ) , and glucose-6-phosphate dehydrogenase ( g6pd ) was analyzed in hybrids of gamma-irradiated mink fibroblasts and chinese hamster cells and in hybrids of nonirradiated mink fibroblasts and mouse hepatoma cells .
NA
{ "id": "C0007634", "name": "cells", "pos": [ 286, 291 ] }
{ "id": "C0016030", "name": "fibroblasts", "pos": [ 329, 340 ] }
both biochemical and genetic evidence therefore indicate independence of dbh from the pterin-dependent aromatic amino acid hydroxylases of the neurotransmitter pathways .
NA
{ "id": "C0013032", "name": "dbh", "pos": [ 73, 76 ] }
{ "id": "C0020364", "name": "hydroxylases", "pos": [ 123, 135 ] }
autopsy showed enlarged heart , normal coronary arteries , right ventricular septal hypertrophy , quadricuspid pulmonary valve , accessory tricuspid valve , and a moderately elongated and thickened mitral valve .
NA
{ "id": "C0018800", "name": "enlarged heart", "pos": [ 15, 29 ] }
{ "id": "C0162770", "name": "right ventricular", "pos": [ 59, 76 ] }
epac showed higher and longer-lasting erythromycin levels in serum , sputum and pure bronchial mucus than es .
NA
{ "id": "C0014806", "name": "erythromycin", "pos": [ 38, 50 ] }
{ "id": "C0059566", "name": "es", "pos": [ 106, 108 ] }
the isolates were tested against netilmicin , piperacillin , cefoxitin , cefuroxime , and cefotaxime , alone and in different combinations .
NA
{ "id": "C0007562", "name": "cefuroxime", "pos": [ 73, 83 ] }
{ "id": "C0007554", "name": "cefotaxime", "pos": [ 90, 100 ] }
the in vitro activity of fleroxacin ( ro 23-6240 ) against 441 bacterial isolates was compared with those of ciprofloxacin , ofloxacin , amoxycillin , cefadroxil , cefuroxime and tobramycin .
NA
{ "id": "C0085161", "name": "fleroxacin", "pos": [ 25, 35 ] }
{ "id": "C0008809", "name": "ciprofloxacin", "pos": [ 109, 122 ] }
ciprofloxacin showed the highest activity against the enterobacteriaceae , 95 % of the isolates were inhibited by 0.06 mg/l , but fleroxacin and ofloxacin were also highly active ( mic 90 % = 0.5 and 0.25 mg/l , respectively ) .
NA
{ "id": "C0008809", "name": "ciprofloxacin", "pos": [ 0, 13 ] }
{ "id": "C0085161", "name": "fleroxacin", "pos": [ 130, 140 ] }
ciprofloxacin was the most active agent against pseudomonas aeruginosa ( mic 90 % = 0.12 mg/l ) , whereas the activities of fleroxacin and ofloxacin were more variable .
NA
{ "id": "C0008809", "name": "ciprofloxacin", "pos": [ 0, 13 ] }
{ "id": "C0085161", "name": "fleroxacin", "pos": [ 124, 134 ] }
putrescine levels increased in the mononuclear cells of all patients , cellular spermidine levels increased in 4 and cellular spermine levels increased in 5 patients .
NA
{ "id": "C0034170", "name": "putrescine", "pos": [ 0, 10 ] }
{ "id": "C0037871", "name": "levels", "pos": [ 135, 141 ] }
putrescine levels increased in the mononuclear cells of all patients , cellular spermidine levels increased in 4 and cellular spermine levels increased in 5 patients .
NA
{ "id": "C0037871", "name": "levels", "pos": [ 11, 17 ] }
{ "id": "C0037874", "name": "levels", "pos": [ 135, 141 ] }
comparison of two cell lines such as friend murine erythroleukemia cells ( melc ) and fibroblasts fr3t3 cells has shown that this analysis can be used for cell-cycle characterization of a given cell line .
NA
{ "id": "C0007634", "name": "cells", "pos": [ 67, 72 ] }
{ "id": "C0016030", "name": "fibroblasts", "pos": [ 86, 97 ] }
and 3 ) using the two antibodies ( mab b72.3 and mab anti-caa ) , a malignancy ratio was obtained that determined malignancy risk for individual polyps .
NA
{ "id": "C0003241", "name": "antibodies", "pos": [ 22, 32 ] }
{ "id": "C0003250", "name": "mab", "pos": [ 49, 52 ] }
a diagnosis of turcot 's syndrome should be restricted to those patients with familial polyposis coli associated with gliomas or medulloblastomas .
NA
{ "id": "C0017638", "name": "gliomas", "pos": [ 118, 125 ] }
{ "id": "C0025149", "name": "medulloblastomas", "pos": [ 129, 145 ] }
solitary rectal ulcer syndrome ( srus ) is sufficiently uncommon that the clinician or general pathologist may lack familiarity with the disorder and may confuse it with other inflammatory bowel diseases .
NA
{ "id": "C0039082", "name": "syndrome", "pos": [ 22, 30 ] }
{ "id": "C0012634", "name": "disorder", "pos": [ 137, 145 ] }
the proximal small intestinal mucosa of rats fed lectin showed gradual increases in protein and dna contents throughout the experimental period .
NA
{ "id": "C0023206", "name": "lectin", "pos": [ 49, 55 ] }
{ "id": "C0033684", "name": "protein", "pos": [ 84, 91 ] }
in contrast , intravenous infusion of nahco3 ( 3 mmol/kg/hr ) ameliorated the acid-base imbalance caused by he , and significantly restored the impaired hco3- responses induced by he but not by indomethacin .
NA
{ "id": "C0074722", "name": "nahco3", "pos": [ 38, 44 ] }
{ "id": "C0005367", "name": "hco3", "pos": [ 153, 157 ] }
clinical expressions of hyperfunctional adrenocortical syndromes include cushing 's syndrome , primary hyperaldosteronism , and the adrenogenital syndrome .
NA
{ "id": "C0001622", "name": "hyperfunctional adrenocortical", "pos": [ 24, 54 ] }
{ "id": "C0010481", "name": "cushing 's", "pos": [ 73, 83 ] }
2 ) maternal factor ( s ) affected cytochrome p-450-specific content and the activities of acetanilide hydroxylase and aryl hydrocarbon hydroxylase but not of testosterone 15 alpha- and 16 alpha-hydroxylases or nadph-cytochrome c reductase ;
NA
{ "id": "C0010762", "name": "cytochrome p-450", "pos": [ 35, 51 ] }
{ "id": "C0003927", "name": "aryl hydrocarbon hydroxylase", "pos": [ 119, 147 ] }
among the most prominent features of this interaction is the activation and high-level expression of the genes encoding the major myelin proteins p0 and myelin basic protein ( mbp ) .
NA
{ "id": "C0026972", "name": "myelin proteins", "pos": [ 130, 145 ] }
{ "id": "C0014063", "name": "myelin basic protein", "pos": [ 153, 173 ] }
bismuth intoxication ( encephalopathy ) has been reported with prolonged administration of bismuth salts , and there has been 1 report of similar intoxication in a patient receiving unusually high doses of cbs for a prolonged period .
NA
{ "id": "C0005642", "name": "bismuth", "pos": [ 0, 7 ] }
{ "id": "C0106556", "name": "cbs", "pos": [ 206, 209 ] }
milrinone is a bipyridine derivative of amrinone , with approximately 10 to 75 times greater positive inotropic potency , and separate direct vasodilatory properties .
NA
{ "id": "C0128513", "name": "milrinone", "pos": [ 0, 9 ] }
{ "id": "C0002697", "name": "amrinone", "pos": [ 40, 48 ] }
preliminary long term studies suggest that tolerance to the haemodynamic effects of milrinone does not occur , and that the drug is well tolerated and without the thrombocytopenic effects , fever and gastrointestinal complications observed with amrinone .
NA
{ "id": "C0128513", "name": "milrinone", "pos": [ 84, 93 ] }
{ "id": "C0002697", "name": "amrinone", "pos": [ 245, 253 ] }
all of the fluoroquinolones except ofloxacin are associated with a variable increase in the serum concentration of theophylline , warfarin and caffeine .
NA
{ "id": "C0949665", "name": "fluoroquinolones", "pos": [ 11, 27 ] }
{ "id": "C0028902", "name": "ofloxacin", "pos": [ 35, 44 ] }
[ hypercholesterolemia and the diagnosis and management of hyper- lipidemia in adults . recommendations of the working groups of the finnish society of internal medicine and the finnish cardiology society ] .
NA
{ "id": "C0020443", "name": "hypercholesterolemia", "pos": [ 2, 22 ] }
{ "id": "C0020473", "name": "lipidemia", "pos": [ 66, 75 ] }
the ultrastructure characteristics of leaves during the development of cell organelles , in the `` '' greening process '' '' of spring , have been studied in pollutant-tolerant and susceptible individuals of beech ( fagus silvatica ) and hornbeam ( carpinus betulus ) in an area polluted with so2 ( the main pollutant may reach 0.06-2.72 mg/m3 ) , heavy metals , and other gases discharged by non-iron metal processing factories .
NA
{ "id": "C0347988", "name": ", heavy meta", "pos": [ 346, 358 ] }
{ "id": "C0302583", "name": "n-ir", "pos": [ 395, 399 ] }
when allowance was made for cytoplasmic na concentration , the pump rate was slower in younger ( 12 months and under ) normal children than in older children .
NA
{ "id": "C0008059", "name": "children", "pos": [ 126, 134 ] }
{ "id": "C1455726", "name": "older children", "pos": [ 143, 157 ] }
the accumulation of the two extracellular matrix proteins in the medium was differentially affected by fetal calf serum and tgf-beta and the increase was in both cases higher for tenascin .
NA
{ "id": "C0079323", "name": "extracellular matrix", "pos": [ 28, 48 ] }
{ "id": "C0076088", "name": "tenascin", "pos": [ 179, 187 ] }
the rat m1 muscarinic receptor gene was cloned and expressed in a rat cell line lacking endogenous muscarinic receptors .
NA
{ "id": "C0531859", "name": "m1", "pos": [ 8, 10 ] }
{ "id": "C0034826", "name": "muscarinic receptors", "pos": [ 99, 119 ] }
phorbol ester ( pma ) modulated the binding affinity of wild-type and mutant receptors in a similar manner .
NA
{ "id": "C0031586", "name": "phorbol", "pos": [ 0, 7 ] }
{ "id": "C0039654", "name": "pma", "pos": [ 16, 19 ] }
despite the similarities shared by all lamin proteins , the lamin liii sequence neither possesses the features diagnostic for either type-a or type-b lamins nor does it show greater sequence similarity to one of the lamin types than to the other and thus it may represent a third type of lamin protein which may reflect its special function in oogenesis and early development .
NA
{ "id": "C0064635", "name": "lamin", "pos": [ 39, 44 ] }
{ "id": "C0125258", "name": "a", "pos": [ 359, 360 ] }
the sequence gly-x-gly-lys-thr , believed to be involved in the interaction with purine nucleotides in proteins that bind and hydrolyze the nucleotides , is present in the rad3 primary structure between amino acids 45 and 49 .
NA
{ "id": "C0034137", "name": "purine nucleotides", "pos": [ 81, 99 ] }
{ "id": "C0028630", "name": "nucleotides", "pos": [ 140, 151 ] }
to demonstrate that the 3'-domain of rna c determines virulence , a chimeric satellite was constructed composed mostly of the 5'-domain of the avirulent satellite ( rna f ) and the 3'-domain of the virulent satellite ( rna c ) .
NA
{ "id": "C0035668", "name": "rna", "pos": [ 37, 40 ] }
{ "id": "C0074081", "name": "satellite", "pos": [ 207, 216 ] }
between 2.5 % and 4.9 % of antibodies were obtained from two different anti-fibronectin sera indicating that this region represents an antigenic epitope in native fibronectin .
NA
{ "id": "C0003320", "name": "antigenic", "pos": [ 135, 144 ] }
{ "id": "C0003316", "name": "epitope", "pos": [ 145, 152 ] }
in the insulin-secreting beta cell line rin m 5f , galanin , a newly discovered ubiquitous neuropeptide , inhibited , by 50 % , the stimulation of insulin release induced by gastric inhibitory polypeptide ( gip ) or forskolin , i.e . two camp-generating effectors .
NA
{ "id": "C0060993", "name": "galanin", "pos": [ 51, 58 ] }
{ "id": "C0027895", "name": "neuropeptide", "pos": [ 91, 103 ] }
by the identification of mannobiosido- , and mannotriosido-di-n-acetylchitobiose mixed with n-acetyl-lactosaminic and oligomannosidic-types oligosaccharides , we demonstrate the high microheterogeneity of the glycans presents in the neutral fraction of this glycoprotein and suggest that ovomucoid glycosylation uses several pathways .
NA
{ "id": "C0028959", "name": "oligosaccharides", "pos": [ 140, 156 ] }
{ "id": "C0032594", "name": "glycans", "pos": [ 209, 216 ] }
gel-filtered human platelets that had been pre-labelled with [ 32p ] pi were stimulated with thrombin , ionomycin or the phorbol ester 12-o-tetradecanoyl-phorbol 13-acetate ( tpa ) .
NA
{ "id": "C0031586", "name": "phorbol ester", "pos": [ 121, 134 ] }
{ "id": "C0039654", "name": "12-o-tetradecanoyl-phorbol 13-acetate", "pos": [ 135, 172 ] }
the in vitro activity of the new oral macrolide azithromycin was compared with that of erythromycin against gram-positive and gram-negative aerobic and anaerobic bacteria .
NA
{ "id": "C0052796", "name": "azithromycin", "pos": [ 48, 60 ] }
{ "id": "C0014806", "name": "erythromycin", "pos": [ 87, 99 ] }
azithromycin was more active than erythromycin against haemophilus influenzae ( mic90 1 microgram/ml ) and neisseria gonorrhoeae .
NA
{ "id": "C0052796", "name": "azithromycin", "pos": [ 0, 12 ] }
{ "id": "C0014806", "name": "erythromycin", "pos": [ 34, 46 ] }
susceptibility testing of clinical isolates of several gram-negative and gram-positive species showed ly163892 to be more active than cefaclor and cephalexin .
NA
{ "id": "C0007537", "name": "cefaclor", "pos": [ 134, 142 ] }
{ "id": "C0007716", "name": "cephalexin", "pos": [ 147, 157 ] }
in vitro activity of azithromycin and erythromycin against organisms associated with bacterial vaginosis and chancroid .
NA
{ "id": "C0052796", "name": "azithromycin", "pos": [ 21, 33 ] }
{ "id": "C0014806", "name": "erythromycin", "pos": [ 38, 50 ] }
the in vitro activity of the new macrolide azithromycin and erythromycin against haemophilus ducreyi , gardnerella vaginalis , bacteroides spp . and mobiluncus spp . was compared .
NA
{ "id": "C0052796", "name": "azithromycin", "pos": [ 43, 55 ] }
{ "id": "C0014806", "name": "erythromycin", "pos": [ 60, 72 ] }
collectively , 62 % of all bacteroides strains were susceptible to erythromycin ( mic 1 mg/1 ) and 74 % were susceptible to azithromycin .
NA
{ "id": "C0014806", "name": "erythromycin", "pos": [ 67, 79 ] }
{ "id": "C0052796", "name": "azithromycin", "pos": [ 124, 136 ] }
the beta-lactams ( penicillin , ampicillin , cefoxitin and cephalexin ) , macrolides ( erythromycin and azithromycin ) , quinolones ( ciprofloxacin and ofloxacin ) , nitrofurans , gentamicin and tetracycline all had mic90 values of less than or equal to 0.5 mg/l .
NA
{ "id": "C0282215", "name": "beta-lactams", "pos": [ 4, 16 ] }
{ "id": "C0030842", "name": "penicillin", "pos": [ 19, 29 ] }
the beta-lactams ( penicillin , ampicillin , cefoxitin and cephalexin ) , macrolides ( erythromycin and azithromycin ) , quinolones ( ciprofloxacin and ofloxacin ) , nitrofurans , gentamicin and tetracycline all had mic90 values of less than or equal to 0.5 mg/l .
NA
{ "id": "C0014806", "name": "erythromycin", "pos": [ 87, 99 ] }
{ "id": "C0052796", "name": "azithromycin", "pos": [ 104, 116 ] }
antibodies against following peroxisomal enzymes : catalase , urate oxidase , alpha-hydroxy acid oxidase , acyl-coa oxidase , bifunctional enzyme ( hydratase-dehydrogenase ) and thiolase , were raised in rabbits , and their monospecificities were confirmed by immunoblotting .
NA
{ "id": "C0041931", "name": "urate oxidase", "pos": [ 62, 75 ] }
{ "id": "C0030016", "name": "dehydrogenase", "pos": [ 158, 171 ] }
assuming carbohydrate-protein interactions play important physiological roles here , then specific carbohydrate-binding proteins should be prominent components of this microvasculature , in addition to the wealth of endogenous glycoconjugates reported by other authors .
NA
{ "id": "C0007004", "name": "carbohydrate", "pos": [ 9, 21 ] }
{ "id": "C0017906", "name": "glycoconjugates", "pos": [ 227, 242 ] }
platelet viability ( aggregation , migration , recovery ) after radiolabelling from hypercholesterolemics using various tracers ( oxine , oxine-sulphate , tropolone , mpo ) .
NA
{ "id": "C0000665", "name": "oxine", "pos": [ 130, 135 ] }
{ "id": "C0086760", "name": "oxine-sulphate", "pos": [ 138, 152 ] }
a total of 100 patients receiving fluphenazine ( fpz ) decanoate for at least 12 months ( 96 schizophrenics and 4 other diagnoses ) were investigated for plasma levels of fpz and prolactin on the day of injection ( day 0 ) and 7 days later ( day 7 ) .
NA
{ "id": "C0060580", "name": "fluphenazine", "pos": [ 34, 46 ] }
{ "id": "C0016368", "name": "fpz", "pos": [ 171, 174 ] }
adenosine 5'-monophosphate ( amp ) , adenosine 5'-diphosphate ( adp ) and adenosine 5'-triphosphate ( atp ) , injected intraperitoneally into tumor-bearing ( s.c. implanted footpad tumors ) mice , exhibited significant anticancer activity .
NA
{ "id": "C0001413", "name": "adenosine 5", "pos": [ 0, 11 ] }
{ "id": "C0001459", "name": "adenosine 5", "pos": [ 74, 85 ] }
adenosine 5'-monophosphate ( amp ) , adenosine 5'-diphosphate ( adp ) and adenosine 5'-triphosphate ( atp ) , injected intraperitoneally into tumor-bearing ( s.c. implanted footpad tumors ) mice , exhibited significant anticancer activity .
NA
{ "id": "C0001413", "name": "adenosine 5", "pos": [ 0, 11 ] }
{ "id": "C0001480", "name": "adenosine", "pos": [ 74, 83 ] }
intraperitoneal injections of 1 ml of 50 mm amp , adp or atp in saline , yielded elevated blood and plasma levels of atp which lasted for several hours in both strains of mice .
NA
{ "id": "C0001413", "name": "amp", "pos": [ 44, 47 ] }
{ "id": "C0001459", "name": "adp", "pos": [ 50, 53 ] }
intraperitoneal injections of 1 ml of 50 mm amp , adp or atp in saline , yielded elevated blood and plasma levels of atp which lasted for several hours in both strains of mice .
NA
{ "id": "C0001413", "name": "amp", "pos": [ 44, 47 ] }
{ "id": "C0001480", "name": "atp", "pos": [ 117, 120 ] }
the pharmacokinetics of disopyramide was studied in 15 patients with renal dysfunction ( 4 with pyelonephritis , 7 with glomerular nephritis and 4 with interstitial nephritis ) .
NA
{ "id": "C0034186", "name": "pyelonephritis", "pos": [ 96, 110 ] }
{ "id": "C0027707", "name": "interstitial nephritis", "pos": [ 152, 174 ] }
the effects of optical isomers of fenfluramine and their metabolites , d- and l-norfenfluramine on the serotonergic system were studied in the nucleus accumbens and hippocampus of freely moving rats by in vivo voltammetry .
NA
{ "id": "C0015827", "name": "fenfluramine", "pos": [ 34, 46 ] }
{ "id": "C0028362", "name": "norfenfluramine", "pos": [ 80, 95 ] }
both isomers and the metabolites induced a slow , sustained decrease in 5hiaa but only d-fenfluramine and its metabolite , d-norfenfluramine , increased the 5hiaa levels in nucleus accumbens shortly after injection , the increase being greater after the metabolite .
NA
{ "id": "C0015827", "name": "fenfluramine", "pos": [ 89, 101 ] }
{ "id": "C0028362", "name": "norfenfluramine", "pos": [ 125, 140 ] }
intravenous injection of the synthetic trh analog , mk-771 , to anesthetised cats raised the blood pressure by a central mechanism , i.e . by activating the outflow of sympathetic stimuli from the cns to the periphery and raising the plasma concentration of adrenaline and noradrenaline .
NA
{ "id": "C0014563", "name": "adrenaline", "pos": [ 258, 268 ] }
{ "id": "C0028351", "name": "noradrenaline", "pos": [ 273, 286 ] }
we find that the levels of each mrna analysed appear to cycle in the +/+ adult retina , with the greatest amount of opsin and the three subunits of g-protein mrnas occurring just before light onset and the greatest amount of 48-kda protein mrna occurring just before lights off .
NA
{ "id": "C0599220", "name": "subunits", "pos": [ 136, 144 ] }
{ "id": "C0033684", "name": "protein", "pos": [ 232, 239 ] }
during the western blot analyses , the antiserum exhibited specific immuno-reaction with alpha-crystallin and 20-kda gamma-crystallin species and with degraded polypeptides among various human lens crystallins tested .
NA
{ "id": "C0002257", "name": "alpha-crystallin", "pos": [ 89, 105 ] }
{ "id": "C0010422", "name": "crystallins", "pos": [ 198, 209 ] }
during the western blot analyses , the antiserum exhibited specific immuno-reaction with alpha-crystallin and 20-kda gamma-crystallin species and with degraded polypeptides among various human lens crystallins tested .
NA
{ "id": "C0017030", "name": "gamma-crystallin", "pos": [ 117, 133 ] }
{ "id": "C0010422", "name": "crystallins", "pos": [ 198, 209 ] }
in order to examine the cellular basis of the low production of bpa by pha-stimulated cord blood mononuclear cells in the context of the functional immaturity of t cells or monocytes , we studied bpa production by t cells or monocytes from cord blood and adult peripheral blood .
NA
{ "id": "C0007634", "name": "cellular", "pos": [ 24, 32 ] }
{ "id": "C1321301", "name": "blood mononuclear cells", "pos": [ 91, 114 ] }
there are two major hypotheses proposed to explain why adrenal medullary grafts may promote functional recovery in human parkinsonism : ( 1 ) replacement of lost striatal neurotransmitter ( dopamine ) by the viable grafted tissue , or ( 2 ) induction of recovery of remaining host dopaminergic systems by the implantation procedure .
NA
{ "id": "C0013030", "name": "dopamine", "pos": [ 190, 198 ] }
{ "id": "C0282151", "name": "dopaminergic", "pos": [ 281, 293 ] }
we have used retrograde labeling with horseradish peroxidase ( hrp ) and a wheat germ agglutinin conjugate of hrp ( wga : hrp ) to investigate the projections of the nucleus postglomerulosus ( npg ) both in normal goldfish and in animals which had undergone retinal removal .
NA
{ "id": "C0078473", "name": "wheat", "pos": [ 75, 80 ] }
{ "id": "C0019941", "name": "hrp", "pos": [ 122, 125 ] }
sera from patients with other types of head and neck cancer and relatively high levels of igg antibody against viral capsid antigen ( vca ) and ea did not react reproducibly with any of the ebv-associated proteins .
NA
{ "id": "C0003342", "name": "viral", "pos": [ 111, 116 ] }
{ "id": "C0003320", "name": "ea", "pos": [ 156, 158 ] }
retinoic acid regulates igg fc receptor expression in human myelomonocytic leukemia cells and normal peripheral monocytes .
NA
{ "id": "C0007634", "name": "cells", "pos": [ 84, 89 ] }
{ "id": "C1321301", "name": "peripheral monocytes", "pos": [ 101, 121 ] }
however , ra increased the percentage of ea rosetting promyelocytes of hl-60 and of patients with acute promyelocytic leukemia and a part of myeloblasts isolated from acute myelogenous leukemia patients .
NA
{ "id": "C0023487", "name": "acute promyelocytic leukemia", "pos": [ 98, 126 ] }
{ "id": "C0023467", "name": "acute myelogenous leukemia", "pos": [ 167, 193 ] }
our results suggest that tp and long toxins recognize the neuromuscular nicotinic acetylcholine receptor ( achr ) and/or bind to the achr in a different mode than the short toxins do .
NA
{ "id": "C0034830", "name": "nicotinic acetylcholine receptor", "pos": [ 72, 104 ] }
{ "id": "C0034792", "name": "achr", "pos": [ 133, 137 ] }
we previously established a human t cell line , tpa-mat , which can proliferate in response to not only interleukin-2 ( il-2 ) , but also phorbol esters such as 12-o-tetradecanoylphorbol-13-acetate ( tpa ) and phorbol-12,13-dibutyrate ( pdbu ) .
NA
{ "id": "C0031586", "name": "phorbol esters", "pos": [ 138, 152 ] }
{ "id": "C0039654", "name": "12-o-tetradecanoylphorbol-13-acetate", "pos": [ 161, 197 ] }
furthermore , whereas the accumulation of ip1 , ip2 and ip3 rapidly increased by as much as 125-175 % in chemotactic-factor-stimulated ams from healthy subjects , stimulation of cells from aas increased these inositol phosphates only slightly .
NA
{ "id": "C0021549", "name": "ip3", "pos": [ 56, 59 ] }
{ "id": "C0021554", "name": "inositol phosphates", "pos": [ 209, 228 ] }
our findings suggest that this dna-binding protein ( s ) may be a trans-acting factor in the regulation of the transcription of wheat histone genes .
NA
{ "id": "C0012940", "name": "dna-binding protein", "pos": [ 31, 50 ] }
{ "id": "C0040627", "name": "trans-acting factor", "pos": [ 66, 85 ] }
in the combined pge2/naproxen treatment the pge levels were significantly ( p less than 0.05 ) elevated in the ejaculate 48 hours after treatment .
NA
{ "id": "C0012472", "name": "pge2", "pos": [ 16, 20 ] }
{ "id": "C0033559", "name": "pge", "pos": [ 44, 47 ] }
among three dna polymerases , the level of dna polymerase beta activity well correlated with the histological findings ( johnsen 's score ) , i.e. , the extent of differentiation of germinal cells .
NA
{ "id": "C0012892", "name": "dna polymerases", "pos": [ 12, 27 ] }
{ "id": "C0525039", "name": "dna polymerase beta", "pos": [ 43, 62 ] }
an increase in total phospholipids of lung extracts as well as that of separate fractions of phospholipids especially of phosphatidylcholine was revealed along with a direct interrelationship between the alveoli area and the phosphatidylcholine rate .
NA
{ "id": "C0031676", "name": "phospholipids", "pos": [ 21, 34 ] }
{ "id": "C0771648", "name": "of", "pos": [ 118, 120 ] }
the levels of hormones of the hypophysis ( acth , tth , cth ) , thyroid gland ( t3 , t4 ) , adrenal glands ( epinephrine , norepinephrine , cortisol ) and pancreas ( insulin , glucagon ) increased during a prolonged electrostimulation of the reticular nucleus of mesencephalon in rabbits .
NA
{ "id": "C0014563", "name": "epinephrine", "pos": [ 109, 120 ] }
{ "id": "C0028351", "name": "norepinephrine", "pos": [ 123, 137 ] }
to examine the mechanism of induction of differentiation in the human malignant t-lymphoblastic cell line , molt-3 , by 12-o-tetradecanoylphorbol-13-acetate ( tpa ) , the role of receptors for phorbol esters was investigated .
NA
{ "id": "C0039654", "name": "12-o-tetradecanoylphorbol-13-acetate", "pos": [ 120, 156 ] }
{ "id": "C0031586", "name": "phorbol esters", "pos": [ 193, 207 ] }
the 7-ethoxyresorufin and 7-ethoxycoumarin deethylase , aryl hydrocarbon hydroxylase and cytochrome c-reductase activities were increased by benzo ( a ) pyrene in all the dietary groups .
NA
{ "id": "C0000644", "name": "ethoxycoumarin deethylase", "pos": [ 28, 53 ] }
{ "id": "C0003927", "name": "aryl hydrocarbon hydroxylase", "pos": [ 56, 84 ] }
randomised trial comparing combinations of cyclophosphamide and cisplatin without or with doxorubicin or 4'-epi-doxorubicin in the treatment of advanced ovarian cancer .
NA
{ "id": "C0013089", "name": "doxorubicin", "pos": [ 90, 101 ] }
{ "id": "C0014582", "name": "4", "pos": [ 105, 106 ] }
to this end , porcine granulosa cells were incubated in monolayer culture for 1-4 days in the presence of fsh ( 200 ng/ml ) , forskolin ( 85 microm ) , or cholera toxin ( 3 micrograms/ml ) with or without an activator of protein kinase c , the phorbol ester 12-o-tetradecanoylphorbol 13-acetate ( tpa ) ( 30 ng/ml ) .
NA
{ "id": "C0031586", "name": "phorbol", "pos": [ 244, 251 ] }
{ "id": "C0039654", "name": "12-o-tetradecanoylphorbol 13-acetate", "pos": [ 258, 294 ] }
the immunofluorescence distribution of alpha- and beta-mhc isoproteins in newly isolated and cultured cardiomyocytes changed from 100 % alpha-mhc and 70 % beta-mhc in rod-shaped cells to about 100 % beta-mhc and 70 % alpha-mhc in spread out cultured cells .
NA
{ "id": "C0027100", "name": "mhc", "pos": [ 55, 58 ] }
{ "id": "C0027096", "name": "mhc", "pos": [ 223, 226 ] }
in previous work , we found that the phorbol ester drug 12-o-tetradecanoyl phorbol acetate ( tpa ) reversed the developmental restriction of melanogenesis that normally occurs in neural crest-derived schwann cell precursors around embryonic day 5 of quail development .
NA
{ "id": "C0031586", "name": "phorbol ester", "pos": [ 37, 50 ] }
{ "id": "C0039654", "name": "tetradecanoyl", "pos": [ 61, 74 ] }
according to the area and linearity of the tracks , the migratory behavior of the different cells can be classified into three groups : ( i ) fibroblasts and the nonpigmented bowes melanoma cells form straight and long tracks ;
NA
{ "id": "C0007634", "name": "the", "pos": [ 13, 16 ] }
{ "id": "C0016030", "name": "fibroblasts", "pos": [ 142, 153 ] }
influence of camp and calcium on [ 3h ] inositol efflux , inositol phosphate accumulation , and insulin release from isolated rat islets .
NA
{ "id": "C0021547", "name": "inositol", "pos": [ 40, 48 ] }
{ "id": "C0021554", "name": "inositol phosphate", "pos": [ 58, 76 ] }
all three stimulants increased the hydrolysis of inositol-containing phospholipids , an event monitored by an increase in [ 3h ] inositol efflux from [ 3h ] inositol-prelabeled islets and by the accumulation of labeled inositol phosphates .
NA
{ "id": "C0021547", "name": "inositol", "pos": [ 49, 57 ] }
{ "id": "C0021554", "name": "inositol phosphates", "pos": [ 219, 238 ] }