prompt
stringlengths
120
209
completion
stringlengths
15
103
input_smiles
stringlengths
14
103
output_smiles
stringlengths
15
103
task_id
int64
102
102
winner_action
dict
Can you make molecule CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1 less soluble in water? The output molecule should be similar to the input molecule.
C=CCC[C@]1(C)NC(=O)[C@H](CCC)N(Cc2nc(C)cs2)C1=O
CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1
C=CCC[C@]1(C)NC(=O)[C@H](CCC)N(Cc2nc(C)cs2)C1=O
102
{ "fragment_index": 0, "new_substring": "C=CCC&", "old_substring": "C4C" }
Can you make molecule CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H]1C(=O)N[C@@](C)(CCCCl)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CCCCl)C(=O)N1Cc1nc(C)cs1
102
{ "fragment_index": 0, "new_substring": "C&CCCl", "old_substring": "C4C" }
Can you make molecule CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H]1C(=O)N[C@@](C)(CCCCS)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CCCCS)C(=O)N1Cc1nc(C)cs1
102
{ "fragment_index": 0, "new_substring": "C&CCCS", "old_substring": "C4C" }
Can you make molecule CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H]1C(=O)N[C@@](C)(CCCBr)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CCCBr)C(=O)N1Cc1nc(C)cs1
102
{ "fragment_index": 0, "new_substring": "C&CCBr", "old_substring": "C4C" }
Can you make molecule CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H]1C(=O)N[C@@](C)(CCCCF)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CC)C(=O)N1Cc1nc(C)cs1
CCC[C@H]1C(=O)N[C@@](C)(CCCCF)C(=O)N1Cc1nc(C)cs1
102
{ "fragment_index": 0, "new_substring": "C&CCCF", "old_substring": "C4C" }
Can you make molecule Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)n([C@H]2CNC[C@@H]2C)n1
Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1
Cc1cc(C)n([C@H]2CNC[C@@H]2C)n1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CN&C[C@@H]1C", "old_substring": "[C@H]13CCC[NH2+]C1" }
Can you make molecule Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)n([C@H]2C=CCC2)n1
Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1
Cc1cc(C)n([C@H]2C=CCC2)n1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&C=C[C@H]&C1", "old_substring": "[C@H]13CCC[NH2+]C1" }
Can you make molecule Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)n(C2CCCCC2)n1
Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1
Cc1cc(C)n(C2CCCCC2)n1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCC[C@H]&C1", "old_substring": "[C@H]13CCC[NH2+]C1" }
Can you make molecule Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)n([C@H]2C=CCC2)n1
Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1
Cc1cc(C)n([C@H]2C=CCC2)n1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&C=C[C@@H]&C1", "old_substring": "[C@H]13CCC[NH2+]C1" }
Can you make molecule Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)n(C2CCCCCC2)n1
Cc1cc(C)n([C@H]2CCC[NH2+]C2)n1
Cc1cc(C)n(C2CCCCCC2)n1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCC[C@H]&CC1", "old_substring": "[C@H]13CCC[NH2+]C1" }
Can you make molecule C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCN(SC(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(SC(=O)CNc2c(F)cccc2F)C1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C3(=O)C4" }
Can you make molecule C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCN(C(=O)CCCC(=O)Nc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CCCC(=O)Nc2c(F)cccc2F)C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C3(=O)C4" }
Can you make molecule C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCN(C(=O)CC(C)(C)Nc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CC(C)(C)Nc2c(F)cccc2F)C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C3(=O)C4" }
Can you make molecule C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCN(C[S@+]([O-])CCCNc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(C[S@+]([O-])CCCNc2c(F)cccc2F)C1
102
{ "fragment_index": 0, "new_substring": "C&[S@](=O)CCC&", "old_substring": "C3(=O)C4" }
Can you make molecule C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCN(C(=O)CCC(C)(C)Nc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CNc2c(F)cccc2F)C1
C[C@H]1CCCN(C(=O)CCC(C)(C)Nc2c(F)cccc2F)C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C3(=O)C4" }
Can you make molecule CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CCNC(=O)N1CC[C@@H]([NH2+][C@H]2CC[C@@](c3ccc(Br)cc3)(C3CC3)C2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H]2CC[C@@](c3ccc(Br)cc3)(C3CC3)C2)C1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC[C@]&&C1", "old_substring": "[C@H]689" }
Can you make molecule CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CCNC(=O)N1CC[C@@H]([NH2+][C@H]2CC[C@](c3ccc(Br)cc3)(C3CC3)C2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H]2CC[C@](c3ccc(Br)cc3)(C3CC3)C2)C1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC[C@@]&&C1", "old_substring": "[C@H]689" }
Can you make molecule CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CCNC(=O)N1CC[C@@H]([NH2+][C@@H](CCCC2CC2)C(C)(C)c2ccc(Br)cc2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@@H](CCCC2CC2)C(C)(C)c2ccc(Br)cc2)C1
102
{ "fragment_index": 0, "new_substring": "[C@H]&(CCC&)C&(C)C", "old_substring": "[C@H]689" }
Can you make molecule CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CCNC(=O)N1CC[C@@H]([NH2+][C@@H]2CCC[C@@](c3ccc(Br)cc3)(C3CC3)C2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@@H]2CCC[C@@](c3ccc(Br)cc3)(C3CC3)C2)C1
102
{ "fragment_index": 0, "new_substring": "[C@@H]1&CCC[C@]&&C1", "old_substring": "[C@H]689" }
Can you make molecule CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CCNC(=O)N1CC[C@@H]([NH2+]CC[C@H](CC2CC2)C(=O)c2ccc(Br)cc2)C1
CCNC(=O)N1CC[C@@H]([NH2+][C@H](c2ccc(Br)cc2)C2CC2)C1
CCNC(=O)N1CC[C@@H]([NH2+]CC[C@H](CC2CC2)C(=O)c2ccc(Br)cc2)C1
102
{ "fragment_index": 0, "new_substring": "C&C[C@H](C&)C&=O", "old_substring": "[C@H]689" }
Can you make molecule CC[C@H](CBr)C[C@H]1Cc2ccccc2S1 less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C)C[C@H](CC)[C@H]1Cc2ccccc2S1
CC[C@H](CBr)C[C@H]1Cc2ccccc2S1
CC[C@@H](C)C[C@H](CC)[C@H]1Cc2ccccc2S1
102
{ "fragment_index": 0, "new_substring": "CC[C@H]&C[C@H](C)CC", "old_substring": "CC[C@@H](C3)CBr" }
Can you make molecule CC[C@H](CBr)C[C@H]1Cc2ccccc2S1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H](Br)CC[C@H]1Cc2ccccc2S1
CC[C@H](CBr)C[C@H]1Cc2ccccc2S1
CCC[C@H](Br)CC[C@H]1Cc2ccccc2S1
102
{ "fragment_index": 0, "new_substring": "CCC[C@H](Br)CC&", "old_substring": "CC[C@@H](C3)CBr" }
Can you make molecule CC[C@H](CBr)C[C@H]1Cc2ccccc2S1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)(C)CC[C@@H](CBr)[C@H]1Cc2ccccc2S1
CC[C@H](CBr)C[C@H]1Cc2ccccc2S1
CC(C)(C)CC[C@@H](CBr)[C@H]1Cc2ccccc2S1
102
{ "fragment_index": 0, "new_substring": "CC(C)(C)CC[C@H]&CBr", "old_substring": "CC[C@@H](C3)CBr" }
Can you make molecule CC[C@H](CBr)C[C@H]1Cc2ccccc2S1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)CC[C@H](Br)C[C@H]1Cc2ccccc2S1
CC[C@H](CBr)C[C@H]1Cc2ccccc2S1
CC(C)CC[C@H](Br)C[C@H]1Cc2ccccc2S1
102
{ "fragment_index": 0, "new_substring": "C&[C@@H](Br)CCC(C)C", "old_substring": "CC[C@@H](C3)CBr" }
Can you make molecule CC[C@H](CBr)C[C@H]1Cc2ccccc2S1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC[C@H](CC)C[C@H]1Cc2ccccc2S1
CC[C@H](CBr)C[C@H]1Cc2ccccc2S1
CCCC[C@H](CC)C[C@H]1Cc2ccccc2S1
102
{ "fragment_index": 0, "new_substring": "CCCC[C@@H](C&)CC", "old_substring": "CC[C@@H](C3)CBr" }
Can you make molecule O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NNC(=O)[C@H]1Cc2ccccc2S1)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@H]1Cc2ccccc2S1)[C@H]1COc2ccc(F)cc2C1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&Cc2ccccc2S1", "old_substring": "[C@H]13Cc2ccccc2O1" }
Can you make molecule O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NNC(=O)[C@@H]1Nc2ccccc2S1)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@@H]1Nc2ccccc2S1)[C@H]1COc2ccc(F)cc2C1
102
{ "fragment_index": 0, "new_substring": "[C@@H]1&Nc2ccccc2S1", "old_substring": "[C@H]13Cc2ccccc2O1" }
Can you make molecule O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NNC(=O)[C@H]1COc2ccc(F)cc2C1)N[C@H]1CCc2ccccc21
O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@H]1COc2ccc(F)cc2C1)N[C@H]1CCc2ccccc21
102
{ "fragment_index": 0, "new_substring": "N&[C@H]1CCc2ccccc21", "old_substring": "[C@H]13Cc2ccccc2O1" }
Can you make molecule O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1Cc2cc(C(=O)NNC(=O)[C@H]3COc4ccc(F)cc4C3)ccc2O1
O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1
C[C@H]1Cc2cc(C(=O)NNC(=O)[C@H]3COc4ccc(F)cc4C3)ccc2O1
102
{ "fragment_index": 0, "new_substring": "C[C@H]1Cc2cc&ccc2O1", "old_substring": "[C@H]13Cc2ccccc2O1" }
Can you make molecule O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(C[C@H]1Cc2ccccc21)NNC(=O)[C@H]1COc2ccc(F)cc2C1
O=C(NNC(=O)[C@H]1Cc2ccccc2O1)[C@H]1COc2ccc(F)cc2C1
O=C(C[C@H]1Cc2ccccc21)NNC(=O)[C@H]1COc2ccc(F)cc2C1
102
{ "fragment_index": 0, "new_substring": "C&[C@H]1Cc2ccccc21", "old_substring": "[C@H]13Cc2ccccc2O1" }
Can you make molecule CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12 less soluble in water? The output molecule should be similar to the input molecule.
CCSC(=S)OC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCSC(=S)OC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
102
{ "fragment_index": 0, "new_substring": "O&C(=S)S&", "old_substring": "O34" }
Can you make molecule CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12 less soluble in water? The output molecule should be similar to the input molecule.
CCCC(=N)OC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCCC(=N)OC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
102
{ "fragment_index": 0, "new_substring": "O&C(=N)C&", "old_substring": "O34" }
Can you make molecule CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12 less soluble in water? The output molecule should be similar to the input molecule.
CCCC[C@@H](O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCCC[C@@H](O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
102
{ "fragment_index": 0, "new_substring": "O[C@@H]&CC&", "old_substring": "O34" }
Can you make molecule CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12 less soluble in water? The output molecule should be similar to the input molecule.
CCS/C=C/C(=O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCS/C=C/C(=O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
102
{ "fragment_index": 0, "new_substring": "O=C&/C=C/S&", "old_substring": "O34" }
Can you make molecule CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12 less soluble in water? The output molecule should be similar to the input molecule.
CCCCC[C@@H](O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCOC(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
CCCCC[C@@H](O)C(=O)[C@]1(CC)O[C@]12CCCc1ccc(OC)cc12
102
{ "fragment_index": 0, "new_substring": "O[C@@H]&CCC&", "old_substring": "O34" }
Can you make molecule CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1 less soluble in water? The output molecule should be similar to the input molecule.
Clc1ccc(N2CCC(Cc3ccccc3N3CCOCC3)CC2)nc1
CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1
Clc1ccc(N2CCC(Cc3ccccc3N3CCOCC3)CC2)nc1
102
{ "fragment_index": 0, "new_substring": "C1&CCN&CC1", "old_substring": "CN23" }
Can you make molecule CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1 less soluble in water? The output molecule should be similar to the input molecule.
CN(Cc1ccccc1N1CCOCC1)C(=S)Sc1ccc(Cl)cn1
CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1
CN(Cc1ccccc1N1CCOCC1)C(=S)Sc1ccc(Cl)cn1
102
{ "fragment_index": 0, "new_substring": "CN&C(=S)S&", "old_substring": "CN23" }
Can you make molecule CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1 less soluble in water? The output molecule should be similar to the input molecule.
Clc1ccc(C2CCN(CCc3ccccc3N3CCOCC3)CC2)nc1
CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1
Clc1ccc(C2CCN(CCc3ccccc3N3CCOCC3)CC2)nc1
102
{ "fragment_index": 0, "new_substring": "C&N1CCC&CC1", "old_substring": "CN23" }
Can you make molecule CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1 less soluble in water? The output molecule should be similar to the input molecule.
S=C1SCN(Cc2ccccc2N2CCOCC2)CN1c1ccc(Cl)cn1
CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1
S=C1SCN(Cc2ccccc2N2CCOCC2)CN1c1ccc(Cl)cn1
102
{ "fragment_index": 0, "new_substring": "S=C1SCN&CN1&", "old_substring": "CN23" }
Can you make molecule CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1 less soluble in water? The output molecule should be similar to the input molecule.
N#CC1(Cc2ccccc2N2CCOCC2)CCC(c2ccc(Cl)cn2)CC1
CN(Cc1ccccc1N1CCOCC1)c1ccc(Cl)cn1
N#CC1(Cc2ccccc2N2CCOCC2)CCC(c2ccc(Cl)cn2)CC1
102
{ "fragment_index": 0, "new_substring": "C1&(C#N)CCC&CC1", "old_substring": "CN23" }
Can you make molecule COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
COCc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
COCc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO3" }
Can you make molecule COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
COCSc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
COCSc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO3" }
Can you make molecule COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Sc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
CC(=O)Sc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO3" }
Can you make molecule COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OCC(=O)NNC(=O)c2ccccc2)c(C(=O)CS)c1
COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
Cc1ccc(OCC(=O)NNC(=O)c2ccccc2)c(C(=O)CS)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO3" }
Can you make molecule COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OCC(=O)NNC(=O)c2ccccc2)c(C(=O)CI)c1
COc1cc(C)ccc1OCC(=O)NNC(=O)c1ccccc1
Cc1ccc(OCC(=O)NNC(=O)c2ccccc2)c(C(=O)CI)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO3" }
Can you make molecule CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C)S(=O)(=O)Nc1cc(Cl)ccc1Cl
CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl
CC[C@@H](C)S(=O)(=O)Nc1cc(Cl)ccc1Cl
102
{ "fragment_index": 0, "new_substring": "CC[C@@H](C)S&(=O)=O", "old_substring": "CC[S@@](=O)CC2=O" }
Can you make molecule CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl less soluble in water? The output molecule should be similar to the input molecule.
CCCC[S@@+]([O-])CNc1cc(Cl)ccc1Cl
CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl
CCCC[S@@+]([O-])CNc1cc(Cl)ccc1Cl
102
{ "fragment_index": 0, "new_substring": "CCCC[S@@](=O)C&", "old_substring": "CC[S@@](=O)CC2=O" }
Can you make molecule CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl less soluble in water? The output molecule should be similar to the input molecule.
CC[C@H](C)S(=O)(=O)Nc1cc(Cl)ccc1Cl
CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl
CC[C@H](C)S(=O)(=O)Nc1cc(Cl)ccc1Cl
102
{ "fragment_index": 0, "new_substring": "CC[C@H](C)S&(=O)=O", "old_substring": "CC[S@@](=O)CC2=O" }
Can you make molecule CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl less soluble in water? The output molecule should be similar to the input molecule.
CCCC[S@+]([O-])CNc1cc(Cl)ccc1Cl
CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl
CCCC[S@+]([O-])CNc1cc(Cl)ccc1Cl
102
{ "fragment_index": 0, "new_substring": "CCCC[S@](=O)C&", "old_substring": "CC[S@@](=O)CC2=O" }
Can you make molecule CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl less soluble in water? The output molecule should be similar to the input molecule.
CC[C@H](C)CS(=O)(=O)Nc1cc(Cl)ccc1Cl
CC[S@@+]([O-])CC(=O)Nc1cc(Cl)ccc1Cl
CC[C@H](C)CS(=O)(=O)Nc1cc(Cl)ccc1Cl
102
{ "fragment_index": 0, "new_substring": "CC[C@H](C)CS&(=O)=O", "old_substring": "CC[S@@](=O)CC2=O" }
Can you make molecule CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(C(=O)CCCC(=O)N2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CCCC(=O)N2CCO[C@H](C#N)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C4(=O)C3" }
Can you make molecule CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(C(=O)CC(C)(C)N2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CC(C)(C)N2CCO[C@H](C#N)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C4(=O)C3" }
Can you make molecule CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(C(=O)CCC(C)(C)N2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CCC(C)(C)N2CCO[C@H](C#N)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C4(=O)C3" }
Can you make molecule CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(C(=O)C[C@H](C)N2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)C[C@H](C)N2CCO[C@H](C#N)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)C[C@@H]&C", "old_substring": "C4(=O)C3" }
Can you make molecule CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(C(=O)C[C@@H](Br)N2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)CN2CCO[C@H](C#N)C2)cc1
CCc1ccc(C(=O)C[C@@H](Br)N2CCO[C@H](C#N)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)C[C@H]&Br", "old_substring": "C4(=O)C3" }
Can you make molecule Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1 less soluble in water? The output molecule should be similar to the input molecule.
Oc1cc(Br)cc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
Oc1cc(Br)cc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
102
{ "fragment_index": 0, "new_substring": "Oc1cc&cc(Br)c1", "old_substring": "Oc1ccccc14" }
Can you make molecule Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1 less soluble in water? The output molecule should be similar to the input molecule.
Oc1ccc(Br)cc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
Oc1ccc(Br)cc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
102
{ "fragment_index": 0, "new_substring": "Oc1ccc(Br)cc1&", "old_substring": "Oc1ccccc14" }
Can you make molecule Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1 less soluble in water? The output molecule should be similar to the input molecule.
C1=C(c2ccc3c(c2)OCCO3)N=[NH+][C@@H]1c1ccccc1
Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
C1=C(c2ccc3c(c2)OCCO3)N=[NH+][C@@H]1c1ccccc1
102
{ "fragment_index": 0, "new_substring": "c1&ccccc1", "old_substring": "Oc1ccccc14" }
Can you make molecule Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1 less soluble in water? The output molecule should be similar to the input molecule.
Fc1cccc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
Fc1cccc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
102
{ "fragment_index": 0, "new_substring": "Fc1cccc&c1", "old_substring": "Oc1ccccc14" }
Can you make molecule Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
Oc1ccccc1[C@@H]1C=C(c2ccc3c(c2)OCCO3)N=[NH+]1
Cc1cccc([C@@H]2C=C(c3ccc4c(c3)OCCO4)N=[NH+]2)c1
102
{ "fragment_index": 0, "new_substring": "Cc1cccc&c1", "old_substring": "Oc1ccccc14" }
Can you make molecule CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1ccc(Cl)s1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1ccc(Cl)s1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)s1", "old_substring": "c12cccs1" }
Can you make molecule CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1ccc(Br)s1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1ccc(Br)s1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Br)s1", "old_substring": "c12cccs1" }
Can you make molecule CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1scc2c1CCCC2
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1scc2c1CCCC2
102
{ "fragment_index": 0, "new_substring": "c1&scc2c1CCCC2", "old_substring": "c12cccs1" }
Can you make molecule CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1sccc1Br
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1sccc1Br
102
{ "fragment_index": 0, "new_substring": "c1&sccc1Br", "old_substring": "c12cccs1" }
Can you make molecule CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1c(C/C([O-])=N/S(=O)(=O)CC(C)(C)C)sc2ccccc12
CC(C)(C)CS(=O)(=O)/N=C(\[O-])Cc1cccs1
Cc1c(C/C([O-])=N/S(=O)(=O)CC(C)(C)C)sc2ccccc12
102
{ "fragment_index": 0, "new_substring": "c1&sc2ccccc2c1C", "old_substring": "c12cccs1" }
Can you make molecule COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12 less soluble in water? The output molecule should be similar to the input molecule.
COCc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COCc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO7" }
Can you make molecule COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12 less soluble in water? The output molecule should be similar to the input molecule.
COCSc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COCSc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO7" }
Can you make molecule COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(SC(C)=O)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COc1ccc(SC(C)=O)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO7" }
Can you make molecule COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C(=O)CS)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COc1ccc(C(=O)CS)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO7" }
Can you make molecule COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C(=O)CI)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
COc1ccc(OC)c2sc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)nc12
COc1ccc(C(=O)CI)c2nc(NC(=O)c3cc4c(ccc5ccccc54)oc3=O)sc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO7" }
Can you make molecule Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(O)c(C(=O)NCSC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)NCSC[C@H]2CCC[C@@H](O)C2)c1
102
{ "fragment_index": 0, "new_substring": "N&CS&", "old_substring": "N34" }
Can you make molecule Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(O)c(C(=O)N2CC(C[C@H]3CCC[C@@H](O)C3)C2)c1
Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)N2CC(C[C@H]3CCC[C@@H](O)C3)C2)c1
102
{ "fragment_index": 0, "new_substring": "N1&CC&C1", "old_substring": "N34" }
Can you make molecule Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(O)c(C(=O)NC(=N)SC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)NC(=N)SC[C@H]2CCC[C@@H](O)C2)c1
102
{ "fragment_index": 0, "new_substring": "N&C(=N)S&", "old_substring": "N34" }
Can you make molecule Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(O)c(C(=O)c2nsc(C[C@H]3CCC[C@@H](O)C3)c2N)c1
Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)c2nsc(C[C@H]3CCC[C@@H](O)C3)c2N)c1
102
{ "fragment_index": 0, "new_substring": "Nc1c&nsc1&", "old_substring": "N34" }
Can you make molecule Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(O)c(C(=O)N(C)C(=S)SC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1
Cc1ccc(O)c(C(=O)N(C)C(=S)SC[C@H]2CCC[C@@H](O)C2)c1
102
{ "fragment_index": 0, "new_substring": "CN&C(=S)S&", "old_substring": "N34" }
Can you make molecule O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1C=CO[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)C1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1
O=C1C=CO[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)C1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC(=O)C=CO1", "old_substring": "[C@H]14CCS(=O)(=O)C1" }
Can you make molecule O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1C[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)CS1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1
O=C1C[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)CS1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CSC(=O)C1", "old_substring": "[C@H]14CCS(=O)(=O)C1" }
Can you make molecule O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CC=CS2)CC1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CC=CS2)CC1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC=CS1", "old_substring": "[C@H]14CCS(=O)(=O)C1" }
Can you make molecule O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
N=C1C=C[C@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)S1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1
N=C1C=C[C@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)S1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&C=CC(=N)S1", "old_substring": "[C@H]14CCS(=O)(=O)C1" }
Can you make molecule O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1=C(C)[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)N=N1
O=C(c1cc(=O)c2cc(Cl)ccc2o1)N1CCN([C@H]2CCS(=O)(=O)C2)CC1
CC1=C(C)[C@@H](N2CCN(C(=O)c3cc(=O)c4cc(Cl)ccc4o3)CC2)N=N1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&N=NC(C)=C1C", "old_substring": "[C@H]14CCS(=O)(=O)C1" }
Can you make molecule COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(/C=N/NC(=O)c2ccccc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2ccccc2)cc1[N+](=O)[O-]
102
{ "fragment_index": 0, "new_substring": "c1&ccccc1", "old_substring": "c14cccnc1" }
Can you make molecule COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(/C=N/NC(=O)c2ccc(I)nc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2ccc(I)nc2)cc1[N+](=O)[O-]
102
{ "fragment_index": 0, "new_substring": "c1&ccc(I)nc1", "old_substring": "c14cccnc1" }
Can you make molecule COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(/C=N/NC(=O)c2cc3cnsc3s2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cc3cnsc3s2)cc1[N+](=O)[O-]
102
{ "fragment_index": 0, "new_substring": "c1&cc2cnsc2s1", "old_substring": "c14cccnc1" }
Can you make molecule COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(/C=N/NC(=O)c2ccc(C)nc2C)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2ccc(C)nc2C)cc1[N+](=O)[O-]
102
{ "fragment_index": 0, "new_substring": "c1&ccc(C)nc1C", "old_substring": "c14cccnc1" }
Can you make molecule COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(/C=N/NC(=O)c2ccncc2Cl)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2cccnc2)cc1[N+](=O)[O-]
COc1ccc(/C=N/NC(=O)c2ccncc2Cl)cc1[N+](=O)[O-]
102
{ "fragment_index": 0, "new_substring": "c1&ccncc1Cl", "old_substring": "c14cccnc1" }
Can you make molecule O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1 less soluble in water? The output molecule should be similar to the input molecule.
O=Cc1cn([C@H]2CC(=O)C=CO2)nc1-c1ccoc1
O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1
O=Cc1cn([C@H]2CC(=O)C=CO2)nc1-c1ccoc1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC(=O)C=CO1", "old_substring": "[C@H]13CCS(=O)(=O)C1" }
Can you make molecule O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1 less soluble in water? The output molecule should be similar to the input molecule.
O=Cc1cn([C@H]2CSC(=O)C2)nc1-c1ccoc1
O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1
O=Cc1cn([C@H]2CSC(=O)C2)nc1-c1ccoc1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CSC(=O)C1", "old_substring": "[C@H]13CCS(=O)(=O)C1" }
Can you make molecule O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1 less soluble in water? The output molecule should be similar to the input molecule.
O=Cc1cn([C@H]2CC=CS2)nc1-c1ccoc1
O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1
O=Cc1cn([C@H]2CC=CS2)nc1-c1ccoc1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC=CS1", "old_substring": "[C@H]13CCS(=O)(=O)C1" }
Can you make molecule O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1 less soluble in water? The output molecule should be similar to the input molecule.
N=C1C=C[C@H](n2cc(C=O)c(-c3ccoc3)n2)S1
O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1
N=C1C=C[C@H](n2cc(C=O)c(-c3ccoc3)n2)S1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&C=CC(=N)S1", "old_substring": "[C@H]13CCS(=O)(=O)C1" }
Can you make molecule O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1 less soluble in water? The output molecule should be similar to the input molecule.
CC1=C(C)[C@@H](n2cc(C=O)c(-c3ccoc3)n2)N=N1
O=Cc1cn([C@H]2CCS(=O)(=O)C2)nc1-c1ccoc1
CC1=C(C)[C@@H](n2cc(C=O)c(-c3ccoc3)n2)N=N1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&N=NC(C)=C1C", "old_substring": "[C@H]13CCS(=O)(=O)C1" }
Can you make molecule Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CCCC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CCCC(F)(F)F
102
{ "fragment_index": 0, "new_substring": "C&CCC(F)(F)F", "old_substring": "C5C(F)(F)F" }
Can you make molecule Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CCCCC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CCCCC(F)(F)F
102
{ "fragment_index": 0, "new_substring": "C&CCCC(F)(F)F", "old_substring": "C5C(F)(F)F" }
Can you make molecule Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1S/C=C/C(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1S/C=C/C(F)(F)F
102
{ "fragment_index": 0, "new_substring": "S&/C=C/C(F)(F)F", "old_substring": "C5C(F)(F)F" }
Can you make molecule Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)C(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)C(F)(F)F
102
{ "fragment_index": 0, "new_substring": "C&C(F)(F)C(F)(F)F", "old_substring": "C5C(F)(F)F" }
Can you make molecule Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1C1CCC(F)(F)CC1
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1CC(F)(F)F
Cc1cc(C(=O)C(C#N)=Cc2cn(C)nc2C(C)(C)C)c(C)n1C1CCC(F)(F)CC1
102
{ "fragment_index": 0, "new_substring": "C1&CCC(F)(F)CC1", "old_substring": "C5C(F)(F)F" }
Can you make molecule C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1 less soluble in water? The output molecule should be similar to the input molecule.
C/[NH+]=C(/NCc1[nH+]ccn1C(C)(C)CCBr)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1C(C)(C)CCBr)N1C[C@H]2CC=CC[C@@H]2C1
102
{ "fragment_index": 0, "new_substring": "CC&(C)CCBr", "old_substring": "C4C(C)C" }
Can you make molecule C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC(C)(C)n1cc[nH+]c1CN/C(=[NH+]/C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
CCCC(C)(C)n1cc[nH+]c1CN/C(=[NH+]/C)N1C[C@H]2CC=CC[C@@H]2C1
102
{ "fragment_index": 0, "new_substring": "CCCC&(C)C", "old_substring": "C4C(C)C" }
Can you make molecule C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1 less soluble in water? The output molecule should be similar to the input molecule.
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)(C)CBr)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)(C)CBr)N1C[C@H]2CC=CC[C@@H]2C1
102
{ "fragment_index": 0, "new_substring": "C&C(C)(C)CBr", "old_substring": "C4C(C)C" }
Can you make molecule C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1 less soluble in water? The output molecule should be similar to the input molecule.
C/[NH+]=C(/NCc1[nH+]ccn1C(C(C)C)C(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1C(C(C)C)C(C)C)N1C[C@H]2CC=CC[C@@H]2C1
102
{ "fragment_index": 0, "new_substring": "CC(C)C&C(C)C", "old_substring": "C4C(C)C" }
Can you make molecule C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1 less soluble in water? The output molecule should be similar to the input molecule.
C/[NH+]=C(/NCc1[nH+]ccn1C(=O)CCCC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1CC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
C/[NH+]=C(/NCc1[nH+]ccn1C(=O)CCCC(C)C)N1C[C@H]2CC=CC[C@@H]2C1
102
{ "fragment_index": 0, "new_substring": "CC(C)CCCC&=O", "old_substring": "C4C(C)C" }