prompt
stringlengths
120
209
completion
stringlengths
15
103
input_smiles
stringlengths
14
103
output_smiles
stringlengths
15
103
task_id
int64
102
102
winner_action
dict
Can you make molecule COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)c1
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)c1
102
{ "fragment_index": 0, "new_substring": "c1&csc&c1", "old_substring": "c18csc7n1" }
Can you make molecule COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)c1C
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)c1C
102
{ "fragment_index": 0, "new_substring": "c1&csc&c1C", "old_substring": "c18csc7n1" }
Can you make molecule COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C)cc1-c1ccc(NC(=O)COC2CCCC2)s1
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1
COc1ccc(C)cc1-c1ccc(NC(=O)COC2CCCC2)s1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&s1", "old_substring": "c18csc7n1" }
Can you make molecule COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C)cc1-c1cc(NC(=O)COC2CCCC2)cnc1Cl
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1
COc1ccc(C)cc1-c1cc(NC(=O)COC2CCCC2)cnc1Cl
102
{ "fragment_index": 0, "new_substring": "c1&cc&cnc1Cl", "old_substring": "c18csc7n1" }
Can you make molecule COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C)cc1-c1cc(NC(=O)COC2CCCC2)ncc1Cl
COc1ccc(C)cc1-c1csc(NC(=O)COC2CCCC2)n1
COc1ccc(C)cc1-c1cc(NC(=O)COC2CCCC2)ncc1Cl
102
{ "fragment_index": 0, "new_substring": "c1&cc&ncc1Cl", "old_substring": "c18csc7n1" }
Can you make molecule COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C less soluble in water? The output molecule should be similar to the input molecule.
COCc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
COCc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO6" }
Can you make molecule COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C less soluble in water? The output molecule should be similar to the input molecule.
COCSc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
COCSc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO6" }
Can you make molecule COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Sc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
CC(=O)Sc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO6" }
Can you make molecule COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C less soluble in water? The output molecule should be similar to the input molecule.
CC1=C(C(=O)Nc2ccc(C)cc2C)[C@H](c2ccc(OC(C)C)c(C(=O)CS)c2)n2ncnc2N1
COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
CC1=C(C(=O)Nc2ccc(C)cc2C)[C@H](c2ccc(OC(C)C)c(C(=O)CS)c2)n2ncnc2N1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO6" }
Can you make molecule COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C less soluble in water? The output molecule should be similar to the input molecule.
CC1=C(C(=O)Nc2ccc(C)cc2C)[C@H](c2ccc(OC(C)C)c(C(=O)CI)c2)n2ncnc2N1
COc1cc([C@H]2C(C(=O)Nc3ccc(C)cc3C)=C(C)Nc3ncnn32)ccc1OC(C)C
CC1=C(C(=O)Nc2ccc(C)cc2C)[C@H](c2ccc(OC(C)C)c(C(=O)CI)c2)n2ncnc2N1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO6" }
Can you make molecule COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc2cc(C(=O)C3=C(N=Cc4ccccc4F)CCS3)oc12
COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C3=C(N=Cc4ccccc4F)CCS3)oc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)C1=C(N&)CCS1", "old_substring": "C5(=O)C=6" }
Can you make molecule COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc2cc(C(=O)C(N=Cc3ccccc3F)=C(Cl)Cl)oc12
COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C(N=Cc3ccccc3F)=C(Cl)Cl)oc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)C(N&)=C(Cl)Cl", "old_substring": "C5(=O)C=6" }
Can you make molecule COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc2cc(C(=O)C(C=Cc3ccccc3F)=C(Cl)Cl)oc12
COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C(C=Cc3ccccc3F)=C(Cl)Cl)oc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)C(C&)=C(Cl)Cl", "old_substring": "C5(=O)C=6" }
Can you make molecule COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc2cc(C(=O)[C@H](C)CC=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)[C@H](C)CC=Cc3ccccc3F)oc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)[C@H](C)CC&", "old_substring": "C5(=O)C=6" }
Can you make molecule COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc2cc(C(=O)C(C)(C)CCC=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C=Cc3ccccc3F)oc12
COc1cccc2cc(C(=O)C(C)(C)CCC=Cc3ccccc3F)oc12
102
{ "fragment_index": 0, "new_substring": "C&(=O)C(C)(C)CCC&", "old_substring": "C5(=O)C=6" }
Can you make molecule CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C(=O)[O-])c1ccc(O)c(-c2ccc(C)nc2C[NH3+])c2onc1-2
CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-]
CC[C@@H](C(=O)[O-])c1ccc(O)c(-c2ccc(C)nc2C[NH3+])c2onc1-2
102
{ "fragment_index": 0, "new_substring": "Oc1ccc2c&noc2c1&", "old_substring": "O23" }
Can you make molecule CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C(=O)[O-])N1CCOc2ccc(-c3ccc(C)nc3C[NH3+])cc2C1
CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-]
CC[C@@H](C(=O)[O-])N1CCOc2ccc(-c3ccc(C)nc3C[NH3+])cc2C1
102
{ "fragment_index": 0, "new_substring": "N1&CCOc2ccc&cc2C1", "old_substring": "O23" }
Can you make molecule CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C(=O)[O-])c1cc2ccc-2ncn(-c2ccc(C)nc2C[NH3+])c1=O
CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-]
CC[C@@H](C(=O)[O-])c1cc2ccc-2ncn(-c2ccc(C)nc2C[NH3+])c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cc&ccc2ncn1&", "old_substring": "O23" }
Can you make molecule CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C(=O)[O-])c1ccc2nc-2ccn(-c2ccc(C)nc2C[NH3+])c1=O
CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-]
CC[C@@H](C(=O)[O-])c1ccc2nc-2ccn(-c2ccc(C)nc2C[NH3+])c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2ccc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@H](C(=O)[O-])c1cnc2nc-2ccn(-c2ccc(C)nc2C[NH3+])c1=O
CC[C@H](Oc1ccc(C)nc1C[NH3+])C(=O)[O-]
CC[C@@H](C(=O)[O-])c1cnc2nc-2ccn(-c2ccc(C)nc2C[NH3+])c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cnc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1c2ccc(Oc3ccc(NC(=O)C(F)(F)F)cc3I)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3ccc(NC(=O)C(F)(F)F)cc3I)cc2C(=O)N1C[C@H]1CCCO1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&cc1I", "old_substring": "c16cccc7c1" }
Can you make molecule O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1c2ccc(Oc3cc(NC(=O)C(F)(F)F)ccc3Br)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cc(NC(=O)C(F)(F)F)ccc3Br)cc2C(=O)N1C[C@H]1CCCO1
102
{ "fragment_index": 0, "new_substring": "c1&cc&ccc1Br", "old_substring": "c16cccc7c1" }
Can you make molecule O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1c2ccc(Oc3ccc(NC(=O)C(F)(F)F)cc3Cl)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3ccc(NC(=O)C(F)(F)F)cc3Cl)cc2C(=O)N1C[C@H]1CCCO1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&cc1Cl", "old_substring": "c16cccc7c1" }
Can you make molecule O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3Br)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3Br)cc2C(=O)N1C[C@H]1CCCO1
102
{ "fragment_index": 0, "new_substring": "c1&cccc&c1Br", "old_substring": "c16cccc7c1" }
Can you make molecule O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3Cl)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3)cc2C(=O)N1C[C@H]1CCCO1
O=C1c2ccc(Oc3cccc(NC(=O)C(F)(F)F)c3Cl)cc2C(=O)N1C[C@H]1CCCO1
102
{ "fragment_index": 0, "new_substring": "c1&cccc&c1Cl", "old_substring": "c16cccc7c1" }
Can you make molecule CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2I)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2I)c1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&cc1I", "old_substring": "c17ccc6cc1" }
Can you make molecule CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1cccc(O[C@H](C)C(=O)Nc2cc(OC)ccc2Br)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1
CCc1cccc(O[C@H](C)C(=O)Nc2cc(OC)ccc2Br)c1
102
{ "fragment_index": 0, "new_substring": "c1&cc&ccc1Br", "old_substring": "c17ccc6cc1" }
Can you make molecule CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2Cl)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2Cl)c1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&cc1Cl", "old_substring": "c17ccc6cc1" }
Can you make molecule CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1cccc(O[C@H](C)C(=O)Nc2cccc(OC)c2Br)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1
CCc1cccc(O[C@H](C)C(=O)Nc2cccc(OC)c2Br)c1
102
{ "fragment_index": 0, "new_substring": "c1&cccc&c1Br", "old_substring": "c17ccc6cc1" }
Can you make molecule CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1cccc(O[C@H](C)C(=O)Nc2cccc(OC)c2Cl)c1
CCc1cccc(O[C@H](C)C(=O)Nc2ccc(OC)cc2)c1
CCc1cccc(O[C@H](C)C(=O)Nc2cccc(OC)c2Cl)c1
102
{ "fragment_index": 0, "new_substring": "c1&cccc&c1Cl", "old_substring": "c17ccc6cc1" }
Can you make molecule COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1 less soluble in water? The output molecule should be similar to the input molecule.
COCc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COCc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO6" }
Can you make molecule COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1 less soluble in water? The output molecule should be similar to the input molecule.
COCSc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COCSc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO6" }
Can you make molecule COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(SC(C)=O)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COc1ccc(SC(C)=O)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO6" }
Can you make molecule COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C(=O)CS)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COc1ccc(C(=O)CS)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO6" }
Can you make molecule COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(C(=O)CI)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
COc1ccc(OC)c([C@H]2OC(COc3ccc4c(c3)OCO4)=NN2C(C)=O)c1
COc1ccc(C(=O)CI)cc1[C@H]1OC(COc2ccc3c(c2)OCO3)=NN1C(C)=O
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO6" }
Can you make molecule CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
C=CSn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
C=CSn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
102
{ "fragment_index": 0, "new_substring": "C=CS&", "old_substring": "CC4" }
Can you make molecule CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2C(C)C)cc1
CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2C(C)C)cc1
102
{ "fragment_index": 0, "new_substring": "C&(C)C", "old_substring": "CC4" }
Can you make molecule CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
C=CCCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
C=CCCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
102
{ "fragment_index": 0, "new_substring": "C=CCC&", "old_substring": "CC4" }
Can you make molecule CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2CCCCl)cc1
CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2CCCCl)cc1
102
{ "fragment_index": 0, "new_substring": "C&CCCl", "old_substring": "CC4" }
Can you make molecule CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F less soluble in water? The output molecule should be similar to the input molecule.
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2CCCCS)cc1
CCn1c(-c2ccc(OC)cc2)ccc1[C@@H](O)C(F)(F)F
COc1ccc(-c2ccc([C@@H](O)C(F)(F)F)n2CCCCS)cc1
102
{ "fragment_index": 0, "new_substring": "C&CCCS", "old_substring": "CC4" }
Can you make molecule CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1(C)Cc2ccccc2C1
CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-]
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "CC1&Cc2ccccc2C1", "old_substring": "CC2" }
Can you make molecule CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1=CC2=CC=C2OC(C)(C)C1
CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-]
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1=CC2=CC=C2OC(C)(C)C1
102
{ "fragment_index": 0, "new_substring": "CC1(C)Cc2cc&ccc2O1", "old_substring": "CC2" }
Can you make molecule CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1N1CC(C)(C)Oc2ccccc21
CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-]
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1N1CC(C)(C)Oc2ccccc21
102
{ "fragment_index": 0, "new_substring": "CC1(C)CN&c2ccccc2O1", "old_substring": "CC2" }
Can you make molecule CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1N1CC(C)(C)Sc2ccccc21
CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-]
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1N1CC(C)(C)Sc2ccccc21
102
{ "fragment_index": 0, "new_substring": "CC1(C)CN&c2ccccc2S1", "old_substring": "CC2" }
Can you make molecule CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-] less soluble in water? The output molecule should be similar to the input molecule.
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1C2CCC1CC2
CC[NH+]1CCC[C@@H]1C[NH+](C)CCC(=O)[O-]
C[NH+](CCC(=O)[O-])C[C@H]1CCC[NH+]1C1C2CCC1CC2
102
{ "fragment_index": 0, "new_substring": "C1&C2CCC1CC2", "old_substring": "CC2" }
Can you make molecule C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](CC(C)(C)c1ccc(S(C)(=O)=O)c(F)c1)NC(=O)C[C@H](O)c1ccccc1
C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1
C[C@H](CC(C)(C)c1ccc(S(C)(=O)=O)c(F)c1)NC(=O)C[C@H](O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "C[C@@H]&CC&(C)C", "old_substring": "C[C@H]34" }
Can you make molecule C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](CCNC(=O)C[C@H](O)c1ccccc1)CC(=O)c1ccc(S(C)(=O)=O)c(F)c1
C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1
C[C@H](CCNC(=O)C[C@H](O)c1ccccc1)CC(=O)c1ccc(S(C)(=O)=O)c(F)c1
102
{ "fragment_index": 0, "new_substring": "C[C@H](CC&)CC&=O", "old_substring": "C[C@H]34" }
Can you make molecule C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](Cc1ccc(S(C)(=O)=O)c(F)c1)[C@H](C)NC(=O)C[C@H](O)c1ccccc1
C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1
C[C@H](Cc1ccc(S(C)(=O)=O)c(F)c1)[C@H](C)NC(=O)C[C@H](O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "C[C@H]&[C@H](C)C&", "old_substring": "C[C@H]34" }
Can you make molecule C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H](CCNC(=O)C[C@H](O)c1ccccc1)CC(=O)c1ccc(S(C)(=O)=O)c(F)c1
C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1
C[C@@H](CCNC(=O)C[C@H](O)c1ccccc1)CC(=O)c1ccc(S(C)(=O)=O)c(F)c1
102
{ "fragment_index": 0, "new_substring": "C[C@@H](CC&)CC&=O", "old_substring": "C[C@H]34" }
Can you make molecule C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@H](CCc1ccc(S(C)(=O)=O)c(F)c1)NC(=O)C[C@H](O)c1ccccc1
C[C@H](NC(=O)C[C@H](O)c1ccccc1)c1ccc(S(C)(=O)=O)c(F)c1
CCC[C@@H](CCc1ccc(S(C)(=O)=O)c(F)c1)NC(=O)C[C@H](O)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "CCC[C@H]&CC&", "old_substring": "C[C@H]34" }
Can you make molecule C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
C/C(COC(=O)[C@@H](C)c1cccs1)=N/ON(C)[C@@H]1CCCc2ccccc21
C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
C/C(COC(=O)[C@@H](C)c1cccs1)=N/ON(C)[C@@H]1CCCc2ccccc21
102
{ "fragment_index": 0, "new_substring": "C/C(C&)=N/O&", "old_substring": "C5C4=O" }
Can you make molecule C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC(CC)(OC(=O)[C@@H](C)c1cccs1)C(=O)CN(C)[C@@H]1CCCc2ccccc21
C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
CCC(CC)(OC(=O)[C@@H](C)c1cccs1)C(=O)CN(C)[C@@H]1CCCc2ccccc21
102
{ "fragment_index": 0, "new_substring": "CCC&(CC)C(=O)C&", "old_substring": "C5C4=O" }
Can you make molecule C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](C(=O)OSSC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
C[C@H](C(=O)OSSC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
102
{ "fragment_index": 0, "new_substring": "S&SC&=O", "old_substring": "C5C4=O" }
Can you make molecule C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC(CC)(OC(=O)[C@@H](C)c1cccs1)C(=O)CCN(C)[C@@H]1CCCc2ccccc21
C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
CCC(CC)(OC(=O)[C@@H](C)c1cccs1)C(=O)CCN(C)[C@@H]1CCCc2ccccc21
102
{ "fragment_index": 0, "new_substring": "CCC&(CC)C(=O)CC&", "old_substring": "C5C4=O" }
Can you make molecule C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1 less soluble in water? The output molecule should be similar to the input molecule.
CC[C@H](C(=O)OC(=O)[C@@H](C)c1cccs1)C(=O)N(C)[C@@H]1CCCc2ccccc21
C[C@H](C(=O)OCC(=O)N(C)[C@@H]1CCCc2ccccc21)c1cccs1
CC[C@H](C(=O)OC(=O)[C@@H](C)c1cccs1)C(=O)N(C)[C@@H]1CCCc2ccccc21
102
{ "fragment_index": 0, "new_substring": "CC[C@H](C&=O)C&=O", "old_substring": "C5C4=O" }
Can you make molecule CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=CC=C3CC3(C)C2)n1
CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=CC=C3CC3(C)C2)n1
102
{ "fragment_index": 0, "new_substring": "CC1&Cc2ccccc2C1", "old_substring": "CC2" }
Can you make molecule CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=NC3=C(CCCC2(C)C)S3)n1
CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=NC3=C(CCCC2(C)C)S3)n1
102
{ "fragment_index": 0, "new_substring": "CC1(C)CCCc2sc&nc21", "old_substring": "CC2" }
Can you make molecule CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=C3C=C3CC(C)(C)O2)n1
CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=C3C=C3CC(C)(C)O2)n1
102
{ "fragment_index": 0, "new_substring": "CC1(C)Cc2cc&ccc2O1", "old_substring": "CC2" }
Can you make molecule CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=C3C=C3CCN2C)n1
CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NC2=CC=C3C=C3CCN2C)n1
102
{ "fragment_index": 0, "new_substring": "CN1CCc2cc&ccc21", "old_substring": "CC2" }
Can you make molecule CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NCCCCC23CC2C3)n1
CCN[C@H]1CCCC[C@@H]1[NH+](C)Cc1cccc(C)n1
Cc1cccc(C[NH+](C)[C@H]2CCCC[C@@H]2NCCCCC23CC2C3)n1
102
{ "fragment_index": 0, "new_substring": "C1&CC2(CCCC2)C1", "old_substring": "CC2" }
Can you make molecule COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COCc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COCc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO3" }
Can you make molecule COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COCSc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COCSc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO3" }
Can you make molecule COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1SC(C)=O
COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1SC(C)=O
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO3" }
Can you make molecule COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1C(=O)CS
COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1C(=O)CS
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO3" }
Can you make molecule COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1C(=O)CI
COc1ccc(C(=O)CCCC2OCC(C)(C)CO2)cc1OC
COc1cc(C(=O)CCCC2OCC(C)(C)CO2)ccc1C(=O)CI
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO3" }
Can you make molecule Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)NNc2cccc(C(F)(F)F)c2)c(Cl)cc1F
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F
Cc1cc(C(=O)NNc2cccc(C(F)(F)F)c2)c(Cl)cc1F
102
{ "fragment_index": 0, "new_substring": "Cc1cc&c(Cl)cc1F", "old_substring": "Cc1ccc3cc1F" }
Can you make molecule Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1Cl
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1Cl
102
{ "fragment_index": 0, "new_substring": "Cc1ccc&cc1Cl", "old_substring": "Cc1ccc3cc1F" }
Can you make molecule Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(F)c(C(=O)NNc2cccc(C(F)(F)F)c2)c1Cl
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F
Cc1ccc(F)c(C(=O)NNc2cccc(C(F)(F)F)c2)c1Cl
102
{ "fragment_index": 0, "new_substring": "Cc1ccc(F)c&c1Cl", "old_substring": "Cc1ccc3cc1F" }
Can you make molecule Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(Br)c(C(=O)NNc2cccc(C(F)(F)F)c2)c1
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F
Cc1ccc(Br)c(C(=O)NNc2cccc(C(F)(F)F)c2)c1
102
{ "fragment_index": 0, "new_substring": "Cc1ccc(Br)c&c1", "old_substring": "Cc1ccc3cc1F" }
Can you make molecule Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(=O)NNc2cccc(C(F)(F)F)c2)c(C)cc1I
Cc1ccc(C(=O)NNc2cccc(C(F)(F)F)c2)cc1F
Cc1cc(C(=O)NNc2cccc(C(F)(F)F)c2)c(C)cc1I
102
{ "fragment_index": 0, "new_substring": "Cc1cc&c(C)cc1I", "old_substring": "Cc1ccc3cc1F" }
Can you make molecule COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)cc1I
COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1
COc1cc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)cc1I
102
{ "fragment_index": 0, "new_substring": "c1&cc&c&cc1I", "old_substring": "c14ccc5c8c1" }
Can you make molecule COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)cc1Cl
COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1
COc1cc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)cc1Cl
102
{ "fragment_index": 0, "new_substring": "c1&cc&c&cc1Cl", "old_substring": "c14ccc5c8c1" }
Can you make molecule COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(I)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)c1
COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1
COc1cc(I)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)c1
102
{ "fragment_index": 0, "new_substring": "c1&cc&cc(I)c1&", "old_substring": "c14ccc5c8c1" }
Can you make molecule COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(Br)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)c1
COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1
COc1cc(Br)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)c1
102
{ "fragment_index": 0, "new_substring": "c1&cc&c&c(Br)c1", "old_substring": "c14ccc5c8c1" }
Can you make molecule COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cc([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)cc1Br
COc1ccc(OC)c([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c1
COc1cc([C@H](c2nnnn2C2CCCC2)N2CCc3ccccc3C2)c(OC)cc1Br
102
{ "fragment_index": 0, "new_substring": "c1&cc(Br)c&cc1&", "old_substring": "c14ccc5c8c1" }
Can you make molecule C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCCN1S(=O)(=O)c1cccc(CC(=O)SN(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(CC(=O)SN(C)c2ccc(F)cc2)c1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C36=O" }
Can you make molecule C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)CCCC(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)CCCC(=O)N(C)c2ccc(F)cc2)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C36=O" }
Can you make molecule C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(C)(C)CC(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(C)(C)CC(=O)N(C)c2ccc(F)cc2)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C36=O" }
Can you make molecule C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(C)(C)CCC(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(C)(C)CCC(=O)N(C)c2ccc(F)cc2)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C36=O" }
Can you make molecule C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](C(=O)SN(C)c1ccc(F)cc1)c1cccc(S(=O)(=O)N2CCCC[C@@H]2C)c1
C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N(C)c2ccc(F)cc2)c1
C[C@H](C(=O)SN(C)c1ccc(F)cc1)c1cccc(S(=O)(=O)N2CCCC[C@@H]2C)c1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)[C@H]&C", "old_substring": "C36=O" }
Can you make molecule C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](O)C[C@H]1CCCN1C(=O)CC(C)(C)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)CC(C)(C)NCC1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C34=O" }
Can you make molecule C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](O)C[C@H]1CCCN1C(=O)CCC(C)(C)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)CCC(C)(C)NCC1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C34=O" }
Can you make molecule C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](O)C[C@H]1CCCN1C(=O)C[C@@H](Br)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)C[C@@H](Br)NCC1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "C&(=O)C[C@H]&Br", "old_substring": "C34=O" }
Can you make molecule C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(N2CCC[C@@H]2C[C@H](C)O)cc(=O)n1NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1
Cc1cc(N2CCC[C@@H]2C[C@H](C)O)cc(=O)n1NCC1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "Cc1cc&cc(=O)n1&", "old_substring": "C34=O" }
Can you make molecule C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1c(N2CCC[C@@H]2C[C@H](C)O)c(=O)ccn1NCC1(C)Cc2ccccc2C1
C[C@H](O)C[C@H]1CCCN1C(=O)NCC1(C)Cc2ccccc2C1
Cc1c(N2CCC[C@@H]2C[C@H](C)O)c(=O)ccn1NCC1(C)Cc2ccccc2C1
102
{ "fragment_index": 0, "new_substring": "Cc1c&c(=O)ccn1&", "old_substring": "C34=O" }
Can you make molecule O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCOCC1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCOCC1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCCOCC1", "old_substring": "[C@H]17CCCO1" }
Can you make molecule O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCc1nnc2ccccn12)NC[C@H]1CSCCS1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CSCCS1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CSCCS1", "old_substring": "[C@H]17CCCO1" }
Can you make molecule O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCc1nnc2ccccn12)NC[C@H]1CC=CS1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CC=CS1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC=CS1", "old_substring": "[C@H]17CCCO1" }
Can you make molecule O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCc1nnc2ccccn12)NC[C@@H]1CCSC1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1
O=C(NCCc1nnc2ccccn12)NC[C@@H]1CCSC1
102
{ "fragment_index": 0, "new_substring": "[C@@H]1&CCSC1", "old_substring": "[C@H]17CCCO1" }
Can you make molecule O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCc1nnc2ccccn12)NC[C@H]1CC12CCOCC2
O=C(NCCc1nnc2ccccn12)NC[C@H]1CCCO1
O=C(NCCc1nnc2ccccn12)NC[C@H]1CC12CCOCC2
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC12CCOCC2", "old_substring": "[C@H]17CCCO1" }
Can you make molecule CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1CCN(SC(=O)Cc2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(SC(=O)Cc2ccccc2NC(=O)NCCc2cccs2)CC1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C38=O" }
Can you make molecule CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1CCN(C(=O)CCCC(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)CCCC(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C38=O" }
Can you make molecule CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1CCN(C(=O)CC(C)(C)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)CC(C)(C)c2ccccc2NC(=O)NCCc2cccs2)CC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C38=O" }
Can you make molecule CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1CCN(C(=O)CCC(C)(C)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)CCC(C)(C)c2ccccc2NC(=O)NCCc2cccs2)CC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C38=O" }
Can you make molecule CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1CCN(SC(=O)[C@@H](C)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(C(=O)c2ccccc2NC(=O)NCCc2cccs2)CC1
CC1CCN(SC(=O)[C@@H](C)c2ccccc2NC(=O)NCCc2cccs2)CC1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)[C@H]&C", "old_substring": "C38=O" }
Can you make molecule CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O less soluble in water? The output molecule should be similar to the input molecule.
CCCCn1c(N)c(N(C)SC(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)SC(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C3(=O)C4" }
Can you make molecule CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O less soluble in water? The output molecule should be similar to the input molecule.
CCCCn1c(N)c(N(C)C(=O)CCCC(=O)Sc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CCCC(=O)Sc2ccc(F)cc2)c(=O)[nH]c1=O
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C3(=O)C4" }
Can you make molecule CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O less soluble in water? The output molecule should be similar to the input molecule.
CCCCn1c(N)c(N(C)C(=O)CC(C)(C)Sc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CC(C)(C)Sc2ccc(F)cc2)c(=O)[nH]c1=O
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C3(=O)C4" }
Can you make molecule CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O less soluble in water? The output molecule should be similar to the input molecule.
CCCCn1c(N)c(N(C)C[S@+]([O-])CCCSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C[S@+]([O-])CCCSc2ccc(F)cc2)c(=O)[nH]c1=O
102
{ "fragment_index": 0, "new_substring": "C&[S@](=O)CCC&", "old_substring": "C3(=O)C4" }
Can you make molecule CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O less soluble in water? The output molecule should be similar to the input molecule.
CCCCn1c(N)c(N(C)C(=O)CCC(C)(C)Sc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CSc2ccc(F)cc2)c(=O)[nH]c1=O
CCCCn1c(N)c(N(C)C(=O)CCC(C)(C)Sc2ccc(F)cc2)c(=O)[nH]c1=O
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C3(=O)C4" }