prompt
stringlengths
120
209
completion
stringlengths
15
103
input_smiles
stringlengths
14
103
output_smiles
stringlengths
15
103
task_id
int64
102
102
winner_action
dict
Can you make molecule O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C([O-])CCC[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])CCC[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
102
{ "fragment_index": 0, "new_substring": "O=C([O-])CCC&", "old_substring": "O=C6[O-]" }
Can you make molecule O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C([O-])CCCCC[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])CCCCC[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
102
{ "fragment_index": 0, "new_substring": "O=C([O-])CCCCC&", "old_substring": "O=C6[O-]" }
Can you make molecule O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C([O-])CCCC(=O)[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])CCCC(=O)[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
102
{ "fragment_index": 0, "new_substring": "O=C([O-])CCCC&=O", "old_substring": "O=C6[O-]" }
Can you make molecule O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1 less soluble in water? The output molecule should be similar to the input molecule.
O=CO[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=CO[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
102
{ "fragment_index": 0, "new_substring": "O=CO&", "old_substring": "O=C6[O-]" }
Can you make molecule O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NO)[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C([O-])[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
O=C(NO)[C@H]1C=C[C@H](NS(=O)(=O)c2ccc3c(c2)CCO3)C1
102
{ "fragment_index": 0, "new_substring": "O=C&NO", "old_substring": "O=C6[O-]" }
Can you make molecule CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)NCC1CCN(C(=O)[C@@H](CC=C(C)C)C(C)(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@@H](CC=C(C)C)C(C)(C)C)CC1
102
{ "fragment_index": 0, "new_substring": "[C@H]&(CC&)C(C)(C)C", "old_substring": "[C@H]16[C@@H](C=7)C1(C)C" }
Can you make molecule CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)NCC1CCN(C(=O)[C@@H](C)CC(C)(C)C=C(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@@H](C)CC(C)(C)C=C(C)C)CC1
102
{ "fragment_index": 0, "new_substring": "[C@H]&(C)CC(C)(C)C&", "old_substring": "[C@H]16[C@@H](C=7)C1(C)C" }
Can you make molecule CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@](C)(C=C(C)C)CC(=O)N1CCC(CNC(C)=O)CC1
CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1
CCC[C@@](C)(C=C(C)C)CC(=O)N1CCC(CNC(C)=O)CC1
102
{ "fragment_index": 0, "new_substring": "CCC[C@](C)(C&)C&", "old_substring": "[C@H]16[C@@H](C=7)C1(C)C" }
Can you make molecule CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)NCC1CCN(C(=O)[C@@H](CBr)CCC=C(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1
CC(=O)NCC1CCN(C(=O)[C@@H](CBr)CCC=C(C)C)CC1
102
{ "fragment_index": 0, "new_substring": "[C@H]&(CBr)CCC&", "old_substring": "[C@H]16[C@@H](C=7)C1(C)C" }
Can you make molecule CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@H](CC=C(C)C)C(=O)N1CCC(CNC(C)=O)CC1
CC(=O)NCC1CCN(C(=O)[C@H]2[C@@H](C=C(C)C)C2(C)C)CC1
CCC[C@@H](CC=C(C)C)C(=O)N1CCC(CNC(C)=O)CC1
102
{ "fragment_index": 0, "new_substring": "CCC[C@H]&CC&", "old_substring": "[C@H]16[C@@H](C=7)C1(C)C" }
Can you make molecule CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CCOSC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOSC(=O)C=CC(=O)N[C@H](C)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C2(=O)C=6" }
Can you make molecule CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=O)C1=C(N=CC(=O)N[C@H](C)c2ccccc2)CCS1
CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOC(=O)C1=C(N=CC(=O)N[C@H](C)c2ccccc2)CCS1
102
{ "fragment_index": 0, "new_substring": "C&(=O)C1=C(N&)CCS1", "old_substring": "C2(=O)C=6" }
Can you make molecule CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=O)C(N=CC(=O)N[C@H](C)c1ccccc1)=C(Cl)Cl
CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOC(=O)C(N=CC(=O)N[C@H](C)c1ccccc1)=C(Cl)Cl
102
{ "fragment_index": 0, "new_substring": "C&(=O)C(N&)=C(Cl)Cl", "old_substring": "C2(=O)C=6" }
Can you make molecule CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=O)C(C=CC(=O)N[C@H](C)c1ccccc1)=C(Cl)Cl
CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOC(=O)C(C=CC(=O)N[C@H](C)c1ccccc1)=C(Cl)Cl
102
{ "fragment_index": 0, "new_substring": "C&(=O)C(C&)=C(Cl)Cl", "old_substring": "C2(=O)C=6" }
Can you make molecule CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC[S@+]([O-])CCC=CC(=O)N[C@H](C)c1ccccc1
CCOC(=O)C=CC(=O)N[C@H](C)c1ccccc1
CCOC[S@+]([O-])CCC=CC(=O)N[C@H](C)c1ccccc1
102
{ "fragment_index": 0, "new_substring": "C&[S@](=O)CCC&", "old_substring": "C2(=O)C=6" }
Can you make molecule Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
Clc1ccc(CCCCOc2ccc(CNn3cnnc3)cc2)cc1
Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1
Clc1ccc(CCCCOc2ccc(CNn3cnnc3)cc2)cc1
102
{ "fragment_index": 0, "new_substring": "C&CCC&", "old_substring": "C46" }
Can you make molecule Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
Clc1ccc(CCCCCOc2ccc(CNn3cnnc3)cc2)cc1
Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1
Clc1ccc(CCCCCOc2ccc(CNn3cnnc3)cc2)cc1
102
{ "fragment_index": 0, "new_substring": "C&CCCC&", "old_substring": "C46" }
Can you make molecule Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
Clc1ccc(C2CC(Oc3ccc(CNn4cnnc4)cc3)C2)cc1
Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1
Clc1ccc(C2CC(Oc3ccc(CNn4cnnc4)cc3)C2)cc1
102
{ "fragment_index": 0, "new_substring": "C1&CC&C1", "old_substring": "C46" }
Can you make molecule Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
S=C(OOc1ccc(CNn2cnnc2)cc1)Sc1ccc(Cl)cc1
Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1
S=C(OOc1ccc(CNn2cnnc2)cc1)Sc1ccc(Cl)cc1
102
{ "fragment_index": 0, "new_substring": "O&C(=S)S&", "old_substring": "C46" }
Can you make molecule Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1 less soluble in water? The output molecule should be similar to the input molecule.
S=C(Nc1ccc(Cl)cc1)SOc1ccc(CNn2cnnc2)cc1
Clc1ccc(COc2ccc(CNn3cnnc3)cc2)cc1
S=C(Nc1ccc(Cl)cc1)SOc1ccc(CNn2cnnc2)cc1
102
{ "fragment_index": 0, "new_substring": "S&C(=S)N&", "old_substring": "C46" }
Can you make molecule CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1nn(C)cc1CNC[C@@H](c1ccc(Br)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(Br)o1)N1CCOCC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Br)o1", "old_substring": "c16ccc(C)o1" }
Can you make molecule CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1nn(C)cc1CNC[C@@H](c1ccc(Cl)s1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(Cl)s1)N1CCOCC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)s1", "old_substring": "c16ccc(C)o1" }
Can you make molecule CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1nn(C)cc1CNC[C@@H](c1cccc(C)c1C)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1cccc(C)c1C)N1CCOCC1
102
{ "fragment_index": 0, "new_substring": "c1&cccc(C)c1C", "old_substring": "c16ccc(C)o1" }
Can you make molecule CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1nn(C)cc1CNC[C@@H](c1cc2cc(C)ccc2o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1cc2cc(C)ccc2o1)N1CCOCC1
102
{ "fragment_index": 0, "new_substring": "c1&cc2cc(C)ccc2o1", "old_substring": "c16ccc(C)o1" }
Can you make molecule CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCc1nn(C)cc1CNC[C@@H](c1cc2cc(Cl)ccc2o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1ccc(C)o1)N1CCOCC1
CCc1nn(C)cc1CNC[C@@H](c1cc2cc(Cl)ccc2o1)N1CCOCC1
102
{ "fragment_index": 0, "new_substring": "c1&cc2cc(Cl)ccc2o1", "old_substring": "c16ccc(C)o1" }
Can you make molecule NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
NC(=O)N1CCC2(CCC(=CC(=O)OCC(=O)Nc3c(Cl)cc(Cl)cc3Cl)CC2)CC1
NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1
NC(=O)N1CCC2(CCC(=CC(=O)OCC(=O)Nc3c(Cl)cc(Cl)cc3Cl)CC2)CC1
102
{ "fragment_index": 0, "new_substring": "N1&CCC2(CCC&CC2)CC1", "old_substring": "c17ccc(C=8)cc1" }
Can you make molecule NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC[C@@H](CC=CC(=O)OCC(=O)Nc1c(Cl)cc(Cl)cc1Cl)C(N)=O
NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1
CCCC[C@@H](CC=CC(=O)OCC(=O)Nc1c(Cl)cc(Cl)cc1Cl)C(N)=O
102
{ "fragment_index": 0, "new_substring": "CCCC[C@H]&CC&", "old_substring": "c17ccc(C=8)cc1" }
Can you make molecule NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@](C)(C=CC(=O)OCC(=O)Nc1c(Cl)cc(Cl)cc1Cl)CC(N)=O
NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1
CCC[C@@](C)(C=CC(=O)OCC(=O)Nc1c(Cl)cc(Cl)cc1Cl)CC(N)=O
102
{ "fragment_index": 0, "new_substring": "CCC[C@](C)(C&)C&", "old_substring": "c17ccc(C=8)cc1" }
Can you make molecule NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
NC(=O)c1ccc(C=CC(=O)OCCC(CO)=Nc2c(Cl)cc(Cl)cc2Cl)cc1
NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1
NC(=O)c1ccc(C=CC(=O)OCCC(CO)=Nc2c(Cl)cc(Cl)cc2Cl)cc1
102
{ "fragment_index": 0, "new_substring": "C&CC=&CO", "old_substring": "C5C4=O" }
Can you make molecule NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
C/C(COC(=O)C=Cc1ccc(C(N)=O)cc1)=N/ONc1c(Cl)cc(Cl)cc1Cl
NC(=O)c1ccc(C=CC(=O)OCC(=O)Nc2c(Cl)cc(Cl)cc2Cl)cc1
C/C(COC(=O)C=Cc1ccc(C(N)=O)cc1)=N/ONc1c(Cl)cc(Cl)cc1Cl
102
{ "fragment_index": 0, "new_substring": "C/C(C&)=N/O&", "old_substring": "C5C4=O" }
Can you make molecule O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2I)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2I)CC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)cc1I", "old_substring": "c18ccc(Cl)cc1" }
Can you make molecule O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2Br)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2Br)CC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)cc1Br", "old_substring": "c18ccc(Cl)cc1" }
Can you make molecule O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)c(I)c2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)c(I)c2)CC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)c(I)c1", "old_substring": "c18ccc(Cl)cc1" }
Can you make molecule O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2cc(Cl)ccc2Cl)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2cc(Cl)ccc2Cl)CC1
102
{ "fragment_index": 0, "new_substring": "Clc1ccc(Cl)c&c1", "old_substring": "c18ccc(Cl)cc1" }
Can you make molecule O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)c(Cl)c2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)cc2)CC1
O=C(NC[C@H]1Cc2cccc(-c3cncnc3)c2O1)C1(c2ccc(Cl)c(Cl)c2)CC1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(Cl)c(Cl)c1", "old_substring": "c18ccc(Cl)cc1" }
Can you make molecule Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C(F)(F)CBr)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)(F)CBr)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
102
{ "fragment_index": 0, "new_substring": "C&(F)(F)CBr", "old_substring": "C7(F)F" }
Can you make molecule Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(SC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(SC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
102
{ "fragment_index": 0, "new_substring": "S&C(F)(F)F", "old_substring": "C7(F)F" }
Can you make molecule Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(CCCC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(CCCC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
102
{ "fragment_index": 0, "new_substring": "C&CCC(F)(F)F", "old_substring": "C7(F)F" }
Can you make molecule Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(CCCCC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(CCCCC(F)(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
102
{ "fragment_index": 0, "new_substring": "C&CCCC(F)(F)F", "old_substring": "C7(F)F" }
Can you make molecule Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(CC(F)(F)C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
Cc1cc(CC(F)(F)C(F)F)n2ncc(C(=O)Nc3ccc(Br)cc3C(F)(F)F)c2n1
102
{ "fragment_index": 0, "new_substring": "C&C(F)(F)C(F)F", "old_substring": "C7(F)F" }
Can you make molecule COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
COc1c(F)cc(NC(=O)CC(C)(C)c2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CC(C)(C)c2cnn(-c3ccccc3)c2)cc1F
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C4(=O)CC7" }
Can you make molecule COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
COc1c(F)cc(NC(=O)CCC(C)(C)c2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCC(C)(C)c2cnn(-c3ccccc3)c2)cc1F
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C4(=O)CC7" }
Can you make molecule COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
COc1c(F)cc(NC(=O)C[C@H](C)c2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)C[C@H](C)c2cnn(-c3ccccc3)c2)cc1F
102
{ "fragment_index": 0, "new_substring": "C&(=O)C[C@@H]&C", "old_substring": "C4(=O)CC7" }
Can you make molecule COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
COc1c(F)cc(NC(=O)C[C@@H](Br)c2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)C[C@@H](Br)c2cnn(-c3ccccc3)c2)cc1F
102
{ "fragment_index": 0, "new_substring": "C&(=O)C[C@H]&Br", "old_substring": "C4(=O)CC7" }
Can you make molecule COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F less soluble in water? The output molecule should be similar to the input molecule.
COc1c(F)cc(NSC(=O)[C@@H](C)c2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NC(=O)CCc2cnn(-c3ccccc3)c2)cc1F
COc1c(F)cc(NSC(=O)[C@@H](C)c2cnn(-c3ccccc3)c2)cc1F
102
{ "fragment_index": 0, "new_substring": "S&C(=O)[C@H]&C", "old_substring": "C4(=O)CC7" }
Can you make molecule O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC[C@@H](CCCS)CN1C(=O)Cc2ccc(Cl)cc21
O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1
CCCC[C@@H](CCCS)CN1C(=O)Cc2ccc(Cl)cc21
102
{ "fragment_index": 0, "new_substring": "CCCC[C@H]&CC&", "old_substring": "C134CCCCC1" }
Can you make molecule O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@](C)(CCS)CCN1C(=O)Cc2ccc(Cl)cc21
O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1
CCC[C@@](C)(CCS)CCN1C(=O)Cc2ccc(Cl)cc21
102
{ "fragment_index": 0, "new_substring": "CCC[C@](C)(C&)C&", "old_substring": "C134CCCCC1" }
Can you make molecule O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1c(C)c(CN2C(=O)Cc3ccc(Cl)cc32)c(C)c(C)c1CS
O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1
Cc1c(C)c(CN2C(=O)Cc3ccc(Cl)cc32)c(C)c(C)c1CS
102
{ "fragment_index": 0, "new_substring": "Cc1c&c(C)c(C)c&c1C", "old_substring": "C134CCCCC1" }
Can you make molecule O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CC1(C)CCc2c(CN3C(=O)Cc4ccc(Cl)cc43)cc(CS)cc21
O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1
CC1(C)CCc2c(CN3C(=O)Cc4ccc(Cl)cc43)cc(CS)cc21
102
{ "fragment_index": 0, "new_substring": "c1&cc&cc2c1CCC2(C)C", "old_substring": "C134CCCCC1" }
Can you make molecule O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(CN2C(=O)Cc3ccc(Cl)cc32)c(Cl)cc1CS
O=C1Cc2ccc(Cl)cc2N1CC1(CS)CCCCC1
Cc1cc(CN2C(=O)Cc3ccc(Cl)cc32)c(Cl)cc1CS
102
{ "fragment_index": 0, "new_substring": "Cc1cc&c(Cl)cc1&", "old_substring": "C134CCCCC1" }
Can you make molecule CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=S)Sc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOC(=S)Sc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
102
{ "fragment_index": 0, "new_substring": "O&C(=S)S&", "old_substring": "O34" }
Can you make molecule CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=N)Cc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOC(=N)Cc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
102
{ "fragment_index": 0, "new_substring": "O&C(=N)C&", "old_substring": "O34" }
Can you make molecule CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2 less soluble in water? The output molecule should be similar to the input molecule.
CCC(=O)CCC(=O)c1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCC(=O)CCC(=O)c1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
102
{ "fragment_index": 0, "new_substring": "O=C&CCC&=O", "old_substring": "O34" }
Can you make molecule CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2 less soluble in water? The output molecule should be similar to the input molecule.
CC[C@H](O)CCc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CC[C@H](O)CCc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
102
{ "fragment_index": 0, "new_substring": "O[C@@H]&CC&", "old_substring": "O34" }
Can you make molecule CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2 less soluble in water? The output molecule should be similar to the input molecule.
CCC(=O)/C=C/Sc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCOc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
CCC(=O)/C=C/Sc1ccc(Cl)cc1S(=O)(=O)Nc1ccc2c(c1)OCCO2
102
{ "fragment_index": 0, "new_substring": "O=C&/C=C/S&", "old_substring": "O34" }
Can you make molecule CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C less soluble in water? The output molecule should be similar to the input molecule.
C=CSOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
C=CSOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
102
{ "fragment_index": 0, "new_substring": "C=CS&", "old_substring": "CC3" }
Can you make molecule CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C less soluble in water? The output molecule should be similar to the input molecule.
C=CCCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
C=CCCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
102
{ "fragment_index": 0, "new_substring": "C=CCC&", "old_substring": "CC3" }
Can you make molecule CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCCl)c(C)c1
CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCCl)c(C)c1
102
{ "fragment_index": 0, "new_substring": "C&CCCl", "old_substring": "CC3" }
Can you make molecule CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCCS)c(C)c1
CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCCS)c(C)c1
102
{ "fragment_index": 0, "new_substring": "C&CCCS", "old_substring": "CC3" }
Can you make molecule CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCBr)c(C)c1
CCOC(=O)c1c(C)[nH]c(C)c1S(=O)(=O)Nc1ccc(C)cc1C
Cc1ccc(NS(=O)(=O)c2c(C)[nH]c(C)c2C(=O)OCCCBr)c(C)c1
102
{ "fragment_index": 0, "new_substring": "C&CCBr", "old_substring": "CC3" }
Can you make molecule C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
C[NH+]1CCN(CCCCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(CCCCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
102
{ "fragment_index": 0, "new_substring": "C&CCCC&", "old_substring": "C4CC5" }
Can you make molecule C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
C[NH+]1CCN(C2CCC(NC(=O)C(=O)c3ccc(Br)cc3)CC2)CC1
C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(C2CCC(NC(=O)C(=O)c3ccc(Br)cc3)CC2)CC1
102
{ "fragment_index": 0, "new_substring": "C1&CCC&CC1", "old_substring": "C4CC5" }
Can you make molecule C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
C[NH+]1CCN(CC(C)(C)CNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(CC(C)(C)CNC(=O)C(=O)c2ccc(Br)cc2)CC1
102
{ "fragment_index": 0, "new_substring": "CC(C)(C&)C&", "old_substring": "C4CC5" }
Can you make molecule C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
C[NH+]1CCN(C2CCC(=NC(=O)C(=O)c3ccc(Br)cc3)CC2)CC1
C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
C[NH+]1CCN(C2CCC(=NC(=O)C(=O)c3ccc(Br)cc3)CC2)CC1
102
{ "fragment_index": 0, "new_substring": "C1&CCC=&CC1", "old_substring": "C4CC5" }
Can you make molecule C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@H](CCNC(=O)C(=O)c1ccc(Br)cc1)N1CC[NH+](C)CC1
C[NH+]1CCN(CCCNC(=O)C(=O)c2ccc(Br)cc2)CC1
CCC[C@@H](CCNC(=O)C(=O)c1ccc(Br)cc1)N1CC[NH+](C)CC1
102
{ "fragment_index": 0, "new_substring": "CCC[C@H]&CC&", "old_substring": "C4CC5" }
Can you make molecule C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](CC(C)(C)c1nccs1)NC(=O)N[C@H](c1ccccc1)c1nccn1C
C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1
C[C@H](CC(C)(C)c1nccs1)NC(=O)N[C@H](c1ccccc1)c1nccn1C
102
{ "fragment_index": 0, "new_substring": "C[C@@H]&CC&(C)C", "old_substring": "C[C@H]46" }
Can you make molecule C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](CCNC(=O)N[C@H](c1ccccc1)c1nccn1C)CC(=O)c1nccs1
C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1
C[C@H](CCNC(=O)N[C@H](c1ccccc1)c1nccn1C)CC(=O)c1nccs1
102
{ "fragment_index": 0, "new_substring": "C[C@H](CC&)CC&=O", "old_substring": "C[C@H]46" }
Can you make molecule C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](Cc1nccs1)[C@H](C)NC(=O)N[C@H](c1ccccc1)c1nccn1C
C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1
C[C@H](Cc1nccs1)[C@H](C)NC(=O)N[C@H](c1ccccc1)c1nccn1C
102
{ "fragment_index": 0, "new_substring": "C[C@H]&[C@H](C)C&", "old_substring": "C[C@H]46" }
Can you make molecule C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H](CCNC(=O)N[C@H](c1ccccc1)c1nccn1C)CC(=O)c1nccs1
C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1
C[C@@H](CCNC(=O)N[C@H](c1ccccc1)c1nccn1C)CC(=O)c1nccs1
102
{ "fragment_index": 0, "new_substring": "C[C@@H](CC&)CC&=O", "old_substring": "C[C@H]46" }
Can you make molecule C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@H](CCc1nccs1)NC(=O)N[C@H](c1ccccc1)c1nccn1C
C[C@H](NC(=O)N[C@H](c1ccccc1)c1nccn1C)c1nccs1
CCC[C@@H](CCc1nccs1)NC(=O)N[C@H](c1ccccc1)c1nccn1C
102
{ "fragment_index": 0, "new_substring": "CCC[C@H]&CC&", "old_substring": "C[C@H]46" }
Can you make molecule COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COCc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COCc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
102
{ "fragment_index": 0, "new_substring": "COC&", "old_substring": "CO4" }
Can you make molecule COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COCSc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COCSc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO4" }
Can you make molecule COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1SC(C)=O
COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1SC(C)=O
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO4" }
Can you make molecule COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1C(=O)CS
COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1C(=O)CS
102
{ "fragment_index": 0, "new_substring": "C&(=O)CS", "old_substring": "CO4" }
Can you make molecule COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC less soluble in water? The output molecule should be similar to the input molecule.
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1C(=O)CI
COc1ccc(-c2noc([C@H]3CCO[C@H]3C)n2)cc1OC
COc1cc(-c2noc([C@H]3CCO[C@H]3C)n2)ccc1C(=O)CI
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO4" }
Can you make molecule Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(Cl)sc2Cl)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(Cl)sc2Cl)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc(Cl)sc1Cl", "old_substring": "c13cc(C)sc1C" }
Can you make molecule Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)c(Br)s2)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)c(Br)s2)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc(C)c(Br)s1", "old_substring": "c13cc(C)sc1C" }
Can you make molecule Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)nc([C@H](C#N)C(=O)c2oc3c(Cl)cccc3c2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2oc3c(Cl)cccc3c2C)n1
102
{ "fragment_index": 0, "new_substring": "c1&oc2c(Cl)cccc2c1C", "old_substring": "c13cc(C)sc1C" }
Can you make molecule Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)nc([C@H](C#N)C(=O)c2ccc(I)c(C)c2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2ccc(I)c(C)c2C)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(I)c(C)c1C", "old_substring": "c13cc(C)sc1C" }
Can you make molecule Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(Br)ccc2Cl)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(C)sc2C)n1
Cc1cc(C)nc([C@H](C#N)C(=O)c2cc(Br)ccc2Cl)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc(Br)ccc1Cl", "old_substring": "c13cc(C)sc1C" }
Can you make molecule CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC[NH+]1CCN(c2ccc(NCCC(CO)=C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NCCC(CO)=C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
102
{ "fragment_index": 0, "new_substring": "C&CC=&CO", "old_substring": "C48=O" }
Can you make molecule CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC[NH+]1CCN(c2ccc(NSC(=O)CC3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NSC(=O)CC3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C48=O" }
Can you make molecule CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC[NH+]1CCN(c2ccc(N=CC(=O)C=C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(N=CC(=O)C=C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
102
{ "fragment_index": 0, "new_substring": "C=&C(=O)C=&", "old_substring": "C48=O" }
Can you make molecule CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC[NH+]1CCN(c2ccc(NCC(=C=O)CC3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NCC(=C=O)CC3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
102
{ "fragment_index": 0, "new_substring": "C&C(=C=O)C&", "old_substring": "C48=O" }
Can you make molecule CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
CC[NH+]1CCN(c2ccc(NC(=O)CCCC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
CC[NH+]1CCN(c2ccc(NC(=O)CCCC(=O)C3C[C@H](C)O[C@@H](C)C3)c(C)c2)CC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C48=O" }
Can you make molecule COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc(CSN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CSN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
102
{ "fragment_index": 0, "new_substring": "S&N1CCN&CC1", "old_substring": "N15CCN6CC1" }
Can you make molecule COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc(CN2CC(c3ccccc3[C@@H](O)c3nccs3)C2)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CN2CC(c3ccccc3[C@@H](O)c3nccs3)C2)c1
102
{ "fragment_index": 0, "new_substring": "N1&CC&C1", "old_substring": "N15CCN6CC1" }
Can you make molecule COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc(CN2CCCN(c3ccccc3[C@@H](O)c3nccs3)C2=O)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CN2CCCN(c3ccccc3[C@@H](O)c3nccs3)C2=O)c1
102
{ "fragment_index": 0, "new_substring": "N1&CCCN&C1=O", "old_substring": "N15CCN6CC1" }
Can you make molecule COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc(CN2CCN=C2Sc2ccccc2[C@@H](O)c2nccs2)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CN2CCN=C2Sc2ccccc2[C@@H](O)c2nccs2)c1
102
{ "fragment_index": 0, "new_substring": "N1&CCN=C1S&", "old_substring": "N15CCN6CC1" }
Can you make molecule COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)C(C)(C)C2)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)CC2)c1
COc1cccc(CN2CCN(c3ccccc3[C@@H](O)c3nccs3)C(C)(C)C2)c1
102
{ "fragment_index": 0, "new_substring": "N1&CCN&C(C)(C)C1", "old_substring": "N15CCN6CC1" }
Can you make molecule CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+] less soluble in water? The output molecule should be similar to the input molecule.
CC1(C)CCCC[C@H]1[NH+]1CC=C(CCCC[NH3+])CC1
CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+]
CC1(C)CCCC[C@H]1[NH+]1CC=C(CCCC[NH3+])CC1
102
{ "fragment_index": 0, "new_substring": "[NH+]1&CC=C(CC&)CC1", "old_substring": "[NH+]12CCCC[C@@H]13" }
Can you make molecule CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+] less soluble in water? The output molecule should be similar to the input molecule.
C[C@H]1CN(CC[NH3+])C[C@@H]1[C@@H]1CCCCC1(C)C
CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+]
C[C@H]1CN(CC[NH3+])C[C@@H]1[C@@H]1CCCCC1(C)C
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CN&C[C@@H]1C", "old_substring": "[NH+]12CCCC[C@@H]13" }
Can you make molecule CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+] less soluble in water? The output molecule should be similar to the input molecule.
CC1(C)CCCC[C@H]1[C@H]1CCC[C@H](CC[NH3+])C1
CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+]
CC1(C)CCCC[C@H]1[C@H]1CCC[C@H](CC[NH3+])C1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCC[C@H]&C1", "old_substring": "[NH+]12CCCC[C@@H]13" }
Can you make molecule CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+] less soluble in water? The output molecule should be similar to the input molecule.
CC1(C)CCCC[C@H]1[C@H]1CCC[C@H](CC[NH3+])CC1
CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+]
CC1(C)CCCC[C@H]1[C@H]1CCC[C@H](CC[NH3+])CC1
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCC[C@H]&CC1", "old_substring": "[NH+]12CCCC[C@@H]13" }
Can you make molecule CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+] less soluble in water? The output molecule should be similar to the input molecule.
CC1(C)CCCC[C@H]1[C@@H]1NC[C@@H](CC[NH3+])S1
CC1(C)CCCC[C@H]1[NH+]1CCCC[C@@H]1CC[NH3+]
CC1(C)CCCC[C@H]1[C@@H]1NC[C@@H](CC[NH3+])S1
102
{ "fragment_index": 0, "new_substring": "[C@@H]1&NC[C@@H]&S1", "old_substring": "[NH+]12CCCC[C@@H]13" }
Can you make molecule CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC less soluble in water? The output molecule should be similar to the input molecule.
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CCCC2(C)C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CCCC2(C)C)ccc1OC
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCCC1(C)C", "old_substring": "[C@H]18N=C(C)C=C1C" }
Can you make molecule CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC less soluble in water? The output molecule should be similar to the input molecule.
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CC=CC=C2Cl)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CC=CC=C2Cl)ccc1OC
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC=CC=C1Cl", "old_substring": "[C@H]18N=C(C)C=C1C" }
Can you make molecule CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC less soluble in water? The output molecule should be similar to the input molecule.
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CCC=CCCC2)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CCC=CCCC2)ccc1OC
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CCC=CCCC1", "old_substring": "[C@H]18N=C(C)C=C1C" }
Can you make molecule CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC less soluble in water? The output molecule should be similar to the input molecule.
CCCCC(=O)Nc1cc(NC(=O)[C@@H](CCl)C(C)C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@@H](CCl)C(C)C)ccc1OC
102
{ "fragment_index": 0, "new_substring": "[C@H]&(CCl)C(C)C", "old_substring": "[C@H]18N=C(C)C=C1C" }
Can you make molecule CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC less soluble in water? The output molecule should be similar to the input molecule.
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CC23CCCC3)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2N=C(C)C=C2C)ccc1OC
CCCCC(=O)Nc1cc(NC(=O)[C@H]2CC23CCCC3)ccc1OC
102
{ "fragment_index": 0, "new_substring": "[C@H]1&CC12CCCC2", "old_substring": "[C@H]18N=C(C)C=C1C" }