prompt
stringlengths
120
209
completion
stringlengths
15
103
input_smiles
stringlengths
14
103
output_smiles
stringlengths
15
103
task_id
int64
102
102
winner_action
dict
Can you make molecule CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(O)c(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c2onc1-2
CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O
CCc1ccc(O)c(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c2onc1-2
102
{ "fragment_index": 0, "new_substring": "Oc1ccc2c&noc2c1&", "old_substring": "O23" }
Can you make molecule CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O less soluble in water? The output molecule should be similar to the input molecule.
CCN1CCOc2ccc(CCS(=O)(=O)[N-]c3cc(Br)ccc3O)cc2C1
CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O
CCN1CCOc2ccc(CCS(=O)(=O)[N-]c3cc(Br)ccc3O)cc2C1
102
{ "fragment_index": 0, "new_substring": "N1&CCOc2ccc&cc2C1", "old_substring": "O23" }
Can you make molecule CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O less soluble in water? The output molecule should be similar to the input molecule.
CCc1cc2ccc-2ncn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O
CCc1cc2ccc-2ncn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cc&ccc2ncn1&", "old_substring": "O23" }
Can you make molecule CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc2nc-2ccn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O
CCc1ccc2nc-2ccn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2ccc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O less soluble in water? The output molecule should be similar to the input molecule.
CCc1cnc2nc-2ccn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
CCOCCS(=O)(=O)[N-]c1cc(Br)ccc1O
CCc1cnc2nc-2ccn(CCS(=O)(=O)[N-]c2cc(Br)ccc2O)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cnc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1 less soluble in water? The output molecule should be similar to the input molecule.
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3Cl)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3Cl)C2)S1
102
{ "fragment_index": 0, "new_substring": "c1&ccccc1Cl", "old_substring": "c16ccccc1" }
Can you make molecule NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1 less soluble in water? The output molecule should be similar to the input molecule.
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccc(I)cc3)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccc(I)cc3)C2)S1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(I)cc1", "old_substring": "c16ccccc1" }
Can you make molecule NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc([C@H]2CCN(C(=O)C[C@@H]3SC(N)=NC3=O)C2)cc1I
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1
Cc1ccc([C@H]2CCN(C(=O)C[C@@H]3SC(N)=NC3=O)C2)cc1I
102
{ "fragment_index": 0, "new_substring": "Cc1ccc&cc1I", "old_substring": "c16ccccc1" }
Can you make molecule NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1 less soluble in water? The output molecule should be similar to the input molecule.
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3cccc(Br)c3)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3cccc(Br)c3)C2)S1
102
{ "fragment_index": 0, "new_substring": "Brc1cccc&c1", "old_substring": "c16ccccc1" }
Can you make molecule NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cccc([C@H]2CCN(C(=O)C[C@@H]3SC(N)=NC3=O)C2)c1C
NC1=NC(=O)[C@H](CC(=O)N2CC[C@H](c3ccccc3)C2)S1
Cc1cccc([C@H]2CCN(C(=O)C[C@@H]3SC(N)=NC3=O)C2)c1C
102
{ "fragment_index": 0, "new_substring": "c1&cccc(C)c1C", "old_substring": "c16ccccc1" }
Can you make molecule Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3Cl)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3Cl)C2)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(F)cc1Cl", "old_substring": "c16ccc(F)cc1" }
Can you make molecule Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3Br)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3Br)C2)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(F)cc1Br", "old_substring": "c16ccc(F)cc1" }
Can you make molecule Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)c(Cl)c3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)c(Cl)c3)C2)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(F)c(Cl)c1", "old_substring": "c16ccc(F)cc1" }
Can you make molecule Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(I)cc3F)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(I)cc3F)C2)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(I)cc1F", "old_substring": "c16ccc(F)cc1" }
Can you make molecule Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3cc4c(F)cccc4s3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3ccc(F)cc3)C2)n1
Cc1noc(-c2cccnc2N2CC[C@H](NC(=O)COc3cc4c(F)cccc4s3)C2)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc2c(F)cccc2s1", "old_substring": "c16ccc(F)cc1" }
Can you make molecule Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OC(=O)c2cc(I)cc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cc(I)cc(C(=O)Oc3ccc(C)cn3)n2)nc1
102
{ "fragment_index": 0, "new_substring": "c1&cc(I)cc&n1", "old_substring": "c18cccc9n1" }
Can you make molecule Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OC(=O)c2cc(Cl)nc(C(=O)Oc3ccc(C)cn3)c2)nc1
Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cc(Cl)nc(C(=O)Oc3ccc(C)cn3)c2)nc1
102
{ "fragment_index": 0, "new_substring": "c1&cc&cc(Cl)n1", "old_substring": "c18cccc9n1" }
Can you make molecule Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OC(=O)c2cc(Cl)cc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cc(Cl)cc(C(=O)Oc3ccc(C)cn3)n2)nc1
102
{ "fragment_index": 0, "new_substring": "c1&cc(Cl)cc&n1", "old_substring": "c18cccc9n1" }
Can you make molecule Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OC(=O)c2cnc(C(=O)Oc3ccc(C)cn3)c(Cl)c2)nc1
Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cnc(C(=O)Oc3ccc(C)cn3)c(Cl)c2)nc1
102
{ "fragment_index": 0, "new_substring": "c1&ncc&cc1Cl", "old_substring": "c18cccc9n1" }
Can you make molecule Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1ccc(OC(=O)c2cccn(C(=O)Oc3ccc(C)cn3)c2=O)nc1
Cc1ccc(OC(=O)c2cccc(C(=O)Oc3ccc(C)cn3)n2)nc1
Cc1ccc(OC(=O)c2cccn(C(=O)Oc3ccc(C)cn3)c2=O)nc1
102
{ "fragment_index": 0, "new_substring": "c1&cccn&c1=O", "old_substring": "c18cccc9n1" }
Can you make molecule CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CN(C=C1CCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(C=C1CCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
102
{ "fragment_index": 0, "new_substring": "C1=&CCCCC1", "old_substring": "C16CCCC1" }
Can you make molecule CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CN(CC1CCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
102
{ "fragment_index": 0, "new_substring": "C1&CCCCCC1", "old_substring": "C16CCCC1" }
Can you make molecule CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CN(CC1CCCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
102
{ "fragment_index": 0, "new_substring": "C1&CCCCCCC1", "old_substring": "C16CCCC1" }
Can you make molecule CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CN(CSC1=CCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CSC1=CCCCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
102
{ "fragment_index": 0, "new_substring": "C1=C(S&)CCCCC1", "old_substring": "C16CCCC1" }
Can you make molecule CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1 less soluble in water? The output molecule should be similar to the input molecule.
CN(C=CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
CN(C=CC1CCCC1)C(=O)C(=O)Nc1cccc(SC(F)F)c1
102
{ "fragment_index": 0, "new_substring": "C=&C1CCCC1", "old_substring": "C16CCCC1" }
Can you make molecule COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccnc1SC1=NCCN1C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1SC1=NCCN1C(=O)C[C@H](C)Cc1ccc(Cl)cc1
102
{ "fragment_index": 0, "new_substring": "N1&CCN=C1S&", "old_substring": "N24C" }
Can you make molecule COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccnc1-c1oc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)nc1C#N
COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1-c1oc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)nc1C#N
102
{ "fragment_index": 0, "new_substring": "N#Cc1nc&oc1&", "old_substring": "N24C" }
Can you make molecule COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccnc1-c1sc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)cc1C#N
COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1-c1sc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)cc1C#N
102
{ "fragment_index": 0, "new_substring": "N#Cc1cc&sc1&", "old_substring": "N24C" }
Can you make molecule COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccnc1-c1ccc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)cc1C#N
COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1-c1ccc(C(=O)C[C@H](C)Cc2ccc(Cl)cc2)cc1C#N
102
{ "fragment_index": 0, "new_substring": "N#Cc1cc&ccc1&", "old_substring": "N24C" }
Can you make molecule COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1 less soluble in water? The output molecule should be similar to the input molecule.
COc1cccnc1N1CCC(=NOC(=O)C[C@H](C)Cc2ccc(Cl)cc2)CC1
COc1cccnc1N(C)C(=O)C[C@H](C)Cc1ccc(Cl)cc1
COc1cccnc1N1CCC(=NOC(=O)C[C@H](C)Cc2ccc(Cl)cc2)CC1
102
{ "fragment_index": 0, "new_substring": "O&N=C1CCN&CC1", "old_substring": "N24C" }
Can you make molecule O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(/C=C/Sc1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=C(/C=C/Sc1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
102
{ "fragment_index": 0, "new_substring": "O=C&/C=C/S&", "old_substring": "O=C34" }
Can you make molecule O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=Cc1sc(N2CCC([C@H](O)c3ccccc3)CC2)nc1-c1cc(=O)[nH]c2ccccc12
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=Cc1sc(N2CCC([C@H](O)c3ccccc3)CC2)nc1-c1cc(=O)[nH]c2ccccc12
102
{ "fragment_index": 0, "new_substring": "O=Cc1sc&nc1&", "old_substring": "O=C34" }
Can you make molecule O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=Cc1nc(N2CCC([C@H](O)c3ccccc3)CC2)sc1-c1cc(=O)[nH]c2ccccc12
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=Cc1nc(N2CCC([C@H](O)c3ccccc3)CC2)sc1-c1cc(=O)[nH]c2ccccc12
102
{ "fragment_index": 0, "new_substring": "O=Cc1nc&sc1&", "old_substring": "O=C34" }
Can you make molecule O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(N1CCC([C@H](O)c2ccccc2)CC1)n1nc(-c2cc(=O)[nH]c3ccccc23)oc1=S
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=C(N1CCC([C@H](O)c2ccccc2)CC1)n1nc(-c2cc(=O)[nH]c3ccccc23)oc1=S
102
{ "fragment_index": 0, "new_substring": "O=C&n1nc&oc1=S", "old_substring": "O=C34" }
Can you make molecule O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1 less soluble in water? The output molecule should be similar to the input molecule.
O=c1cc(-c2ccc(/C=N/ON3CCC([C@H](O)c4ccccc4)CC3)o2)c2ccccc2[nH]1
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC([C@H](O)c2ccccc2)CC1
O=c1cc(-c2ccc(/C=N/ON3CCC([C@H](O)c4ccccc4)CC3)o2)c2ccccc2[nH]1
102
{ "fragment_index": 0, "new_substring": "O&/N=C/c1ccc&o1", "old_substring": "O=C34" }
Can you make molecule CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc(O)c([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c2onc1-2
CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F
CCc1ccc(O)c([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c2onc1-2
102
{ "fragment_index": 0, "new_substring": "Oc1ccc2c&noc2c1&", "old_substring": "O23" }
Can you make molecule CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F less soluble in water? The output molecule should be similar to the input molecule.
CCN1CCOc2ccc([C@@H]3C[C@@H]([NH3+])[C@@H]3Nc3ncc(Cl)cc3F)cc2C1
CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F
CCN1CCOc2ccc([C@@H]3C[C@@H]([NH3+])[C@@H]3Nc3ncc(Cl)cc3F)cc2C1
102
{ "fragment_index": 0, "new_substring": "N1&CCOc2ccc&cc2C1", "old_substring": "O23" }
Can you make molecule CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F less soluble in water? The output molecule should be similar to the input molecule.
CCc1cc2ccc-2ncn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F
CCc1cc2ccc-2ncn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cc&ccc2ncn1&", "old_substring": "O23" }
Can you make molecule CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F less soluble in water? The output molecule should be similar to the input molecule.
CCc1ccc2nc-2ccn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F
CCc1ccc2nc-2ccn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2ccc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F less soluble in water? The output molecule should be similar to the input molecule.
CCc1cnc2nc-2ccn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
CCO[C@@H]1C[C@@H]([NH3+])[C@@H]1Nc1ncc(Cl)cc1F
CCc1cnc2nc-2ccn([C@@H]2C[C@@H]([NH3+])[C@@H]2Nc2ncc(Cl)cc2F)c1=O
102
{ "fragment_index": 0, "new_substring": "O=c1c2cnc&nc2ccn1&", "old_substring": "O23" }
Can you make molecule CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Nc1ccc(NSC(=O)Cc2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NSC(=O)Cc2ccc3c(c2)Cc2ccccc2-3)cc1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C58=O" }
Can you make molecule CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Nc1ccc(NC(=O)CCCC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)CCCC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C58=O" }
Can you make molecule CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Nc1ccc(NC(=O)CC(C)(C)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)CC(C)(C)c2ccc3c(c2)Cc2ccccc2-3)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C58=O" }
Can you make molecule CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Nc1ccc(NC(=O)CCC(C)(C)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)CCC(C)(C)c2ccc3c(c2)Cc2ccccc2-3)cc1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C58=O" }
Can you make molecule CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)Nc1ccc(NSC(=O)[C@@H](C)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NC(=O)c2ccc3c(c2)Cc2ccccc2-3)cc1
CC(=O)Nc1ccc(NSC(=O)[C@@H](C)c2ccc3c(c2)Cc2ccccc2-3)cc1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)[C@H]&C", "old_substring": "C58=O" }
Can you make molecule COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1 less soluble in water? The output molecule should be similar to the input molecule.
COCSCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
COCSCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
102
{ "fragment_index": 0, "new_substring": "COCS&", "old_substring": "CO3" }
Can you make molecule COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1 less soluble in water? The output molecule should be similar to the input molecule.
CC(=O)SCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
CC(=O)SCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
102
{ "fragment_index": 0, "new_substring": "CC(=O)S&", "old_substring": "CO3" }
Can you make molecule COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H]1CC([NH+]2CC[C@H](COCCC(=O)CI)C2)C[C@@H](C)O1
COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
C[C@@H]1CC([NH+]2CC[C@H](COCCC(=O)CI)C2)C[C@@H](C)O1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CI", "old_substring": "CO3" }
Can you make molecule COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H]1CC([NH+]2CC[C@H](COCCC3OCCCO3)C2)C[C@@H](C)O1
COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
C[C@@H]1CC([NH+]2CC[C@H](COCCC3OCCCO3)C2)C[C@@H](C)O1
102
{ "fragment_index": 0, "new_substring": "C1&OCCCO1", "old_substring": "CO3" }
Can you make molecule COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H]1CC([NH+]2CC[C@H](COCCC(=O)CCl)C2)C[C@@H](C)O1
COCCOC[C@H]1CC[NH+](C2C[C@@H](C)O[C@H](C)C2)C1
C[C@@H]1CC([NH+]2CC[C@H](COCCC(=O)CCl)C2)C[C@@H](C)O1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCl", "old_substring": "CO3" }
Can you make molecule O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(Cl)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(Cl)c1
102
{ "fragment_index": 0, "new_substring": "C=&c1cccc(Cl)c1", "old_substring": "C=4c1cccc(F)c1" }
Can you make molecule O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(Br)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(Br)c1
102
{ "fragment_index": 0, "new_substring": "C=&c1cccc(Br)c1", "old_substring": "C=4c1cccc(F)c1" }
Can you make molecule O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(F)cc1Br
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(F)cc1Br
102
{ "fragment_index": 0, "new_substring": "C=&c1ccc(F)cc1Br", "old_substring": "C=4c1cccc(F)c1" }
Can you make molecule O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(Cl)cc1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(Cl)cc1
102
{ "fragment_index": 0, "new_substring": "C=&c1ccc(Cl)cc1", "old_substring": "C=4c1cccc(F)c1" }
Can you make molecule O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(Br)cc1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1cccc(F)c1
O=C1OC(c2ccccc2OC(F)F)=NC1=Cc1ccc(Br)cc1
102
{ "fragment_index": 0, "new_substring": "C=&c1ccc(Br)cc1", "old_substring": "C=4c1cccc(F)c1" }
Can you make molecule COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1CNSC(=O)Cc1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNSC(=O)Cc1cc2sccc2n1Cc1cccc(F)c1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C36=O" }
Can you make molecule COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1CNC(=O)CCCC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)CCCC(=O)c1cc2sccc2n1Cc1cccc(F)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C36=O" }
Can you make molecule COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1CNC(=O)CC(C)(C)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)CC(C)(C)c1cc2sccc2n1Cc1cccc(F)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C36=O" }
Can you make molecule COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1CNC(=O)CCC(C)(C)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)CCC(C)(C)c1cc2sccc2n1Cc1cccc(F)c1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCC&(C)C", "old_substring": "C36=O" }
Can you make molecule COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1CNSC(=O)[C@@H](C)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNC(=O)c1cc2sccc2n1Cc1cccc(F)c1
COc1ccccc1CNSC(=O)[C@@H](C)c1cc2sccc2n1Cc1cccc(F)c1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)[C@H]&C", "old_substring": "C36=O" }
Can you make molecule CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCOSC(=O)CC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOSC(=O)CC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
102
{ "fragment_index": 0, "new_substring": "S&C(=O)C&", "old_substring": "C48=O" }
Can you make molecule CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCOCC(=C=O)CC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOCC(=C=O)CC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
102
{ "fragment_index": 0, "new_substring": "C&C(=C=O)C&", "old_substring": "C48=O" }
Can you make molecule CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=O)CCCC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)CCCC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CCCC&=O", "old_substring": "C48=O" }
Can you make molecule CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC(=O)CC(C)(C)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)CC(C)(C)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CC&(C)C", "old_substring": "C48=O" }
Can you make molecule CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1 less soluble in water? The output molecule should be similar to the input molecule.
CCOC[S@+]([O-])CCCC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC(=O)C1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
CCOC[S@+]([O-])CCCC1(NCc2nnc(-c3cc(C)oc3C)o2)CCCC1
102
{ "fragment_index": 0, "new_substring": "C&[S@](=O)CCC&", "old_substring": "C48=O" }
Can you make molecule N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
N#Cc1cccc(NC(=O)N2CCCc3cc(NC(=O)CC4CCCC4)ccc3C2)c1
N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)N2CCCc3cc(NC(=O)CC4CCCC4)ccc3C2)c1
102
{ "fragment_index": 0, "new_substring": "N1&CCCc2cc&ccc2C1", "old_substring": "N15CCC8CC1" }
Can you make molecule N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
N#Cc1cccc(NC(=O)C2CCC(NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)C2CCC(NC(=O)CC3CCCC3)CC2)c1
102
{ "fragment_index": 0, "new_substring": "C1&CCC&CC1", "old_substring": "N15CCC8CC1" }
Can you make molecule N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
N#Cc1cccc(NC(=O)CCCCCNC(=O)CC2CCCC2)c1
N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)CCCCCNC(=O)CC2CCCC2)c1
102
{ "fragment_index": 0, "new_substring": "C&CCCC&", "old_substring": "N15CCC8CC1" }
Can you make molecule N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
N#Cc1cccc(NC(=O)C2CCC(=NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1
N#Cc1cccc(NC(=O)C2CCC(=NC(=O)CC3CCCC3)CC2)c1
102
{ "fragment_index": 0, "new_substring": "C1&CCC=&CC1", "old_substring": "N15CCC8CC1" }
Can you make molecule N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1 less soluble in water? The output molecule should be similar to the input molecule.
CC1(NC(=O)CC2CCCC2)CCC(C(=O)Nc2cccc(C#N)c2)CC1
N#Cc1cccc(NC(=O)N2CCC(NC(=O)CC3CCCC3)CC2)c1
CC1(NC(=O)CC2CCCC2)CCC(C(=O)Nc2cccc(C#N)c2)CC1
102
{ "fragment_index": 0, "new_substring": "C1&CCC&(C)CC1", "old_substring": "N15CCC8CC1" }
Can you make molecule CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCSC(=S)OC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCSC(=S)OC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
102
{ "fragment_index": 0, "new_substring": "O&C(=S)S&", "old_substring": "O34" }
Can you make molecule CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC(=N)OC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCCC(=N)OC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
102
{ "fragment_index": 0, "new_substring": "O&C(=N)C&", "old_substring": "O34" }
Can you make molecule CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCCC[C@@H](O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCCC[C@@H](O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
102
{ "fragment_index": 0, "new_substring": "O[C@@H]&CC&", "old_substring": "O34" }
Can you make molecule CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCS/C=C/C(=O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCS/C=C/C(=O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
102
{ "fragment_index": 0, "new_substring": "O=C&/C=C/S&", "old_substring": "O34" }
Can you make molecule CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1 less soluble in water? The output molecule should be similar to the input molecule.
CCCCC[C@@H](O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCOC(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
CCCCC[C@@H](O)C(=O)C1=C(c2ccccc2)Nc2ncnn2[C@H]1c1ccc(SC)cc1
102
{ "fragment_index": 0, "new_substring": "O[C@@H]&CCC&", "old_substring": "O34" }
Can you make molecule Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccc(I)cc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccc(I)cc2F)n(C)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(I)cc1F", "old_substring": "c17ccccc1F" }
Can you make molecule Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2cc(I)ccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2cc(I)ccc2F)n(C)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc(I)ccc1F", "old_substring": "c17ccccc1F" }
Can you make molecule Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2Cl)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2Cl)n(C)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccccc1Cl", "old_substring": "c17ccccc1F" }
Can you make molecule Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2cc(F)ccc2Br)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2cc(F)ccc2Br)n(C)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc(F)ccc1Br", "old_substring": "c17ccccc1F" }
Can you make molecule Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccc(F)cc2Cl)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccccc2F)n(C)n1
Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)c2ccc(F)cc2Cl)n(C)n1
102
{ "fragment_index": 0, "new_substring": "c1&ccc(F)cc1Cl", "old_substring": "c17ccccc1F" }
Can you make molecule C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](SCSc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](SCSc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
102
{ "fragment_index": 0, "new_substring": "S&CS&", "old_substring": "S57" }
Can you make molecule C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H](C(=O)NC[C@H]1COc2ccccc2O1)N1CCSc2ccc(-c3cccc[n+]3[O-])cc21
C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@@H](C(=O)NC[C@H]1COc2ccccc2O1)N1CCSc2ccc(-c3cccc[n+]3[O-])cc21
102
{ "fragment_index": 0, "new_substring": "N1&CCSc2ccc&cc21", "old_substring": "S57" }
Can you make molecule C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](C[S@@+]([O-])C(Cl)(Cl)c1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](C[S@@+]([O-])C(Cl)(Cl)c1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
102
{ "fragment_index": 0, "new_substring": "O=[S@](C&)C&(Cl)Cl", "old_substring": "S57" }
Can you make molecule C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@H](S/C(Cl)=C(\C#N)Nc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@H](S/C(Cl)=C(\C#N)Nc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
102
{ "fragment_index": 0, "new_substring": "S&/C(Cl)=C(\\C#N)N&", "old_substring": "S57" }
Can you make molecule C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1 less soluble in water? The output molecule should be similar to the input molecule.
C[C@@H](C(=O)NC[C@H]1COc2ccccc2O1)n1c(=S)n(-c2cccc[n+]2[O-])c2ccccc21
C[C@H](Sc1cccc[n+]1[O-])C(=O)NC[C@H]1COc2ccccc2O1
C[C@@H](C(=O)NC[C@H]1COc2ccccc2O1)n1c(=S)n(-c2cccc[n+]2[O-])c2ccccc21
102
{ "fragment_index": 0, "new_substring": "n1&c(=S)n&c2ccccc21", "old_substring": "S57" }
Can you make molecule O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCOc1ccc2c(c1)OCO2)c1ccc(C2CC2)o1
O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1
O=C(NCCOc1ccc2c(c1)OCO2)c1ccc(C2CC2)o1
102
{ "fragment_index": 0, "new_substring": "c1&ccc&o1", "old_substring": "c17cc8on1" }
Can you make molecule O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1oc(C2CC2)cc1C(=O)NCCOc1ccc2c(c1)OCO2
O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1
Cc1oc(C2CC2)cc1C(=O)NCCOc1ccc2c(c1)OCO2
102
{ "fragment_index": 0, "new_substring": "c1&cc&oc1C", "old_substring": "c17cc8on1" }
Can you make molecule O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCOc1ccc2c(c1)OCO2)c1ccc2oc(C3CC3)nc2c1
O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1
O=C(NCCOc1ccc2c(c1)OCO2)c1ccc2oc(C3CC3)nc2c1
102
{ "fragment_index": 0, "new_substring": "c1&ccc2oc&nc2c1", "old_substring": "c17cc8on1" }
Can you make molecule O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1 less soluble in water? The output molecule should be similar to the input molecule.
O=C(NCCOc1ccc2c(c1)OCO2)c1cc2occc2c(C2CC2)n1
O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1
O=C(NCCOc1ccc2c(c1)OCO2)c1cc2occc2c(C2CC2)n1
102
{ "fragment_index": 0, "new_substring": "c1&cc2occc2c&n1", "old_substring": "c17cc8on1" }
Can you make molecule O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1 less soluble in water? The output molecule should be similar to the input molecule.
Cc1nc(C2CC2)ccc1C(=O)NCCOc1ccc2c(c1)OCO2
O=C(NCCOc1ccc2c(c1)OCO2)c1cc(C2CC2)on1
Cc1nc(C2CC2)ccc1C(=O)NCCOc1ccc2c(c1)OCO2
102
{ "fragment_index": 0, "new_substring": "c1&ccc&nc1C", "old_substring": "c17cc8on1" }
Can you make molecule N#CCC[NH2+]C1(C(=O)[O-])CC1 less soluble in water? The output molecule should be similar to the input molecule.
N#CCC[NH2+]C1(CCS(=O)(=O)[O-])CC1
N#CCC[NH2+]C1(C(=O)[O-])CC1
N#CCC[NH2+]C1(CCS(=O)(=O)[O-])CC1
102
{ "fragment_index": 0, "new_substring": "C&CS(=O)(=O)[O-]", "old_substring": "C4(=O)[O-]" }
Can you make molecule N#CCC[NH2+]C1(C(=O)[O-])CC1 less soluble in water? The output molecule should be similar to the input molecule.
N#CCC[NH2+]C1(C(=O)CO)CC1
N#CCC[NH2+]C1(C(=O)[O-])CC1
N#CCC[NH2+]C1(C(=O)CO)CC1
102
{ "fragment_index": 0, "new_substring": "C&(=O)CO", "old_substring": "C4(=O)[O-]" }
Can you make molecule N#CCC[NH2+]C1(C(=O)[O-])CC1 less soluble in water? The output molecule should be similar to the input molecule.
N#CCC[NH2+]C1(C(O)O)CC1
N#CCC[NH2+]C1(C(=O)[O-])CC1
N#CCC[NH2+]C1(C(O)O)CC1
102
{ "fragment_index": 0, "new_substring": "C&(O)O", "old_substring": "C4(=O)[O-]" }
Can you make molecule N#CCC[NH2+]C1(C(=O)[O-])CC1 less soluble in water? The output molecule should be similar to the input molecule.
N#CCC[NH2+]C1(C(F)(F)C(=O)[O-])CC1
N#CCC[NH2+]C1(C(=O)[O-])CC1
N#CCC[NH2+]C1(C(F)(F)C(=O)[O-])CC1
102
{ "fragment_index": 0, "new_substring": "C&(F)(F)C(=O)[O-]", "old_substring": "C4(=O)[O-]" }
Can you make molecule N#CCC[NH2+]C1(C(=O)[O-])CC1 less soluble in water? The output molecule should be similar to the input molecule.
CCC(CC)(C(=O)[O-])C1([NH2+]CCC#N)CC1
N#CCC[NH2+]C1(C(=O)[O-])CC1
CCC(CC)(C(=O)[O-])C1([NH2+]CCC#N)CC1
102
{ "fragment_index": 0, "new_substring": "CCC&(CC)C(=O)[O-]", "old_substring": "C4(=O)[O-]" }
Can you make molecule CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1 less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@](C)(CC(=O)NCc1ccccn1)Oc1ccccc1OC
CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1
CC[C@@](C)(CC(=O)NCc1ccccn1)Oc1ccccc1OC
102
{ "fragment_index": 0, "new_substring": "CC[C@@]&(C)CC&=O", "old_substring": "CC[C@@H]3C2=O" }
Can you make molecule CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1 less soluble in water? The output molecule should be similar to the input molecule.
COc1ccccc1OCC[C@H](Cl)NCc1ccccn1
CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1
COc1ccccc1OCC[C@H](Cl)NCc1ccccn1
102
{ "fragment_index": 0, "new_substring": "C&C[C@@H]&Cl", "old_substring": "CC[C@@H]3C2=O" }
Can you make molecule CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1 less soluble in water? The output molecule should be similar to the input molecule.
CC[C@@](C)(C#CCNCc1ccccn1)Oc1ccccc1OC
CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1
CC[C@@](C)(C#CCNCc1ccccn1)Oc1ccccc1OC
102
{ "fragment_index": 0, "new_substring": "CC[C@@]&(C)C#CC&", "old_substring": "CC[C@@H]3C2=O" }
Can you make molecule CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@H](CC(=O)NCc1ccccn1)Oc1ccccc1OC
CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1
CCC[C@H](CC(=O)NCc1ccccn1)Oc1ccccc1OC
102
{ "fragment_index": 0, "new_substring": "CCC[C@@H]&CC&=O", "old_substring": "CC[C@@H]3C2=O" }
Can you make molecule CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1 less soluble in water? The output molecule should be similar to the input molecule.
CCC[C@@H](CC(=O)NCc1ccccn1)Oc1ccccc1OC
CC[C@@H](Oc1ccccc1OC)C(=O)NCc1ccccn1
CCC[C@@H](CC(=O)NCc1ccccn1)Oc1ccccc1OC
102
{ "fragment_index": 0, "new_substring": "CCC[C@H]&CC&=O", "old_substring": "CC[C@@H]3C2=O" }